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Results: 1-18 |
Results: 18
Cycloaddition reactions of thiazolidine derivatives. An approach to the synthesis of new functionalized heterocyclic systems
Authors: Gomez-Monterrey, IM Campiglia, P Mazzoni, O Novellino, E Diurno, MV
Citation: Im. Gomez-monterrey et al., Cycloaddition reactions of thiazolidine derivatives. An approach to the synthesis of new functionalized heterocyclic systems, TETRAHEDR L, 42(33), 2001, pp. 5755-5757
Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent
Authors: Campiani, G Aiello, F Fabbrini, M Morelli, E Ramunno, A Armaroli, S Nacci, V Garofalo, A Greco, G Novellino, E Maga, G Spadari, S Bergamini, A Ventura, L Bongiovanni, B Capozzi, M Bolacchi, F Marini, S Coletta, M Guiso, G Caccia, S
Citation: G. Campiani et al., Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent, J MED CHEM, 44(3), 2001, pp. 305-315
3-aryl[1,2,4]triazino[4,3-alpha]benzimidazol-4(10H)-ones: A new class of selective A(1) adenosine receptor antagonists
Authors: Da Settimo, F Primofiore, G Taliani, S Marini, AM La Motta, C Novellino, E Greco, G Lavecchia, A Trincavelli, L Martini, C
Citation: F. Da Settimo et al., 3-aryl[1,2,4]triazino[4,3-alpha]benzimidazol-4(10H)-ones: A new class of selective A(1) adenosine receptor antagonists, J MED CHEM, 44(3), 2001, pp. 316-327
[1,2,4]triazino[4,3-a]benzimidazole acetic acid derivatives: A new class of selective aldose reductase inhibitors
Authors: Da Settimo, F Primofiore, G Da Settimo, A La Motta, C Taliani, S Simorini, F Novellino, E Greco, G Lavecchia, A Boldrini, E
Citation: F. Da Settimo et al., [1,2,4]triazino[4,3-a]benzimidazole acetic acid derivatives: A new class of selective aldose reductase inhibitors, J MED CHEM, 44(25), 2001, pp. 4359-4369
A rational approach to the design of selective substrates and potent nontransportable inhibitors of the excitatory amino acid transporter EAAC1 (EAAT3). New glutamate and aspartate analogues as potential neuroprotective agents
Authors: Campiani, G De Angelis, M Armaroli, S Fattorusso, C Catalanotti, B Ramunno, A Nacci, V Novellino, E Grewer, C Ionescu, D Rauen, T Griffiths, R Sinclair, C Fumagalli, E Mennini, T
Citation: G. Campiani et al., A rational approach to the design of selective substrates and potent nontransportable inhibitors of the excitatory amino acid transporter EAAC1 (EAAT3). New glutamate and aspartate analogues as potential neuroprotective agents, J MED CHEM, 44(16), 2001, pp. 2507-2510
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase
Authors: Mai, A Sbardella, G Artico, M Ragno, R Massa, S Novellino, E Greco, G Lavecchia, A Musiu, C La Colla, M Murgioni, C La Colla, P Loddo, R
Citation: A. Mai et al., Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase, J MED CHEM, 44(16), 2001, pp. 2544-2554
Novel N-(arylalkyl) indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: Synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships
Authors: Primofiore, G Da Settimo, F Taliani, S Marini, AM Novellino, E Greco, G Lavecchia, A Besnard, F Trincavelli, L Costa, B Martini, C
Citation: G. Primofiore et al., Novel N-(arylalkyl) indol-3-ylglyoxylylamides targeted as ligands of the benzodiazepine receptor: Synthesis, biological evaluation, and molecular modeling analysis of the structure-activity relationships, J MED CHEM, 44(14), 2001, pp. 2286-2297
Computer-assisted design, synthesis and biological evaluation of novel pyrrolyl heteroaryl sulfones targeted at HIV-1 reverse transcriptase as non-nucleoside inhibitors
Authors: Silvestri, R Artico, M De Martino, G Novellino, E Greco, G Lavecchia, A Massa, S Loi, AG Doratiotto, S La Colla, P
Citation: R. Silvestri et al., Computer-assisted design, synthesis and biological evaluation of novel pyrrolyl heteroaryl sulfones targeted at HIV-1 reverse transcriptase as non-nucleoside inhibitors, BIO MED CH, 8(9), 2000, pp. 2305-2309
Linking CoMFA and protein homology models of enzyme-inhibitor interactions: an application to non-steroidal aromatase inhibitors
Authors: Cavalli, A Greco, G Novellino, E Recanatini, M
Citation: A. Cavalli et al., Linking CoMFA and protein homology models of enzyme-inhibitor interactions: an application to non-steroidal aromatase inhibitors, BIO MED CH, 8(12), 2000, pp. 2771-2780
