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Results: 1-24 |
Results: 24
1,4-BIS(ARYLSULFONYL)-1,2,3,4-TETRAHYDROPYRIDINES IN SYNTHESIS - HIGHLY REGIOSELECTIVE AND STEREOSELECTIVE S(N)1' AND ALKYLATION REACTIONS
Authors: CRAIG D MCCAGUE R POTTER GA WILLIAMS MRV
Citation: D. Craig et al., 1,4-BIS(ARYLSULFONYL)-1,2,3,4-TETRAHYDROPYRIDINES IN SYNTHESIS - HIGHLY REGIOSELECTIVE AND STEREOSELECTIVE S(N)1' AND ALKYLATION REACTIONS, Synlett, (1), 1998, pp. 55
1,4-BIS(ARYLSULFONYL)-1,2,3,4-TETRAHYDROPYRODINES IN SYNTHESIS - INTRAMOLECULAR ALKYLATION REACTIONS AND STEREOSELECTIVE SYNTHESIS OF ANTI-2,6-DISUBSTITUTED PIPERIDINES
Authors: CRAIG D MCCAGUE R POTTER GA WILLIAMS MRV
Citation: D. Craig et al., 1,4-BIS(ARYLSULFONYL)-1,2,3,4-TETRAHYDROPYRODINES IN SYNTHESIS - INTRAMOLECULAR ALKYLATION REACTIONS AND STEREOSELECTIVE SYNTHESIS OF ANTI-2,6-DISUBSTITUTED PIPERIDINES, Synlett, (1), 1998, pp. 58
DYNAMIC DIASTEREOMERIC SALT RESOLUTION OF NARWEDINE AND ITS TRANSFORMATION TO (-)-GALANTHAMINE
Authors: CHAPLIN DA JOHNSON NB PAUL JM POTTER GA
Citation: Da. Chaplin et al., DYNAMIC DIASTEREOMERIC SALT RESOLUTION OF NARWEDINE AND ITS TRANSFORMATION TO (-)-GALANTHAMINE, Tetrahedron letters, 39(37), 1998, pp. 6777-6780
17-(3-PYRIDYL)SUBSTITUTED IRREVERSIBLE INHIBITORS OF CYTOCHROME P450(17-ALPHA)
Authors: BARRIE SE POTTER GA JARMAN M
Citation: Se. Barrie et al., 17-(3-PYRIDYL)SUBSTITUTED IRREVERSIBLE INHIBITORS OF CYTOCHROME P450(17-ALPHA), British Journal of Cancer, 78, 1998, pp. 33-33
BIOCHEMISTRY AND PHARMACOKINETICS OF POTENT NONSTEROIDAL CYTOCHROME P450(17-ALPHA) INHIBITORS
Authors: BARRIE SE HAYNES BP POTTER GA CHAN FCY GODDARD PM DOWSETT M JARMAN M
Citation: Se. Barrie et al., BIOCHEMISTRY AND PHARMACOKINETICS OF POTENT NONSTEROIDAL CYTOCHROME P450(17-ALPHA) INHIBITORS, Journal of steroid biochemistry and molecular biology, 60(5-6), 1997, pp. 347-351
A CONVENIENT, LARGE-SCALE SYNTHESIS OF ABIRATERONE ACETATE 3-BETA-ACETOXY-17-(3-PYRIDYL)ANDROSTA-5,16-DIENE], A POTENTIAL NEW DRUG FOR THE TREATMENT OF PROSTATE-CANCER
Authors: POTTER GA HARDCASTLE IR JARMAN M
Citation: Ga. Potter et al., A CONVENIENT, LARGE-SCALE SYNTHESIS OF ABIRATERONE ACETATE 3-BETA-ACETOXY-17-(3-PYRIDYL)ANDROSTA-5,16-DIENE], A POTENTIAL NEW DRUG FOR THE TREATMENT OF PROSTATE-CANCER, Organic preparations and procedures international, 29(1), 1997, pp. 123-128
RHODIUM-CATALYZED ASYMMETRIC HYDROSILYLATION OF KETONES USING PHOSPHORUS-CONTAINING OXAZOLINE LIGANDS
