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Results: 1-18 |
Results: 18
CLONING AND EXPRESSION OF THE RHESUS-MONKEY OXYTOCIN RECEPTOR
Authors: SALVATORE CA WOYDEN CJ GUIDOTTI MT PETTIBONE DJ JACOBSON MA
Citation: Ca. Salvatore et al., CLONING AND EXPRESSION OF THE RHESUS-MONKEY OXYTOCIN RECEPTOR, Journal of receptor and signal transduction research, 18(1), 1998, pp. 15-24
NONPEPTIDE OXYTOCIN ANTAGONISTS - POTENT, ORALLY BIOAVAILABLE ANALOGSOF L-371,257 CONTAINING A 1-R-(PYRIDYL)ETHYL ETHER TERMINUS
Authors: KUO MS BOCK MG FREIDINGER RM GUIDOTTI MT LIS EV PAWLUCZYK JM PERLOW DS PETTIBONE DJ QUIGLEY AG REISS DR WILLIAMS PD WOYDEN CJ
Citation: Ms. Kuo et al., NONPEPTIDE OXYTOCIN ANTAGONISTS - POTENT, ORALLY BIOAVAILABLE ANALOGSOF L-371,257 CONTAINING A 1-R-(PYRIDYL)ETHYL ETHER TERMINUS, Bioorganic & medicinal chemistry letters, 8(21), 1998, pp. 3081-3086
DEVELOPMENT OF ORALLY-ACTIVE OXYTOCIN ANTAGONISTS - STUDIES ON DIN-3-YLMETHYL)PIPERIDIN-4-YLOXY]-2-METHOXYBENZOYL IPERIDIN-4-YL)-1,4-DIHYDROBENZ[D][1,3]OXAZIN-2-ONE (L-372,662) AND RELATED PYRIDINES
Authors: BELL IM ERB JM FREIDINGER RM GALLICCHIO SN GUARE JP GUIDOTTI MT HALPIN RA HOBBS DW HOMNICK CF KUO MS LIS EV MATHRE DJ MICHELSON SR PAWLUCZYK JM PETTIBONE DJ REISS DR VICKERS S WILLIAMS PD WOYDEN CJ
Citation: Im. Bell et al., DEVELOPMENT OF ORALLY-ACTIVE OXYTOCIN ANTAGONISTS - STUDIES ON DIN-3-YLMETHYL)PIPERIDIN-4-YLOXY]-2-METHOXYBENZOYL IPERIDIN-4-YL)-1,4-DIHYDROBENZ[D][1,3]OXAZIN-2-ONE (L-372,662) AND RELATED PYRIDINES, Journal of medicinal chemistry, 41(12), 1998, pp. 2146-2163
DISCOVERY AND DEVELOPMENT OF NONPEPTIDE ANTAGONISTS OF PEPTIDE-HORMONE RECEPTORS
Authors: PETTIBONE DJ FREIDINGER RM
Citation: Dj. Pettibone et Rm. Freidinger, DISCOVERY AND DEVELOPMENT OF NONPEPTIDE ANTAGONISTS OF PEPTIDE-HORMONE RECEPTORS, Biochemical Society transactions, 25(3), 1997, pp. 1051-1057
SMALL-MOLECULE LIGANDS FOR OXYTOCIN AND VASOPRESSIN RECEPTORS
Authors: FREIDINGER RM PETTIBONE DJ
Citation: Rm. Freidinger et Dj. Pettibone, SMALL-MOLECULE LIGANDS FOR OXYTOCIN AND VASOPRESSIN RECEPTORS, Medicinal research reviews, 17(1), 1997, pp. 1-16
PHARMACOLOGY OF L-744,453, A NOVEL NONPEPTIDYL ENDOTHELIN ANTAGONIST
Authors: WILLIAMS DL MURPHY KL NOLAN NA OBRIEN JA LIS EV PETTIBONE DJ CLINESCHMIDT BV KRAUSE SM VEBER DF NAYLOR EM CHAKRAVARTY PK WALSH TF DHANOA DM CHEN A BAGLEY SW FITCH KJ GREENLEE WJ
Citation: Dl. Williams et al., PHARMACOLOGY OF L-744,453, A NOVEL NONPEPTIDYL ENDOTHELIN ANTAGONIST, Life sciences, 58(14), 1996, pp. 1149-1157
2-HETEROCYCLIC INDOLE-3-SULFONES AS INHIBITORS OF HIV-1 REVERSE-TRANSCRIPTASE
Authors: YOUNG SD AMBLARD MC BRITCHER SF GREY VE TRAN LO LUMMA WC HUFF JR SCHLEIF WA EMINI EE OBRIEN JA PETTIBONE DJ
Citation: Sd. Young et al., 2-HETEROCYCLIC INDOLE-3-SULFONES AS INHIBITORS OF HIV-1 REVERSE-TRANSCRIPTASE, Bioorganic & medicinal chemistry letters, 5(5), 1995, pp. 491-496
NONPEPTIDE OXYTOCIN ANTAGONISTS - IDENTIFICATION AND SYNTHESIS OF A POTENT CAMPHOR AMINOSUCCINIMIDE
Authors: HOBBS DW GOULD NP HOFFMAN JB CLINESCHMIDT BV PETTIBONE DJ VEBER DF FREIDINGER RM
Citation: Dw. Hobbs et al., NONPEPTIDE OXYTOCIN ANTAGONISTS - IDENTIFICATION AND SYNTHESIS OF A POTENT CAMPHOR AMINOSUCCINIMIDE, Bioorganic & medicinal chemistry letters, 5(2), 1995, pp. 119-122
POTENT DUAL ANTAGONISTS OF ENDOTHELIN AND ANGIOTENSIN-II RECEPTORS DERIVED FROM ALPHA-PHENOXYPHENYLACETIC ACIDS .3.
