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Results: 1-25 | 26-49
Results: 1-25/49
NA-DEPENDENT METABOLIC COUPLING UPON 5-HT1B RECEPTOR ACTIVATION BY SUMATRIPTAN AND RELATED AGONISTS()
Authors: PAUWELS PJ
Citation: Pj. Pauwels, NA-DEPENDENT METABOLIC COUPLING UPON 5-HT1B RECEPTOR ACTIVATION BY SUMATRIPTAN AND RELATED AGONISTS(), Receptors & channels, 5(6), 1998, pp. 367-373
SYNTHESIS OF NEW BENZOTHIENYLPIPERAZINE DERIVATIVES AND THEIR CHARACTERIZATION AT BOTH 5HT(1A) AND 5HT(1B) RECEPTOR-SITES
Authors: LAMOTHE M PAUWELS PJ LEBORGNE M HALAZY S
Citation: M. Lamothe et al., SYNTHESIS OF NEW BENZOTHIENYLPIPERAZINE DERIVATIVES AND THEIR CHARACTERIZATION AT BOTH 5HT(1A) AND 5HT(1B) RECEPTOR-SITES, Medicinal chemistry research, 8(3), 1998, pp. 132-142
5-(SULFONYL)OXY-TRYPTAMINES AND ETHYLAMINO SIDE-CHAIN RESTRICTED DERIVATIVES - STRUCTURE-AFFINITY RELATIONSHIPS FOR H5-HT1B AND H5-HT1D RECEPTORS
Authors: BARF T WIKSTROM H PAUWELS PJ PALMIER C TARDIF S LUNDMARK M SUNDELL S
Citation: T. Barf et al., 5-(SULFONYL)OXY-TRYPTAMINES AND ETHYLAMINO SIDE-CHAIN RESTRICTED DERIVATIVES - STRUCTURE-AFFINITY RELATIONSHIPS FOR H5-HT1B AND H5-HT1D RECEPTORS, Bioorganic & medicinal chemistry, 6(9), 1998, pp. 1469-1479
DIMERIZATION OF SUMATRIPTAN AS AN EFFICIENT WAY TO DESIGN A POTENT, CENTRALLY AND ORALLY-ACTIVE 5-HT1B AGONIST
Authors: PEREZ M PAUWELS PJ FOURRIER C CHOPIN P VALENTIN JP JOHN GW MARIEN M HALAZY S
Citation: M. Perez et al., DIMERIZATION OF SUMATRIPTAN AS AN EFFICIENT WAY TO DESIGN A POTENT, CENTRALLY AND ORALLY-ACTIVE 5-HT1B AGONIST, Bioorganic & medicinal chemistry letters, 8(6), 1998, pp. 675-680
DIMERS OF 5HT(1) LIGANDS PREFERENTIALLY BIND TO 5HT(1B 1D) RECEPTOR SUBTYPES/
Authors: PEREZ M JORANDLEBRUN C PAUWELS PJ PALLARD I HALAZY S
Citation: M. Perez et al., DIMERS OF 5HT(1) LIGANDS PREFERENTIALLY BIND TO 5HT(1B 1D) RECEPTOR SUBTYPES/, Bioorganic & medicinal chemistry letters, 8(11), 1998, pp. 1407-1412
A MODIFIED OVERLAP EXTENSION PCR METHOD TO CREATE CHIMERIC GENES IN THE ABSENCE OF RESTRICTION ENZYMES
Authors: WURCH T LESTIENNE F PAUWELS PJ
Citation: T. Wurch et al., A MODIFIED OVERLAP EXTENSION PCR METHOD TO CREATE CHIMERIC GENES IN THE ABSENCE OF RESTRICTION ENZYMES, Biotechnology techniques, 12(9), 1998, pp. 653-657
PREDOMINANT EXPRESSION OF SEROTONIN 5-HT1B RECEPTOR MESSENGER-RNA IN PIG CORONARY-ARTERY
Authors: WURCH T PAUWELS PJ
