AAAAAA

   
Results: 1-25 | 26-28
Results: 1-25/28
STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS - VII - CHARACTERIZATION OF A NOVEL COCAINE BINDING-SITE IDENTIFIED WITH [I-125] RTI-55 IN MEMBRANES PREPARED FROM HUMAN, MONKEY AND GUINEA-PIG CAUDATE
Authors: ROTHMAN RB SILVERTHORN ML GLOWA JR MATECKA D RICE KC CARROLL FI PARTILLA JS UHL GR VANDENBERGH DJ DERSCH CM
Citation: Rb. Rothman et al., STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS - VII - CHARACTERIZATION OF A NOVEL COCAINE BINDING-SITE IDENTIFIED WITH [I-125] RTI-55 IN MEMBRANES PREPARED FROM HUMAN, MONKEY AND GUINEA-PIG CAUDATE, Synapse, 28(4), 1998, pp. 322-338
OPIOID PEPTIDE RECEPTOR STUDIES - 7 - THE METHYLFENTANYL CONGENER RTI-4614-4 AND ITS 4 ENANTIOMERS BIND TO DIFFERENT DOMAINS OF THE RAT MU-OPIOID RECEPTOR
Authors: LU YF XU H LIUCHEN LY CHEN CG PARTILLA JS BRINE GA CARROLL FI RICE KC LAI J PORRECA F SADEE W ROTHMAN RB
Citation: Yf. Lu et al., OPIOID PEPTIDE RECEPTOR STUDIES - 7 - THE METHYLFENTANYL CONGENER RTI-4614-4 AND ITS 4 ENANTIOMERS BIND TO DIFFERENT DOMAINS OF THE RAT MU-OPIOID RECEPTOR, Synapse, 28(2), 1998, pp. 117-124
OPIOID PEPTIDE RECEPTOR STUDIES - 9 - IDENTIFICATION OF A NOVEL NON-MU-LIKE NON-DELTA-LIKE OPIOID PEPTIDE BINDING-SITE IN RAT-BRAIN
Authors: NI Q XU H PARTILLA JS RICE KC MATECKA D CALDERON SN PORRECA F LAI J SCHMIDHAMMER H KRASSNIG R ROTHMAN RB
Citation: Q. Ni et al., OPIOID PEPTIDE RECEPTOR STUDIES - 9 - IDENTIFICATION OF A NOVEL NON-MU-LIKE NON-DELTA-LIKE OPIOID PEPTIDE BINDING-SITE IN RAT-BRAIN, Peptides (New York, N.Y. 1980), 19(6), 1998, pp. 1079-1090
OPIOID PEPTIDE RECEPTOR STUDIES .8. ONE OF THE MOUSE-BRAIN DELTA(NCX)BINDING-SITES IS SIMILAR TO THE CLONED MOUSE OPIOID DELTA-RECEPTOR - FURTHER EVIDENCE FOR HETEROGENEITY OF DELTA-OPIOID RECEPTORS
Authors: XU H LU YF PARTILLA JS PINTO J CALDERON SN MATECKA D RICE KC LAI J PORRECA F ANANTHAN S ROTHMAN RB
Citation: H. Xu et al., OPIOID PEPTIDE RECEPTOR STUDIES .8. ONE OF THE MOUSE-BRAIN DELTA(NCX)BINDING-SITES IS SIMILAR TO THE CLONED MOUSE OPIOID DELTA-RECEPTOR - FURTHER EVIDENCE FOR HETEROGENEITY OF DELTA-OPIOID RECEPTORS, Peptides, 19(2), 1998, pp. 343-350
N-SUBSTITUTED 9-BETA-METHYL-5-(3-HYDROXYPHENYL)MORPHANS ARE OPIOID RECEPTOR PURE ANTAGONISTS
Authors: THOMAS JB ZHENG XL MASCARELLA SW ROTHMAN RB DERSCH CM PARTILLA JS FLIPPENANDERSON JL GEORGE CF CANTRELL BE ZIMMERMAN DM CARROLL FI
Citation: Jb. Thomas et al., N-SUBSTITUTED 9-BETA-METHYL-5-(3-HYDROXYPHENYL)MORPHANS ARE OPIOID RECEPTOR PURE ANTAGONISTS, Journal of medicinal chemistry, 41(21), 1998, pp. 4143-4149