Non-nucleoside HIV-1 reverse transcriptase inhibitors: synthesis and biological evaluation of novel quinoxalinylethylpyridylthioureas as potent antiviral agents
Authors: Campiani, G Fabbrini, M Morelli, E Nacci, V Greco, G Novellino, E Maga, G Spadari, S Bergamini, A Faggioli, E Uccella, I Bolacchi, F Marini, S Coletta, M Fracasso, C Caccia, S
Citation: G. Campiani et al., Non-nucleoside HIV-1 reverse transcriptase inhibitors: synthesis and biological evaluation of novel quinoxalinylethylpyridylthioureas as potent antiviral agents, ANTIVIR CHE, 11(2), 2000, pp. 141-155
A G alpha(s) carboxyl-terminal peptide prevents G(s) activation by the A(2A) adenosine receptor
Authors: Mazzoni, MR Taddei, S Giusti, L Rovero, P Galoppini, C D'Ursi, A Albrizio, S Triolo, A Novellino, E Greco, G Lucacchini, A Hamm, HE
Citation: Mr. Mazzoni et al., A G alpha(s) carboxyl-terminal peptide prevents G(s) activation by the A(2A) adenosine receptor, MOLEC PHARM, 58(1), 2000, pp. 226-236
Structure-based design, synthesis, and biological evaluation of navel pyrrolyl aryl sulfones: HIV-1 non-nucleoside reverse transcriptase inhibitors active at nanomolar concentrations
Authors: Artico, M Silvestri, R Pagnozzi, E Bruno, B Novellino, E Greco, G Massa, S Ettorre, A Loi, AG Scintu, F La Colla, P
Citation: M. Artico et al., Structure-based design, synthesis, and biological evaluation of navel pyrrolyl aryl sulfones: HIV-1 non-nucleoside reverse transcriptase inhibitors active at nanomolar concentrations, J MED CHEM, 43(9), 2000, pp. 1886-1891
Modeling of kappa-opioid receptor/agonists interactions using pharmacophore-based and docking simulations
Authors: Lavecchia, A Greco, G Novellino, E Vittorio, F Ronsisvalle, G
Citation: A. Lavecchia et al., Modeling of kappa-opioid receptor/agonists interactions using pharmacophore-based and docking simulations, J MED CHEM, 43(11), 2000, pp. 2124-2134
3-aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: Tricyclic heteroaromatic derivatives as a new class of benzodiazepine receptor ligands
Authors: Primofiore, G Da Settimo, F Taliani, S Marini, AM La Motta, C Novellino, E Greco, G Gesi, M Trincavelli, L Martini, C
Citation: G. Primofiore et al., 3-aryl-[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: Tricyclic heteroaromatic derivatives as a new class of benzodiazepine receptor ligands, J MED CHEM, 43(1), 2000, pp. 96-102
Conformational studies on a synthetic C-terminal fragment of the alpha subunit of G(S) proteins
Authors: Albrizio, S D'Ursi, A Fattorusso, C Galoppini, C Greco, G Mazzoni, MR Novellino, E Rovero, P
Citation: S. Albrizio et al., Conformational studies on a synthetic C-terminal fragment of the alpha subunit of G(S) proteins, BIOPOLYMERS, 54(3), 2000, pp. 186-194
5-alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones: Novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives
Authors: Mai, A Artico, M Sbardella, G Massa, S Novellino, E Greco, G Loi, AG Tramontano, E Marongiu, ME La Colla, P
Citation: A. Mai et al., 5-alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones: Novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives, J MED CHEM, 42(4), 1999, pp. 619-627
Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT3 receptor agonists: Synthesis, further structure-activity relationships, and biological studies
Authors: Campiani, G Morelli, E Gemma, S Nacci, V Butini, S Hamon, M Novellino, E Greco, G Cagnotto, A Goegan, M Cervo, L Dalla Valle, F Fracasso, C Caccia, S Mennini, T
Citation: G. Campiani et al., Pyrroloquinoxaline derivatives as high-affinity and selective 5-HT3 receptor agonists: Synthesis, further structure-activity relationships, and biological studies, J MED CHEM, 42(21), 1999, pp. 4362-4379
Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: Further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity
Authors: Campiani, G Morelli, E Fabbrini, M Nacci, V Greco, G Novellino, E Ramunno, A Maga, G Spadari, S Caliendo, G Bergamini, A Faggioli, E Uccella, I Bolacchi, F Marini, S Coletta, M Nacca, A Caccia, S
Citation: G. Campiani et al., Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: Further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity, J MED CHEM, 42(21), 1999, pp. 4462-4470
Risultati: 1-18 |