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RABELINK TJ
BRAAM B
OPGENORTH TJ
GRONE HJ
KOOMANS HA
JOLES JA
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Authors:
WUWONG JR
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DAYTON BD
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HEMANDEZ L
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SZCZEPANKIEWICZ B
VONGEIDEM TW
OPGENORTH TJ
Citation: Jr. Wuwong et al., PHARMACOLOGICAL CHARACTERIZATION OF A-216546 - AN ORALLY-ACTIVE AND HIGHLY SELECTIVE ANTAGONIST FOR THE TYPE-A ENDOTHELIN RECEPTOR, The FASEB journal, 12(4), 1998, pp. 579-579
Authors:
MCKENNA CJ
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OPGENORTH TJ
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Citation: Cj. Mckenna et al., SELECTIVE ETA-RECEPTOR ANTAGONISM REDUCES NEOINTIMAL HYPERPLASIA IN APORCINE CORONARY STENT MODEL, Journal of the American College of Cardiology, 31(2), 1998, pp. 144-144
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TATLISUMAK T
CARANO RAD
TAKANO K
OPGENORTH TJ
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FISHER M
Citation: T. Tatlisumak et al., A NOVEL ENDOTHELIN ANTAGONIST, A-127722, ATTENUATES ISCHEMIC LESION SIZE IN RATS WITH TEMPORARY MIDDLE CEREBRAL-ARTERY OCCLUSION - A DIFFUSION AND PERFUSION MRI STUDY, Stroke, 29(4), 1998, pp. 850-857
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Citation: Bg. Szczepankiewicz et al., THE EFFECTS OF DIMINISHING ALBUMIN-BINDING TO SOME ENDOTHELIN RECEPTOR ANTAGONISTS, Life sciences (1973), 63(21), 1998, pp. 1905-1912
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OPGENORTH TJ
Citation: G. Liu et al., PYRROLIDINE-3-CARBOXYLIC ACIDS AS ENDOTHELIN ANTAGONISTS - 3 - DISCOVERY OF A POTENT, 2-NONARYL, HIGHLY SELECTIVE ETA ANTAGONIST (A-216546), Journal of medicinal chemistry, 41(17), 1998, pp. 3261-3275
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FERRAZ JGP
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OPGENORTH TJ
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Citation: Jgp. Ferraz et al., ETHANOL ALTERS ETB RECEPTOR-MEDIATED RESPONSES IN THE CANINE LIVER, BUT NOT IN THE RAT STOMACH, Gastroenterology, 114(4), 1998, pp. 170-170
Citation: Dm. Pollock et al., ROLE OF ENDOTHELIN ETA RECEPTORS IN THE HYPERTENSION PRODUCED BY 4-DAY L-NITROARGININE METHYL-ESTER AND CYCLOSPORINE TREATMENT, European journal of pharmacology, 346(1), 1998, pp. 43-50
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MAGNUSON SR
DIXON D
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OPGENORTH TJ
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Citation: Wj. Chiou et al., DISSOCIATION CHARACTERISTICS OF ENDOTHELIN RECEPTOR AGONISTS AND ANTAGONISTS IN CLONED HUMAN TYPE-B ENDOTHELIN RECEPTOR, Endothelium, 5(3), 1997, pp. 179-189
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VERHAGEN AMG
JOLES JA
BRAAM B
OPGENORTH TJ
GRONE HJ
KOOMANS HA
RABELINK TJ
Citation: Amg. Verhagen et al., ENDOTHELIN(A) RECEPTOR BLOCKADE ALLEVIATES HYPERTENSION AND RENAL LESIONS ASSOCIATED WITH CHRONIC NITRIC-OXIDE SYNTHASE INHIBITION, Journal of the American Society of Nephrology, 8, 1997, pp. 1425-1425
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BURKE SE
NELSON RA
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OPGENORTH TJ