INVESTIGATION OF THE N-SUBSTITUENT CONFORMATION GOVERNING POTENCY ANDMU-RECEPTOR SUBTYPE-SELECTIVITY IN (-(3R,4R)-DIMETHYL-4-(3-HYDROXYPHENYL)PIPERIDINE OPIOID ANTAGONISTS())
Authors: THOMAS JB MASCARELLA SW ROTHMAN RB PARTILLA JS XU H MCCULLOUGH KB DERSCH CN CANTRELL BE ZIMMERMAN DM CARROLL FI
Citation: Jb. Thomas et al., INVESTIGATION OF THE N-SUBSTITUENT CONFORMATION GOVERNING POTENCY ANDMU-RECEPTOR SUBTYPE-SELECTIVITY IN (-(3R,4R)-DIMETHYL-4-(3-HYDROXYPHENYL)PIPERIDINE OPIOID ANTAGONISTS()), Journal of medicinal chemistry, 41(11), 1998, pp. 1980-1990
PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .24. SYNTHESIS, SINGLE-CRYSTAL X-RAY ANALYSES, IN-VITRO AND IN-VIVO PROPERTIES OF -3,14-DIHYDROXY-17-METHYL-4,5-ALPHA-EPOXYMORPHINAN AND -3,14-DIHYDROXY-17-METHYL-4,5-ALPHA-EPOXYMORPHINAN
Authors: KAYAKIRI H JACOBSON AE RICE KC ROTHMAN RB XU H FLIPPENANDERSON JL GEORGE C ACETO MD BOWMAN ER HARRIS LS MAY EL PARTILLA JS BECKETTS K
Citation: H. Kayakiri et al., PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .24. SYNTHESIS, SINGLE-CRYSTAL X-RAY ANALYSES, IN-VITRO AND IN-VIVO PROPERTIES OF -3,14-DIHYDROXY-17-METHYL-4,5-ALPHA-EPOXYMORPHINAN AND -3,14-DIHYDROXY-17-METHYL-4,5-ALPHA-EPOXYMORPHINAN, Medicinal chemistry research, 6(6), 1996, pp. 427-438
PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .22. SYNTHESIS AND CHARACTERIZATION OF OPTICALLY PURE [H-3] IPERAZINYL)-3-METHOXYBENZYL]-N,N-DIETHYLBENZAMIDE, [H-3] SNC-121, A NOVEL HIGH-AFFINITY AND SELECTIVELIGAND FOR DELTA-OPIOID RECEPTORS())
Authors: CALDERON SN BERTHA CM GUTKIND JS XU H PARTILLA JS ROTHMAN RB RICE KC
Citation: Sn. Calderon et al., PROBES FOR NARCOTIC RECEPTOR-MEDIATED PHENOMENA .22. SYNTHESIS AND CHARACTERIZATION OF OPTICALLY PURE [H-3] IPERAZINYL)-3-METHOXYBENZYL]-N,N-DIETHYLBENZAMIDE, [H-3] SNC-121, A NOVEL HIGH-AFFINITY AND SELECTIVELIGAND FOR DELTA-OPIOID RECEPTORS()), Journal of labelled compounds & radiopharmaceuticals, 38(9), 1996, pp. 847-850
DEVELOPMENT OF NOVEL, POTENT, AND SELECTIVE DOPAMINE REUPTAKE INHIBITORS THROUGH ALTERATION OF THE PIPERAZINE RING OF PHENYLMETHOXY)ETHYL]-4-(3-PHENYLPROPYL)PIPERAZINES AND HENYL)METHOXY]ETHYL]-4-(3-PHENYLPROPYL)PIPERAZINES (GBR-12935 AND GBR-12909)
Authors: MATECKA D ROTHMAN RB RADESCA L DECOSTA BR DERSCH CM PARTILLA JS PERT A GLOWA JR WOJNICKI FHE RICE KC
