Authors:
Link, JT
Sorensen, B
Liu, G
Pei, ZH
Reilly, EB
Leitza, S
Okasinski, G
Citation: Jt. Link et al., Discovery and SAR of diarylsulfide cyclopropylamide LFA-1/LCAM-1 interaction antagonists, BIOORG MED, 11(8), 2001, pp. 973-976
Authors:
Liu, G
Huth, JR
Olejniczak, ET
Mendoza, R
DeVries, P
Leitza, S
Reilly, EB
Okasinski, GF
Fesik, SW
von Geldern, TW
Citation: G. Liu et al., Novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intracellular adhesion molecule-1 interaction. 2. Mechanism of inhibition and structure-based improvement of pharmaceutical properties, J MED CHEM, 44(8), 2001, pp. 1202-1210
Authors:
Winn, M
Reilly, EB
Liu, G
Huth, JR
Jae, HS
Freeman, J
Pei, ZH
Xin, ZL
Lynch, J
Kester, J
von Geldern, TW
Leitza, S
DeVries, P
Dickinson, R
Mussatto, D
Okasinski, GF
Citation: M. Winn et al., Discovery of novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intercellular adhesion molecule-1 interaction. 4. Structure-activity relationship of substituents on the benzene ring of the cinnamide, J MED CHEM, 44(25), 2001, pp. 4393-4403
Authors:
Pei, ZH
Xin, ZL
Liu, G
Li, YH
Reilly, EB
Lubbers, NL
Huth, JR
Link, JT
von Geldern, TW
Cox, BF
Leitza, S
Gao, Y
Marsh, KC
DeVries, P
Okasinski, GF
Citation: Zh. Pei et al., Discovery of potent antagonists of leukocyte function-associated antigen-1/intercellular adhesion molecule-1 interaction. 3. Amide (C-ring) structure-activity relationship and improvement of overall properties of arylthio cinnamides, J MED CHEM, 44(18), 2001, pp. 2913-2920
Authors:
Liu, G
Link, JT
Pei, ZH
Reilly, EB
Leitza, S
Nguyen, B
Marsh, KC
Okasinski, GF
von Geldern, TW
Ormes, M
Fowler, K
Gallatin, M
Citation: G. Liu et al., Discovery of novel p-arylthio cinnamides as antagonists of leukocyte function-associated antigen-1/intracellular adhesion molecule-1 interaction. 1. Identification of an additional binding pocket based on an anilino diaryl sulfide lead, J MED CHEM, 43(21), 2000, pp. 4025-4040