Authors:
Liu, G
Huth, JR
Olejniczak, ET
Mendoza, R
DeVries, P
Leitza, S
Reilly, EB
Okasinski, GF
Fesik, SW
von Geldern, TW
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Authors:
Stewart, AO
Bhatia, PA
McCarty, CM
Patel, MV
Staeger, MA
Arendsen, DL
Gunawardana, IW
Melcher, LM
Zhu, GD
Boyd, SA
Fry, DG
Cool, BL
Kifle, L
Lartey, K
Marsh, KC
Kempf-Grote, AJ
Kilgannon, P
Wisdom, W
Meyer, J
Gallatin, WM
Okasinski, GF
Citation: Ao. Stewart et al., Discovery of inhibitors of cell adhesion molecule expression in human endothelial cells. 1. Selective inhibition of ICAM-1 and E-selectin expression, J MED CHEM, 44(6), 2001, pp. 988-1002
Authors:
Winn, M
Reilly, EB
Liu, G
Huth, JR
Jae, HS
Freeman, J
Pei, ZH
Xin, ZL
Lynch, J
Kester, J
von Geldern, TW
Leitza, S
DeVries, P
Dickinson, R
Mussatto, D
Okasinski, GF
Citation: M. Winn et al., Discovery of novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intercellular adhesion molecule-1 interaction. 4. Structure-activity relationship of substituents on the benzene ring of the cinnamide, J MED CHEM, 44(25), 2001, pp. 4393-4403
Authors:
Zhu, GD
Arendsen, DL
Gunawardana, IW
Boyd, SA
Stewart, AO
Fry, DG
Cool, BL
Kifle, L
Shaefer, V
Meuth, J
Marsh, KC
Kempf-Grote, AJ
Kilgannon, P
Gallatin, WM
Okasinski, GF
Citation: Gd. Zhu et al., Selective inhibition of ICAM-1 and E-selectin expression in human endothelial cells. 2. Aryl modifications of 4-(aryloxy)thieno[2,3-c]pyridines with fine-tuning at C-2 carbamides, J MED CHEM, 44(21), 2001, pp. 3469-3487
Authors:
Pei, ZH
Xin, ZL
Liu, G
Li, YH
Reilly, EB
Lubbers, NL
Huth, JR
Link, JT
von Geldern, TW
Cox, BF
Leitza, S
Gao, Y
Marsh, KC
DeVries, P
Okasinski, GF
Citation: Zh. Pei et al., Discovery of potent antagonists of leukocyte function-associated antigen-1/intercellular adhesion molecule-1 interaction. 3. Amide (C-ring) structure-activity relationship and improvement of overall properties of arylthio cinnamides, J MED CHEM, 44(18), 2001, pp. 2913-2920
Authors:
Kaszubska, W
Zhang, HY
Patterson, RL
Suhar, TS
Uchic, ME
Dickinson, RW
Schaefer, VG
Haasch, D
Janis, RS
DeVries, PJ
Okasinski, GF
Meuth, JL
Citation: W. Kaszubska et al., Expression, purification, and characterization of human recombinant thrombopoietin in Chinese hamster ovary cells, PROT EX PUR, 18(2), 2000, pp. 213-220
Authors:
Liu, G
Link, JT
Pei, ZH
Reilly, EB
Leitza, S
Nguyen, B
Marsh, KC
Okasinski, GF
von Geldern, TW
Ormes, M
Fowler, K
Gallatin, M
Citation: G. Liu et al., Discovery of novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intracellular adhesion molecule-1 interaction. 1. Identification of an additional binding pocket based on an anilino diaryl sulfide lead, J MED CHEM, 43(21), 2000, pp. 4025-4040