Citation: D. Matecka et al., DEVELOPMENT OF NOVEL, POTENT, AND SELECTIVE DOPAMINE REUPTAKE INHIBITORS THROUGH ALTERATION OF THE PIPERAZINE RING OF PHENYLMETHOXY)ETHYL]-4-(3-PHENYLPROPYL)PIPERAZINES AND HENYL)METHOXY]ETHYL]-4-(3-PHENYLPROPYL)PIPERAZINES (GBR-12935 AND GBR-12909), Journal of medicinal chemistry, 39(24), 1996, pp. 4704-4716
HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC RESOLUTION OF SYNTHETIC OPIATE AND ANTI-OPIATE PEPTIDES FROM HUMAN PLASMA
Authors: PARTILLA JS YOU J ROTHMAN RB
Citation: Js. Partilla et al., HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC RESOLUTION OF SYNTHETIC OPIATE AND ANTI-OPIATE PEPTIDES FROM HUMAN PLASMA, Journal of chromatography B. Biomedical applications, 667(1), 1995, pp. 49-56
LIGAND SELECTIVITY OF CLONED HUMAN AND RAT OPIOID-MU RECEPTORS
Authors: ROTHMAN RB XU H WANG JB PARTILLA JS KAYAKIRI H RICE KC UHL GR
Citation: Rb. Rothman et al., LIGAND SELECTIVITY OF CLONED HUMAN AND RAT OPIOID-MU RECEPTORS, Synapse, 21(1), 1995, pp. 60-64
-3,14-DIHYDROXY-17-METHYL-4,5-ALPHA-EPOXYMORPHINAN ([I-125]IOXY-AGO) - A POTENT AND SELECTIVE RADIOLIGAND FOR OPIOID MU-RECEPTORS
Authors: XU H GOODMAN CB PARTILLA JS NI Q KAYAKIRI H RICE KC ROTHMAN RB
Citation: H. Xu et al., -3,14-DIHYDROXY-17-METHYL-4,5-ALPHA-EPOXYMORPHINAN ([I-125]IOXY-AGO) - A POTENT AND SELECTIVE RADIOLIGAND FOR OPIOID MU-RECEPTORS, Synapse, 19(2), 1995, pp. 105-111
OPIOID PEPTIDE RECEPTOR STUDIES .3. INTERACTION OF OPIOID-PEPTIDES AND OTHER DRUGS WITH 4 SUBTYPES OF THE KAPPA(2) RECEPTOR IN GUINEA-PIG BRAIN
Authors: NI Q XU H PARTILLA JS DECOSTA BR RICE KC KAYAKIRI H ROTHMAN RB
Citation: Q. Ni et al., OPIOID PEPTIDE RECEPTOR STUDIES .3. INTERACTION OF OPIOID-PEPTIDES AND OTHER DRUGS WITH 4 SUBTYPES OF THE KAPPA(2) RECEPTOR IN GUINEA-PIG BRAIN, Peptides, 16(6), 1995, pp. 1083-1095
OPIOID PEPTIDE RECEPTOR STUDIES .4. ANTISENSE OLIGODEOXYNUCLEOTIDE TOTHE DELTA-OPIOID RECEPTOR DELINEATES OPIOID RECEPTOR SUBTYPES
Authors: CHA XY XU H NI Q PARTILLA JS RICE KC MATECKA D CALDERON SN PORRECA F LAI J ROTHMAN RB
Citation: Xy. Cha et al., OPIOID PEPTIDE RECEPTOR STUDIES .4. ANTISENSE OLIGODEOXYNUCLEOTIDE TOTHE DELTA-OPIOID RECEPTOR DELINEATES OPIOID RECEPTOR SUBTYPES, Regulatory peptides, 59(2), 1995, pp. 247-253
STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .6. CHARACTERIZATION OF A NOVEL COCAINE BINDING-SITE, IDENTIFIED WITH [I-125] RTI-55, IN MEMBRANES PREPARED FROM WHOLE RAT-BRAIN MINUS CAUDATE
Authors: ROTHMAN RB SILVERTHORN ML BAUMANN MH GOODMAN CB CADET JL MATECKA D RICE KC CARROLL FI WANG JB UHL GR PARTILLA JS DERSCH CM