Authors: NEWMAN LM WILLIAMS JMJ MCCAGUE R POTTER GA
Citation: Lm. Newman et al., RHODIUM-CATALYZED ASYMMETRIC HYDROSILYLATION OF KETONES USING PHOSPHORUS-CONTAINING OXAZOLINE LIGANDS, Tetrahedron : asymmetry, 7(6), 1996, pp. 1597-1598
OSCILLATING CRYSTALLIZATION OF (-) ENANTIOMERS DURING RESOLUTION BY ENTRAINMENT OF 2-AZABICYCLO[2.2.1]HEPT-5-EN-3-ONE() AND ()
Authors: POTTER GA GARCIA C MCCAGUE R ADGER B COLLET A
Citation: Ga. Potter et al., OSCILLATING CRYSTALLIZATION OF (-) ENANTIOMERS DURING RESOLUTION BY ENTRAINMENT OF 2-AZABICYCLO[2.2.1]HEPT-5-EN-3-ONE() AND (), Angewandte Chemie, International Edition in English, 35(15), 1996, pp. 1666-1668
3-PYRIDYLALKYL AND 4-PYRIDYLALKYL ADAMANTANECARBOXYLATES - INHIBITORSOF HUMAN CYTOCHROME P450(17-ALPHA) (17-ALPHA-HYDROXYLASE C-17,C-20-LYASE) - POTENTIAL NONSTEROIDAL AGENTS FOR THE TREATMENT OF PROSTATIC-CANCER/
Authors: CHAN FCY POTTER GA BARRIE SE HAYNES BP ROWLANDS MG HOUGHTON J JARMAN M
Citation: Fcy. Chan et al., 3-PYRIDYLALKYL AND 4-PYRIDYLALKYL ADAMANTANECARBOXYLATES - INHIBITORSOF HUMAN CYTOCHROME P450(17-ALPHA) (17-ALPHA-HYDROXYLASE C-17,C-20-LYASE) - POTENTIAL NONSTEROIDAL AGENTS FOR THE TREATMENT OF PROSTATIC-CANCER/, Journal of medicinal chemistry, 39(17), 1996, pp. 3319-3323
PHARMACOKINETICS AND BIODISTRIBUTION OF RADIOLABELED IDOXIFENE - PROSPECTS FOR THE USE OF PET IN THE EVALUATION OF A NOVEL ANTIESTROGEN FORCANCER-THERAPY
Authors: YOUNG H CARNOCHAN P TRIVEDI M POTTER GA ECCLES SA HAYNES BP JARMAN M OTT RJ
Citation: H. Young et al., PHARMACOKINETICS AND BIODISTRIBUTION OF RADIOLABELED IDOXIFENE - PROSPECTS FOR THE USE OF PET IN THE EVALUATION OF A NOVEL ANTIESTROGEN FORCANCER-THERAPY, Nuclear medicine and biology, 22(4), 1995, pp. 405-411
ACTIVE-SITE CONFORMATION OF 17-(3-PYRIDYL)ANDROSTA-5,16-DIEN-3-BETA-OL, A POTENT INHIBITOR OF THE P450 ENZYME C17-ALPHA-HYDROXYLASE C17-20 LYASE/
Authors: BURKE DF LAUGHTON CA SNOOK CF NEIDLE S POTTER GA JARMAN M
Citation: Df. Burke et al., ACTIVE-SITE CONFORMATION OF 17-(3-PYRIDYL)ANDROSTA-5,16-DIEN-3-BETA-OL, A POTENT INHIBITOR OF THE P450 ENZYME C17-ALPHA-HYDROXYLASE C17-20 LYASE/, Bioorganic & medicinal chemistry letters, 5(11), 1995, pp. 1125-1130
THE DEUTERIUM-ISOTOPE EFFECT FOR THE ALPHA-HYDROXYLATION OF TAMOXIFENBY RAT-LIVER MICROSOMES ACCOUNTS FOR THE REDUCED GENOTOXICITY OF [D-5-ETHYL]TAMOXIFEN
Authors: JARMAN M POON GK ROWLANDS MG GRIMSHAW RM HORTON MN POTTER GA MCCAGUE R