Authors: WALSH TF FITCH KJ WILLIAMS DL MURPHY KL NOLAN NA PETTIBONE DJ CHANG RSL OMALLEY SS CLINESCHMIDT BV VEBER DF GREENLEE WJ
Citation: Tf. Walsh et al., POTENT DUAL ANTAGONISTS OF ENDOTHELIN AND ANGIOTENSIN-II RECEPTORS DERIVED FROM ALPHA-PHENOXYPHENYLACETIC ACIDS .3., Bioorganic & medicinal chemistry letters, 5(11), 1995, pp. 1155-1158
THE ROLE OF DRUG-METABOLISM IN DRUG DISCOVERY - A CASE-STUDY IN THE SELECTION OF AN OXYTOCIN RECEPTOR ANTAGONIST FOR DEVELOPMENT
Authors: CHIU SHL THOMPSON KA VINCENT SH ALVARO RF HUSKEY SEW STEARNS RA PETTIBONE DJ
Citation: Shl. Chiu et al., THE ROLE OF DRUG-METABOLISM IN DRUG DISCOVERY - A CASE-STUDY IN THE SELECTION OF AN OXYTOCIN RECEPTOR ANTAGONIST FOR DEVELOPMENT, Toxicologic pathology, 23(2), 1995, pp. 124-130
L-743,726 (DMP-266) - A NOVEL, HIGHLY POTENT NONNUCLEOSIDE INHIBITOR OF THE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE
Authors: YOUNG SD BRITCHER SF TRAN LO PAYNE LS LUMMA WC LYLE TA HUFF JR ANDERSON PS OLSEN DB CARROLL SS PETTIBONE DJ OBRIEN JA BALL RG BALANI SK LIN JH CHEN IW SCHLEIF WA SARDANA VV LONG WJ BYRNES VW EMINI EA
Citation: Sd. Young et al., L-743,726 (DMP-266) - A NOVEL, HIGHLY POTENT NONNUCLEOSIDE INHIBITOR OF THE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE, Antimicrobial agents and chemotherapy, 39(12), 1995, pp. 2602-2605
CHARACTERIZATION OF THE HUMAN OXYTOCIN RECEPTOR STABLY EXPRESSED IN 293 HUMAN EMBRYONIC KIDNEY-CELLS
Authors: JASPER JR HARRELL CM OBRIEN JA PETTIBONE DJ
Citation: Jr. Jasper et al., CHARACTERIZATION OF THE HUMAN OXYTOCIN RECEPTOR STABLY EXPRESSED IN 293 HUMAN EMBRYONIC KIDNEY-CELLS, Life sciences, 57(24), 1995, pp. 2253-2261
PHARMACOLOGY OF L-754,142, A HIGHLY POTENT, ORALLY-ACTIVE, NONPEPTIDYL ENDOTHELIN ANTAGONIST
Authors: WILLIAMS DL MURPHY KL NOLAN NA OBRIEN JA PETTIBONE DJ KIVLIGHN SD KRAUSE SM LIS EV ZINGARO GJ GABEL RA CLAYTON FC SIEGL PKS ZHANG K NAUE J VYAS K WALSH TF FITCH KJ CHAKRAVARTY PK GREENLEE WJ CLINESCHMIDT BV
Citation: Dl. Williams et al., PHARMACOLOGY OF L-754,142, A HIGHLY POTENT, ORALLY-ACTIVE, NONPEPTIDYL ENDOTHELIN ANTAGONIST, The Journal of pharmacology and experimental therapeutics, 275(3), 1995, pp. 1518-1526
ENZOYL]PIPERIDIN-4-YL)-4H-3,1-BENZOXAZIN-2(1H)-ONE (L-371,257) - A NEW, ORALLY BIOAVAILABLE, NONPEPTIDE OXYTOCIN ANTAGONIST