Citation: Rb. Rothman et al., STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .6. CHARACTERIZATION OF A NOVEL COCAINE BINDING-SITE, IDENTIFIED WITH [I-125] RTI-55, IN MEMBRANES PREPARED FROM WHOLE RAT-BRAIN MINUS CAUDATE, The Journal of pharmacology and experimental therapeutics, 274(1), 1995, pp. 385-395
STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .5. DEMONSTRATION OF 2 BINDING-SITES FOR THE COCAINE ANALOG [I-125] RTI-55 ASSOCIATED WITH THE 5-HT TRANSPORTER IN RAT-BRAIN MEMBRANES
Authors: SILVERTHORN ML DERSCH CM BAUMANN MH CADET JL PARTILLA JS RICE KC CARROLL FI BECKETTS KM BROCKINGTON A ROTHMAN RB
Citation: Ml. Silverthorn et al., STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .5. DEMONSTRATION OF 2 BINDING-SITES FOR THE COCAINE ANALOG [I-125] RTI-55 ASSOCIATED WITH THE 5-HT TRANSPORTER IN RAT-BRAIN MEMBRANES, The Journal of pharmacology and experimental therapeutics, 273(1), 1995, pp. 213-222
DIHYDROCODEINONE-HYDRAZONE, DIHYDROCODEINONE-OXIME, NALOXONE-3-OME-OXIME, AND CLOCINNAMOX FAIL TO IRREVERSIBLY INHIBIT OPIOID KAPPA-RECEPTOR-BINDING
Authors: NI Q XU H PARTILLA JS DECOSTA BR RICE KC BORSODI A HOSZTAFI S ROTHMAN RB
Citation: Q. Ni et al., DIHYDROCODEINONE-HYDRAZONE, DIHYDROCODEINONE-OXIME, NALOXONE-3-OME-OXIME, AND CLOCINNAMOX FAIL TO IRREVERSIBLY INHIBIT OPIOID KAPPA-RECEPTOR-BINDING, Neurochemical research, 19(9), 1994, pp. 1159-1163
STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .1. DOPAMINE REUPTAKE BLOCKERS INHIBIT [H-3] MAZINDOL BINDING TO THE DOPAMINE TRANSPORTER BY A COMPETITIVE MECHANISM - PRELIMINARY EVIDENCE FOR DIFFERENT BINDING DOMAINS
Authors: DERSCH CM AKUNNE HC PARTILLA JS CHAR GU DECOSTA BR RICE KC CARROLL FI ROTHMAN RB
Citation: Cm. Dersch et al., STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .1. DOPAMINE REUPTAKE BLOCKERS INHIBIT [H-3] MAZINDOL BINDING TO THE DOPAMINE TRANSPORTER BY A COMPETITIVE MECHANISM - PRELIMINARY EVIDENCE FOR DIFFERENT BINDING DOMAINS, Neurochemical research, 19(2), 1994, pp. 201-208
[H-3] SNC121 - A NOVEL HIGH-AFFINITY LIGAND FOR RAT-BRAIN DELTA-RECEPTORS - PRELIMINARY STUDIES
Authors: NI Q XU H PARTILLA JS PORRECA F CALDERON SN RICE KC SMITH LE MCNUTT RW ROTHMAN RB
Citation: Q. Ni et al., [H-3] SNC121 - A NOVEL HIGH-AFFINITY LIGAND FOR RAT-BRAIN DELTA-RECEPTORS - PRELIMINARY STUDIES, Regulatory peptides, 54(1), 1994, pp. 209-210
THE LIGAND-SELECTIVITY OF CLONED HUMAN AND RAT OPIATE MU-RECEPTORS STUDIED WITH [I-125]IOXY-AGO
Authors: ROTHMAN RB XU H WANG JB PARTILLA JS KAYAKIRI H RICE KC UHL GR