Citation: M. Jarman et al., THE DEUTERIUM-ISOTOPE EFFECT FOR THE ALPHA-HYDROXYLATION OF TAMOXIFENBY RAT-LIVER MICROSOMES ACCOUNTS FOR THE REDUCED GENOTOXICITY OF [D-5-ETHYL]TAMOXIFEN, Carcinogenesis, 16(4), 1995, pp. 683-688
ESTERS OF 3-PYRIDYLACETIC ACID THAT COMBINE POTENT INHIBITION OF 17-ALPHA-HYDROXYLASE C-17,C-20-LYASE (CYTOCHROME P45017-ALPHA) WITH RESISTANCE TO ESTERASE HYDROLYSIS
Authors: ROWLANDS MG BARRIE SE CHAN F HOUGHTON J JARMAN M MCCAGUE R POTTER GA
Citation: Mg. Rowlands et al., ESTERS OF 3-PYRIDYLACETIC ACID THAT COMBINE POTENT INHIBITION OF 17-ALPHA-HYDROXYLASE C-17,C-20-LYASE (CYTOCHROME P45017-ALPHA) WITH RESISTANCE TO ESTERASE HYDROLYSIS, Journal of medicinal chemistry, 38(21), 1995, pp. 4191-4197
RATIONALLY DESIGNED ANALOGS OF TAMOXIFEN WITH IMPROVED CALMODULIN ANTAGONISM
Authors: HARDCASTLE IR ROWLANDS MG HOUGHTON J PARR IB POTTER GA JARMAN M EDWARDS KJ LAUGHTON CA TRENT JO NEIDLE S
Citation: Ir. Hardcastle et al., RATIONALLY DESIGNED ANALOGS OF TAMOXIFEN WITH IMPROVED CALMODULIN ANTAGONISM, Journal of medicinal chemistry, 38(2), 1995, pp. 241-248
NOVEL STEROIDAL INHIBITORS OF HUMAN CYTOCHROME P450(17-ALPHA) (17-ALPHA-HYDROXYLASE-C-17,C-20-LYASE) - POTENTIAL AGENTS FOR THE TREATMENT OF PROSTATIC-CANCER
Authors: POTTER GA BARRIE SE JARMAN M ROWLANDS MG
Citation: Ga. Potter et al., NOVEL STEROIDAL INHIBITORS OF HUMAN CYTOCHROME P450(17-ALPHA) (17-ALPHA-HYDROXYLASE-C-17,C-20-LYASE) - POTENTIAL AGENTS FOR THE TREATMENT OF PROSTATIC-CANCER, Journal of medicinal chemistry, 38(13), 1995, pp. 2463-2471
IDOXIFENE - REPORT OF A PHASE-I STUDY IN PATIENTS WITH METASTATIC BREAST-CANCER
Authors: COOMBES RC HAYNES BP DOWSETT M QUIGLEY M ENGLISH J JUDSON IR GRIGGS LJ POTTER GA MCCAGUE R JARMAN M
Citation: Rc. Coombes et al., IDOXIFENE - REPORT OF A PHASE-I STUDY IN PATIENTS WITH METASTATIC BREAST-CANCER, Cancer research, 55(5), 1995, pp. 1070-1074
NEW LATERAL RESERVOIR FLASH CHROMATOGRAPHY SYSTEM FOR THE EXPEDITIOUSPREPARATIVE PURIFICATION OF ORGANIC-COMPOUNDS
Authors: POTTER GA
Citation: Ga. Potter, NEW LATERAL RESERVOIR FLASH CHROMATOGRAPHY SYSTEM FOR THE EXPEDITIOUSPREPARATIVE PURIFICATION OF ORGANIC-COMPOUNDS, Journal of chromatography, 675(1-2), 1994, pp. 237-239
PHARMACOLOGY OF NOVEL STEROIDAL INHIBITORS OF CYTOCHROME P450(17-ALPHA) (17-ALPHA-HYDROXYLASE C17-20 LYASE)
Authors: BARRIE SE POTTER GA GODDARD PM HAYNES BP DOWSETT M JARMAN M
