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Results: 1-5 |
Results: 5
Synthesis and structure-activity relationships of a new model of arylpiperazines. 5. Study of the physicochemical influence of the pharmacophore on 5-HT1A/alpha(1)-adrenergic receptor affinity: Synthesis of a new derivative with mixed 5-HT1A/D-2 antagonist properties
Authors: Lopez-Rodriguez, ML Morcillo, MJ Fernandez, E Porras, E Orensanz, L Beneytez, ME Manzanares, J Fuentes, JA
Citation: Ml. Lopez-rodriguez et al., Synthesis and structure-activity relationships of a new model of arylpiperazines. 5. Study of the physicochemical influence of the pharmacophore on 5-HT1A/alpha(1)-adrenergic receptor affinity: Synthesis of a new derivative with mixed 5-HT1A/D-2 antagonist properties, J MED CHEM, 44(2), 2001, pp. 186-197
Benzimidazole derivatives. Part 1: Synthesis and structure-activity relationships of new benzimidazole-4-carboxamides and carboxylates as potent and selective 5-HT4 receptor antagonists
Authors: Lopez-Rodriguez, ML Benhamu, B Viso, A Morcillo, MJ Murcia, M Orensanz, L Alfaro, MJ Martin, MI
Citation: Ml. Lopez-rodriguez et al., Benzimidazole derivatives. Part 1: Synthesis and structure-activity relationships of new benzimidazole-4-carboxamides and carboxylates as potent and selective 5-HT4 receptor antagonists, BIO MED CH, 7(11), 1999, pp. 2271-2281
Design and synthesis of 2-[4-[4-(m-(ethylsulfonamido)-phenyl)piperazin-1-yl]butyl]-1,3-dioxoperhydropyrrolo[1,2-c]imidazole (EF-7412) using neural networks. A selective derivative with mixed 5-HT1A/D-2 antagonist properties
Authors: Lopez-Rodriguez, ML Morcillo, MJ Fernandez, E Rosado, ML Orensanz, L Beneytez, ME Manzanares, J Fuentes, JA Schaper, KJ
Citation: Ml. Lopez-rodriguez et al., Design and synthesis of 2-[4-[4-(m-(ethylsulfonamido)-phenyl)piperazin-1-yl]butyl]-1,3-dioxoperhydropyrrolo[1,2-c]imidazole (EF-7412) using neural networks. A selective derivative with mixed 5-HT1A/D-2 antagonist properties, BIOORG MED, 9(12), 1999, pp. 1679-1682
Benzimidazole derivatives. 2. Synthesis and structure-activity relationships of new azabicyclic benzimidazole-4-carboxylic acid derivatives with affinity for serotoninergic 5-HT3 receptors
Authors: Lopez-Rodriguez, ML Benhamu, B Morcillo, MJ Tejada, ID Orensanz, L Alfaro, MJ Martin, MI
Citation: Ml. Lopez-rodriguez et al., Benzimidazole derivatives. 2. Synthesis and structure-activity relationships of new azabicyclic benzimidazole-4-carboxylic acid derivatives with affinity for serotoninergic 5-HT3 receptors, J MED CHEM, 42(24), 1999, pp. 5020-5028
Synthesis and structure-activity relationships of a new model of arylpiperazines. 4. 1-[omega-(4-arylpiperazin-1-yl)alkyl]-3-(diphenylmethylene)-2,5-pyrrolidinediones and -3-(9H-fluoren-9-ylidene)-2,5-pyrrolidinediones: Study of the steric requirements of the terminal amide fragment on 5-HT1A affinity/selectivity
Authors: Lopez-Rodriguez, ML Morcillo, MJ Rovat, TK Fernandez, E Vicente, B Sanz, AM Hernandez, M Orensanz, L
Citation: Ml. Lopez-rodriguez et al., Synthesis and structure-activity relationships of a new model of arylpiperazines. 4. 1-[omega-(4-arylpiperazin-1-yl)alkyl]-3-(diphenylmethylene)-2,5-pyrrolidinediones and -3-(9H-fluoren-9-ylidene)-2,5-pyrrolidinediones: Study of the steric requirements of the terminal amide fragment on 5-HT1A affinity/selectivity, J MED CHEM, 42(1), 1999, pp. 36-49
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