Citation: Rb. Rothman et al., THE LIGAND-SELECTIVITY OF CLONED HUMAN AND RAT OPIATE MU-RECEPTORS STUDIED WITH [I-125]IOXY-AGO, Regulatory peptides, 54(1), 1994, pp. 249-250
[I-125] IOXY-AGO - A HIGH-AFFINITY, MU-SELECTIVE AGONIST OPIOID RECEPTOR-LIGAND
Authors: XU H PARTILLA JS BECKETTS KM KAYAKIRI H RICE KC ROTHMAN RB
Citation: H. Xu et al., [I-125] IOXY-AGO - A HIGH-AFFINITY, MU-SELECTIVE AGONIST OPIOID RECEPTOR-LIGAND, Regulatory peptides, 54(1), 1994, pp. 331-332
STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .4. DEMONSTRATION OF A MULTIPLICITY OF BINDING-SITES IN RAT CAUDATE MEMBRANES FOR THE COCAINE ANALOG [I-125] RTI-55
Authors: ROTHMAN RB CADET JL AKUNNE HC SILVERTHORN ML BAUMANN MH CARROLL FI RICE KC DECOSTA BR PARTILLA JS WANG JB UHL G GLOWA JR DERSCH CM
Citation: Rb. Rothman et al., STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .4. DEMONSTRATION OF A MULTIPLICITY OF BINDING-SITES IN RAT CAUDATE MEMBRANES FOR THE COCAINE ANALOG [I-125] RTI-55, The Journal of pharmacology and experimental therapeutics, 270(1), 1994, pp. 296-309
STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .3. DEMONSTRATION OF 2 BINDING-SITES FOR [H-3] GBR12935 AND [H-3] BTCP IN RAT CAUDATE MEMBRANES
Authors: AKUNNE HC DERSCH CM CADET JL BAUMANN MH CHAR GU PARTILLA JS DECOSTA BR RICE KC CARROLL FI ROTHMAN RB
Citation: Hc. Akunne et al., STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .3. DEMONSTRATION OF 2 BINDING-SITES FOR [H-3] GBR12935 AND [H-3] BTCP IN RAT CAUDATE MEMBRANES, The Journal of pharmacology and experimental therapeutics, 268(3), 1994, pp. 1462-1475
[125I]RTI-55, A HIGH-AFFINITY COCAINE ANALOG, LABELS 2 BINDING-SITES IN HUMAN CAUDATE MEMBRANES POSSIBLY RELATED TO THE 5-HT TRANSPORTER
Authors: SILVERTHOM ML DERSCH CM PARTILLA JS CARROLL FI MATECKA DL RICE KC ROTHMAN RB
Citation: Ml. Silverthom et al., [125I]RTI-55, A HIGH-AFFINITY COCAINE ANALOG, LABELS 2 BINDING-SITES IN HUMAN CAUDATE MEMBRANES POSSIBLY RELATED TO THE 5-HT TRANSPORTER, Biological psychiatry, 35(9), 1994, pp. 644-644
STEREOCHEMICAL REQUIREMENTS FOR PSEUDOIRREVERSIBLE INHIBITION OF OPIOID MU RECEPTOR-BINDING BY THE 3-METHYLFENTANYL CONGENERS, RTI-46144 AND ITS ENANTIOMERS - EVIDENCE FOR DIFFERENT BINDING DOMAINS
Authors: NI Q XU H PARTILLA JS STARK PA CARROLL FI BRINE GA ROTHMAN RB
Citation: Q. Ni et al., STEREOCHEMICAL REQUIREMENTS FOR PSEUDOIRREVERSIBLE INHIBITION OF OPIOID MU RECEPTOR-BINDING BY THE 3-METHYLFENTANYL CONGENERS, RTI-46144 AND ITS ENANTIOMERS - EVIDENCE FOR DIFFERENT BINDING DOMAINS, Synapse, 15(4), 1993, pp. 296-306
Risultati: 1-25 | 26-28