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Citation: Se. Burke et al., SELECTIVITY OF ABT-627, AN ANTAGONIST OF THE ENDOTHELIN-A (ET-A) RECEPTOR, ON PRESSOR-RESPONSES IN THE DOMESTIC PIG, The FASEB journal, 11(3), 1997, pp. 2904-2904
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Citation: Dm. Pollock et al., BENEFICIAL EFFECT OF ETA-RECEPTOR BLOCKADE IN A RAT MODEL OF RADIOCONTRAST-INDUCED NEPHROPATHY, Renal failure, 19(6), 1997, pp. 753-761
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OPGENORTH TJ
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Citation: Dd. Borgeson et al., DIFFERENTIAL REGULATION OF CIRCULATING ATRIAL-NATRIURETIC-PEPTIDE ANDBRAIN NATRIURETIC PEPTIDE BY ENDOGENOUS ENDOTHELIN DURING THE PROGRESSION OF EXPERIMENTAL HEART-FAILURE, Journal of the American College of Cardiology, 29(2), 1997, pp. 8169-8169
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LUBBERS NL
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DAYTON BD
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OPGENORTH TJ
Citation: Se. Burke et al., SELECTIVE ANTAGONISM OF THE ETA-RECEPTOR REDUCES NEOINTIMAL HYPERPLASIA AFTER BALLOON-INDUCED VASCULAR INJURY IN PIGS, Journal of cardiovascular pharmacology, 30(1), 1997, pp. 33-41
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CHEN YF
OPGENORTH TJ
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DURAND J
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OPARIL S
Citation: Sj. Chen et al., THE ORALLY-ACTIVE NONPEPTIDE ENDOTHELIN A-RECEPTOR ANTAGONIST A-127722 PREVENTS AND REVERSES HYPOXIA-INDUCED PULMONARY-HYPERTENSION AND PULMONARY VASCULAR REMODELING IN SPRAGUE-DAWLEY RATS, Journal of cardiovascular pharmacology, 29(6), 1997, pp. 713-725
Citation: Jr. Wuwong et al., ENDOTHELIN RECEPTOR ANTAGONISTS - EFFECT OF SERUM-ALBUMIN ON POTENCY AND COMPARISON OF PHARMACOLOGICAL CHARACTERISTICS, The Journal of pharmacology and experimental therapeutics, 281(2), 1997, pp. 791-798
Authors:
TASKER AS
SORENSEN BK
JAE HS
WINN M
VONGELDERN TW
DIXON DB
CHIOU WJ
DAYTON BD
CALZADILA S
HERNANDEZ L
MARSH KC
WUWONG JR
OPGENORTH TJ
Citation: As. Tasker et al., POTENT AND SELECTIVE NON-BENZODIOXOLE-CONTAINING ENDOTHELIN-A RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 40(3), 1997, pp. 322-330
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WINN M
DIXON DB
MARSH KC
NGUYEN B
OPGENORTH TJ
VONGELDERN TW
Citation: Hs. Jae et al., PYRROLIDINE-3-CARBOXYLIC ACIDS AS ENDOTHELIN ANTAGONISTS .2. SULFONAMIDE-BASED ETA ETB MIXED ANTAGONISTS/, Journal of medicinal chemistry, 40(20), 1997, pp. 3217-3227
Authors:
FERRAZ JGP
FARO F
STELLA HJ
FARO R
ANTUNES E
OPGENORTH TJ
WITHRINGTON PG
DENUCCI G
Citation: Jgp. Ferraz et al., EFFECTS OF ETHANOL ON HEPATIC VASCULAR-RESPONSES TO ENDOTHELIN-1 AND IRL-1620, Gastroenterology, 112(4), 1997, pp. 1264-1264
Authors:
FERRAZ JGP
STELLA HJ
FARO F
FARO R
ANTUNES E
OPGENORTH TJ
WITHRINGTON PG
DENUCCI G
Citation: Jgp. Ferraz et al., ROLE OF ENDOTHELIN-RECEPTOR ACTIVATION IN PORTAL VASOCONSTRICTION INDUCED BY ET-1 AND IRL-1620, Gastroenterology, 112(4), 1997, pp. 1264-1264
Authors:
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GURBANOV K
MULRONEY SE
POTLOG C
OPGENORTH TJ
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HARAMATI A
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Citation: Za. Abassi et al., IMPAIRED NITRIC OXIDE-MEDIATED RENAL VASODILATION IN RATS WITH EXPERIMENTAL HEART-FAILURE - ROLE OF ANGIOTENSIN-II, Circulation, 96(10), 1997, pp. 3655-3664