Citation: Se. Barrie et al., PHARMACOLOGY OF NOVEL STEROIDAL INHIBITORS OF CYTOCHROME P450(17-ALPHA) (17-ALPHA-HYDROXYLASE C17-20 LYASE), Journal of steroid biochemistry and molecular biology, 50(5-6), 1994, pp. 267-273
SYNTHESIS OF [D5-ETHYL]-TAMOXIFEN - A MECHANISTIC PROBE OF TAMOXIFEN INDUCED HEPATIC DNA ADDUCT FORMATION
Authors: HORTON MN JARMAN M POTTER GA
Citation: Mn. Horton et al., SYNTHESIS OF [D5-ETHYL]-TAMOXIFEN - A MECHANISTIC PROBE OF TAMOXIFEN INDUCED HEPATIC DNA ADDUCT FORMATION, Journal of labelled compounds & radiopharmaceuticals, 34(8), 1994, pp. 767-772
SYNTHESIS OF 4-STANNYLATED TAMOXIFEN ANALOGS - USEFUL PRECURSORS TO RADIOLABELED IDOXIFENE AND AZIRIDINYL 4-IODOTAMOXIFEN
Authors: MCCAGUE R POTTER GA
Citation: R. Mccague et Ga. Potter, SYNTHESIS OF 4-STANNYLATED TAMOXIFEN ANALOGS - USEFUL PRECURSORS TO RADIOLABELED IDOXIFENE AND AZIRIDINYL 4-IODOTAMOXIFEN, Journal of labelled compounds & radiopharmaceuticals, 34(3), 1994, pp. 297-302
REDUCED GENOTOXICITY OF [D-5-ETHYL]-TAMOXIFEN IMPLICATES ALPHA-HYDROXYLATION OF THE ETHYL GROUP AS A MAJOR PATHWAY OF TAMOXIFEN ACTIVATION TO A LIVER CARCINOGEN
Authors: PHILLIPS DH POTTER GA HORTON MN HEWER A CROFTONSLEIGH C JARMAN M VENITT S
Citation: Dh. Phillips et al., REDUCED GENOTOXICITY OF [D-5-ETHYL]-TAMOXIFEN IMPLICATES ALPHA-HYDROXYLATION OF THE ETHYL GROUP AS A MAJOR PATHWAY OF TAMOXIFEN ACTIVATION TO A LIVER CARCINOGEN, Carcinogenesis, 15(8), 1994, pp. 1487-1492
A MECHANISTIC HYPOTHESIS FOR DNA ADDUCT FORMATION BY TAMOXIFEN FOLLOWING HEPATIC OXIDATIVE-METABOLISM
Authors: POTTER GA MCCAGUE R JARMAN M
Citation: Ga. Potter et al., A MECHANISTIC HYPOTHESIS FOR DNA ADDUCT FORMATION BY TAMOXIFEN FOLLOWING HEPATIC OXIDATIVE-METABOLISM, Carcinogenesis, 15(3), 1994, pp. 439-442
AN EFFICIENT, LARGE-SCALE SYNTHESIS OF IDOXIFENE ETHOXY]PHENYL]-1-(4-IODOPHENYL)-2-PHENYL-1-BUTENE)
Authors: MCCAGUE R POTTER GA JARMAN M
Citation: R. Mccague et al., AN EFFICIENT, LARGE-SCALE SYNTHESIS OF IDOXIFENE ETHOXY]PHENYL]-1-(4-IODOPHENYL)-2-PHENYL-1-BUTENE), Organic preparations and procedures international, 26(3), 1994, pp. 343-346
THE DIRECT FORMATION OF ESTERS OF 2-(4-PYRIDYL)PROPANOIC ACID BY REACTION OF A MELDRUM ACID-DERIVATIVE WITH LITHIUM ALKOXIDES
Authors: CHAN FCY POTTER GA JARMAN M
Citation: Fcy. Chan et al., THE DIRECT FORMATION OF ESTERS OF 2-(4-PYRIDYL)PROPANOIC ACID BY REACTION OF A MELDRUM ACID-DERIVATIVE WITH LITHIUM ALKOXIDES, Journal of chemical research. Synopses, (11), 1993, pp. 454-455
Risultati: 1-24 |