Citation: T. Wurch et Pj. Pauwels, PREDOMINANT EXPRESSION OF SEROTONIN 5-HT1B RECEPTOR MESSENGER-RNA IN PIG CORONARY-ARTERY, Neuroscience research communications, 23(1), 1998, pp. 45-53
DIMERIZATION OF 8-OH-DPAT INCREASES ACTIVITY AT SEROTONIN 5-HT1A RECEPTORS
Authors: PAUWELS PJ DUPUIS DS PEREZ M HALAZY S
Citation: Pj. Pauwels et al., DIMERIZATION OF 8-OH-DPAT INCREASES ACTIVITY AT SEROTONIN 5-HT1A RECEPTORS, Naunyn-Schmiedeberg's archives of pharmacology, 358(4), 1998, pp. 404-410
SPECIFIC INTERACTION OF 5-HT-MODULINE WITH HUMAN 5-HT1B AS WELL AS 5-HT1D RECEPTORS EXPRESSED IN TRANSFECTED CULTURED-CELLS
Authors: ROUSSELLE JC PLANTEFOL M FILLION MP MASSOT O PAUWELS PJ FILLION G
Citation: Jc. Rousselle et al., SPECIFIC INTERACTION OF 5-HT-MODULINE WITH HUMAN 5-HT1B AS WELL AS 5-HT1D RECEPTORS EXPRESSED IN TRANSFECTED CULTURED-CELLS, Naunyn-Schmiedeberg's archives of pharmacology, 358(3), 1998, pp. 279-286
MUTATION OF THR373 IN THE 3RD INTRACELLULAR LOOP OF THE HUMAN ALPHA(2A)-ADRENERGIC RECEPTOR PROMOTES PARTIAL AGONIST ACTIVITY FROM ANTAGONISTS
Authors: WURCH T PALMIER C RAULY I COLPAERT FC PAUWELS PJ
Citation: T. Wurch et al., MUTATION OF THR373 IN THE 3RD INTRACELLULAR LOOP OF THE HUMAN ALPHA(2A)-ADRENERGIC RECEPTOR PROMOTES PARTIAL AGONIST ACTIVITY FROM ANTAGONISTS, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 642-642
IN-VITRO VASCULAR AND NEURONAL ACTIONS OF F-11356, A NOVEL HIGH EFFICACY 5HT(1B D) RECEPTOR AGONIST, IN MODELS RELEVANT TO MIGRAINE/
Authors: JOHN GW VALENTIN JP LEGRAND B BONNAFOUS R PANISSIE A VIE B PEREZ M HALAZY S PAUWELS PJ COLPAERT FC
Citation: Gw. John et al., IN-VITRO VASCULAR AND NEURONAL ACTIONS OF F-11356, A NOVEL HIGH EFFICACY 5HT(1B D) RECEPTOR AGONIST, IN MODELS RELEVANT TO MIGRAINE/, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 5262-5262
F-11356, A NEW 5-HT DERIVATIVE, WITH SELECTIVE, POTENT AND HIGH EFFICACY AGONIST PROPERTIES AT 5-HT1B D RECEPTORS/
Authors: PAUWELS PJ PALMIER C TARDIF S WURCH T PEREZ M CARILLADURAND E JOHN GW HALAZY S COLPAERT FC
Citation: Pj. Pauwels et al., F-11356, A NEW 5-HT DERIVATIVE, WITH SELECTIVE, POTENT AND HIGH EFFICACY AGONIST PROPERTIES AT 5-HT1B D RECEPTORS/, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 5263-5263
INTERACTION OF 5 HT1B D LIGANDS WITH RECOMBINANT-H 5-HT1A RECEPTORS -INTRINSIC ACTIVITY AND MODULATION BY G-PROTEIN ACTIVATION STATE/
Authors: PAUWELS PJ PALMIER C DUPUIS DS COLPAERT FC