Authors: WILLIAMS PD CLINESCHMIDT BV ERB JM FREIDINGER RM GUIDOTTI MT LIS EV PAWLUCZYK JM PETTIBONE DJ REISS DR VEBER DF WOYDEN CJ
Citation: Pd. Williams et al., ENZOYL]PIPERIDIN-4-YL)-4H-3,1-BENZOXAZIN-2(1H)-ONE (L-371,257) - A NEW, ORALLY BIOAVAILABLE, NONPEPTIDE OXYTOCIN ANTAGONIST, Journal of medicinal chemistry, 38(23), 1995, pp. 4634-4636
)-YL)METHYL)SULFONYL)-4-(2-METHYLPHENYL)PIPERAZINE (L-368,899) - AN ORALLY BIOAVAILABLE, NONPEPTIDE OXYTOCIN ANTAGONIST WITH POTENTIAL UTILITY FOR MANAGING PRETERM LABOR
Authors: WILLIAMS PD ANDERSON PS BALL RG BOCK MG CARROLL L CHIU SHL CLINESCHMIDT BV CULBERSON JC ERB JM EVANS BE FITZPATRICK SL FREIDINGER RM KAUFMAN MJ LUNDELL GF MURPHY JS PAWLUCZYK JM PERLOW DS PETTIBONE DJ PITZENBERGER SM THOMPSON KL VEBER DF
Citation: Pd. Williams et al., )-YL)METHYL)SULFONYL)-4-(2-METHYLPHENYL)PIPERAZINE (L-368,899) - AN ORALLY BIOAVAILABLE, NONPEPTIDE OXYTOCIN ANTAGONIST WITH POTENTIAL UTILITY FOR MANAGING PRETERM LABOR, Journal of medicinal chemistry, 37(5), 1994, pp. 565-571
L-368,899, A POTENT ORALLY-ACTIVE OXYTOCIN ANTAGONIST FOR POTENTIAL USE IN PRETERM LABOR
Authors: PETTIBONE DJ CLINESCHMIDT BV GUIDOTTI MT LIS EV REISS DR WOYDEN CJ BOCK MG EVANS BE FREIDINGER RM HOBBS DW VEBER DF WILLIAMS PD CHIU SHL THOMPSON KL SCHORN TW SIEGL PKS KAUFMAN MJ CUKIERSKI MA HALUSKA GJ COOK MJ NOVY MJ
Citation: Dj. Pettibone et al., L-368,899, A POTENT ORALLY-ACTIVE OXYTOCIN ANTAGONIST FOR POTENTIAL USE IN PRETERM LABOR, Drug development research, 30(3), 1993, pp. 129-142
DEVELOPMENT AND PHARMACOLOGICAL ASSESSMENT OF NOVEL PEPTIDE AND NONPEPTIDE OXYTOCIN ANTAGONISTS
Authors: PETTIBONE DJ CLINESCHMIDT BV BOCK MG EVANS BE FREIDINGER RM VEBER DF WILLIAMS PD
Citation: Dj. Pettibone et al., DEVELOPMENT AND PHARMACOLOGICAL ASSESSMENT OF NOVEL PEPTIDE AND NONPEPTIDE OXYTOCIN ANTAGONISTS, Regulatory peptides, 45(1-2), 1993, pp. 289-293
NANOMOLAR-AFFINITY, NONPEPTIDE OXYTOCIN RECEPTOR ANTAGONISTS
Authors: EVANS BE LUNDELL GF GILBERT KF BOCK MG RITTLE KE CARROLL LA WILLIAMS PD PAWLUCZYK JM LEIGHTON JL YOUNG MB ERB JM HOBBS DW GOULD NP DIPARDO RM HOFFMAN JB PERLOW DS WHITTER WL VEBER DF PETTIBONE DJ CLINESCHMIDT BV ANDERSON PS FREIDINGER RM
Citation: Be. Evans et al., NANOMOLAR-AFFINITY, NONPEPTIDE OXYTOCIN RECEPTOR ANTAGONISTS, Journal of medicinal chemistry, 36(25), 1993, pp. 3993-4005
Risultati: 1-18 |