Authors:
Ryder, TR
Hu, LY
Rafferty, MF
Feng, MR
Lotarski, SM
Rock, DM
Stoehr, SJ
Taylor, CP
Weber, ML
Miljanich, GP
Millerman, E
Szoke, BG
Citation: Tr. Ryder et al., Synthesis and biological activity of 4-aminopiperidine derivatives as N-type calcium channel antagonists, MED CHEM RE, 10(1), 2000, pp. 11-18
Authors:
Hu, LY
Ryder, TR
Rafferty, MF
Taylor, CP
Feng, MR
Kuo, BS
Lotarski, SM
Miljanich, GP
Millerman, E
Siebers, KM
Szoke, BG
Citation: Ly. Hu et al., The discovery of [1-(4-dimethylamino-benzyl)-piperidin-4-yl]-[4-(3,3-dimethylbutyl)-phenyl]-(3-methyl-but-2-enyl)-amine, an N-type Ca+2 channel blocker with oral activity for analgesia, BIO MED CH, 8(6), 2000, pp. 1203-1212
Authors:
Song, YT
Bowersox, SS
Connor, DT
Dooley, DJ
Lotarski, SM
Malone, T
Miljanich, G
Millerman, E
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Rock, D
Roth, BD
Schmidt, J
Stoehr, S
Szoke, BG
Taylor, C
Vartanian, M
Wang, YX
Citation: Yt. Song et al., (S)-4-methyl-2-(methylamino)pentanoic acid [4,4-bis(4-fluorophenyl)butyl] amide hydrochloride, a novel calcium channel antagonist, is efficacious in several animal models of pain, J MED CHEM, 43(19), 2000, pp. 3474-3477
Authors:
Hu, LY
Ryder, TR
Nikam, SS
Millerman, E
Szoke, BG
Rafferty, MF
Citation: Ly. Hu et al., Synthesis and biological evaluation of substituted 4-(OBz)phenylalanine derivatives as novel N-type calcium channel blockers, BIOORG MED, 9(8), 1999, pp. 1121-1126
Authors:
Ryder, TR
Hu, LY
Rafferty, MF
Lotarski, SM
Rock, DM
Stoehr, SJ
Taylor, CP
Weber, ML
Miljanich, GP
Millerman, E
Szoke, BG
Citation: Tr. Ryder et al., Structure-activity relationship at the proximal phenyl group in a series of non-peptidyl N-type calcium channel antagonists, BIOORG MED, 9(16), 1999, pp. 2453-2458
Authors:
Hu, LY
Ryder, TR
Rafferty, MF
Dooley, DJ
Geer, JJ
Lotarski, SM
Miljanich, GP
Millerman, E
Rock, DM
Stoehr, SJ
Szoke, BG
Taylor, CP
Vartanian, MG
Citation: Ly. Hu et al., Structure-activity relationship of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockers, BIOORG MED, 9(15), 1999, pp. 2151-2156
Authors:
Ryder, TR
Hu, LY
Rafferty, MF
Millerman, E
Szoke, BG
Tarczy-Hornoch, K
Citation: Tr. Ryder et al., Multiple parallel synthesis of N,N-dialkyldipeptidylamines as N-type calcium channel blockers, BIOORG MED, 9(13), 1999, pp. 1813-1818
Citation: D. Flynn et Mf. Rafferty, Third Winter Conference on Medicinal and Bioorganic Chemistry Applicationsof Structural Biology to Drug Discovery - Editorial preface, MED RES REV, 19(4), 1999, pp. 271-271
Authors:
Hu, LY
Ryder, TR
Rafferty, MF
Feng, MR
Lotarski, SM
Rock, DM
Sinz, M
Stoehr, SJ
Taylor, CP
Weber, ML
Bowersox, SS
Miljanich, GP
Millerman, E
Wang, YX
Szoke, BG
Citation: Ly. Hu et al., Synthesis of a series of 4-benzyloxyaniline analogues as neuronal N-type calcium channel blockers with improved anticonvulsant and analgesic properties, J MED CHEM, 42(20), 1999, pp. 4239-4249
Authors:
Nikam, SS
Cordon, JJ
Ortwine, DF
Heimbach, TH
Blackburn, AC
Vartanian, MG
Nelson, CB
Schwarz, RD
Boxer, PA
Rafferty, MF
Citation: Ss. Nikam et al., Design and synthesis of novel quinoxaline-2,3-dione AMPA/Gly(N) receptor antagonists: Amino acid derivatives, J MED CHEM, 42(12), 1999, pp. 2266-2271