Citation: Pj. Pauwels et al., INTERACTION OF 5 HT1B D LIGANDS WITH RECOMBINANT-H 5-HT1A RECEPTORS -INTRINSIC ACTIVITY AND MODULATION BY G-PROTEIN ACTIVATION STATE/, Naunyn-Schmiedeberg's archives of pharmacology, 357(5), 1998, pp. 490-499
F-11440, A POTENT, SELECTIVE, HIGH EFFICACY 5-HT1A RECEPTOR AGONIST WITH MARKED ANXIOLYTIC AND ANTIDEPRESSANT POTENTIAL
Authors: KOEK W PATOISEAU JF ASSIE MB COSI C KLEVEN MS DUPONTPASSELAIGUE E CARILLADURAND E PALMIER C VALENTIN JP JOHN G PAUWELS PJ TARAYRE JP COLPAERT FC
Citation: W. Koek et al., F-11440, A POTENT, SELECTIVE, HIGH EFFICACY 5-HT1A RECEPTOR AGONIST WITH MARKED ANXIOLYTIC AND ANTIDEPRESSANT POTENTIAL, The Journal of pharmacology and experimental therapeutics, 287(1), 1998, pp. 266-283
AUTORADIOGRAPHY OF SEROTONIN 5-HT1A RECEPTOR-ACTIVATED G-PROTEINS IN GUINEA-PIG BRAIN SECTIONS BY AGONIST-STIMULATED [S-35] GTP-GAMMA-S BINDING
Authors: DUPUIS DS PALMIER C COLPAERT FC PAUWELS PJ
Citation: Ds. Dupuis et al., AUTORADIOGRAPHY OF SEROTONIN 5-HT1A RECEPTOR-ACTIVATED G-PROTEINS IN GUINEA-PIG BRAIN SECTIONS BY AGONIST-STIMULATED [S-35] GTP-GAMMA-S BINDING, Journal of neurochemistry, 70(3), 1998, pp. 1258-1268
G-PROTEIN ACTIVATION AT 5-HT1A RECEPTORS BY THE 5-HT(1F) LIGAND LY334370 IN GUINEA-PIG BRAIN SECTIONS AND RECOMBINANT CELL-LINES
Authors: DUPUIS DS COLPAERT FC PAUWELS PJ
Citation: Ds. Dupuis et al., G-PROTEIN ACTIVATION AT 5-HT1A RECEPTORS BY THE 5-HT(1F) LIGAND LY334370 IN GUINEA-PIG BRAIN SECTIONS AND RECOMBINANT CELL-LINES, British Journal of Pharmacology, 124(2), 1998, pp. 283-290
PHARMACOLOGICAL ANALYSIS OF G-PROTEIN ACTIVATION MEDIATED BY GUINEA-PIG RECOMBINANT 5-HT1B RECEPTORS IN C6-GLIAL CELLS - SIMILARITIES WITH THE HUMAN 5-HT1B RECEPTOR
Authors: PAUWELS PJ WURCH T PALMIER C COLPAERT FC
Citation: Pj. Pauwels et al., PHARMACOLOGICAL ANALYSIS OF G-PROTEIN ACTIVATION MEDIATED BY GUINEA-PIG RECOMBINANT 5-HT1B RECEPTORS IN C6-GLIAL CELLS - SIMILARITIES WITH THE HUMAN 5-HT1B RECEPTOR, British Journal of Pharmacology, 123(1), 1998, pp. 51-62
REGULATION OF METALLOTHIONEIN-III (GIF) MESSENGER-RNA IN THE BRAIN OFPATIENTS WITH ALZHEIMER-DISEASE IS NOT IMPAIRED
Authors: AMOUREUX MC VANGOOL D HERRERO MT DOM R COLPAERT FC PAUWELS PJ
Citation: Mc. Amoureux et al., REGULATION OF METALLOTHIONEIN-III (GIF) MESSENGER-RNA IN THE BRAIN OFPATIENTS WITH ALZHEIMER-DISEASE IS NOT IMPAIRED, Molecular and chemical neuropathology, 32(1-3), 1997, pp. 101-121
ARYLPIPERAZIDE DERIVATIVES OF PHENYLPIPERAZINES AS A NEW CLASS OF POTENT AND SELECTIVE 5-HT1B RECEPTOR ANTAGONISTS
Authors: JORANDLEBRUN C PAUWELS PJ PALMIER C CHOPIN P MORET C MARIEN M HALAZY S
Citation: C. Jorandlebrun et al., ARYLPIPERAZIDE DERIVATIVES OF PHENYLPIPERAZINES AS A NEW CLASS OF POTENT AND SELECTIVE 5-HT1B RECEPTOR ANTAGONISTS, Bioorganic & medicinal chemistry letters, 7(24), 1997, pp. 3183-3188
COMPETITIVE AND SILENT ANTAGONISM OF RECOMBINANT 5-HT1B RECEPTORS BY AMILORIDE
Authors: PAUWELS PJ
Citation: Pj. Pauwels, COMPETITIVE AND SILENT ANTAGONISM OF RECOMBINANT 5-HT1B RECEPTORS BY AMILORIDE, General pharmacology, 29(5), 1997, pp. 749-751
5-HT1B D RECEPTOR ANTAGONISTS
Authors: PAUWELS PJ
Citation: Pj. Pauwels, 5-HT1B D RECEPTOR ANTAGONISTS, General pharmacology, 29(3), 1997, pp. 293-303
SYNTHESIS, BINDING-AFFINITY AND INTRINSIC ACTIVITY OF NEW ANILIDE DERIVATIVES OF SEROTONIN AT HUMAN 5-HT1D RECEPTORS
Authors: PEREZ M AYERBE N FOURRIER C SIGOGNEAU I PAUWELS PJ PALMIER C JOHN GW VALENTIN JP HALAZY S
Citation: M. Perez et al., SYNTHESIS, BINDING-AFFINITY AND INTRINSIC ACTIVITY OF NEW ANILIDE DERIVATIVES OF SEROTONIN AT HUMAN 5-HT1D RECEPTORS, European journal of medicinal chemistry, 32(2), 1997, pp. 129-134
HOW EFFICACIOUS ARE 5-HT1B D RECEPTOR LIGANDS - AN ANSWER FROM GTP-GAMMA-S BINDING-STUDIES WITH STABLY TRANSFECTED C6-GLIAL CELL-LINES/
Authors: PAUWELS PJ TARDIF S PALMIER C WURCH T COLPAERT FC
Citation: Pj. Pauwels et al., HOW EFFICACIOUS ARE 5-HT1B D RECEPTOR LIGANDS - AN ANSWER FROM GTP-GAMMA-S BINDING-STUDIES WITH STABLY TRANSFECTED C6-GLIAL CELL-LINES/, Neuropharmacology, 36(4-5), 1997, pp. 499-512
STIMULATED [S-35] GTP-GAMMA-S BINDING BY 5-HT1A RECEPTOR AGONISTS IN RECOMBINANT CELL-LINES - MODULATION OF APPARENT EFFICACY BY G-PROTEIN ACTIVATION STATE
Authors: PAUWELS PJ TARDIF S WURCH T COLPAERT FC
Citation: Pj. Pauwels et al., STIMULATED [S-35] GTP-GAMMA-S BINDING BY 5-HT1A RECEPTOR AGONISTS IN RECOMBINANT CELL-LINES - MODULATION OF APPARENT EFFICACY BY G-PROTEIN ACTIVATION STATE, Naunyn-Schmiedeberg's archives of pharmacology, 356(5), 1997, pp. 551-561
SEQUENCE AND FUNCTIONAL-ANALYSIS OF CLONED GUINEA-PIG AND RAT SEROTONIN 5-HT1D RECEPTORS, COMMON PHARMACOLOGICAL FEATURES WITHIN THE 5-HT1DRECEPTOR SUBFAMILY
Authors: WURCH T PALMIER C COLPAERT FC PAUWELS PJ
Citation: T. Wurch et al., SEQUENCE AND FUNCTIONAL-ANALYSIS OF CLONED GUINEA-PIG AND RAT SEROTONIN 5-HT1D RECEPTORS, COMMON PHARMACOLOGICAL FEATURES WITHIN THE 5-HT1DRECEPTOR SUBFAMILY, Journal of neurochemistry, 68(1), 1997, pp. 410-418
Risultati: 1-25 | 26-49