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BRITCHER SF
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PAYNE LS
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LYLE TA
HUFF JR
ANDERSON PS
OLSEN DB
CARROLL SS
PETTIBONE DJ
OBRIEN JA
BALL RG
BALANI SK
LIN JH
CHEN IW
SCHLEIF WA
SARDANA VV
LONG WJ
BYRNES VW
EMINI EA
Citation: Sd. Young et al., L-743,726 (DMP-266) - A NOVEL, HIGHLY POTENT NONNUCLEOSIDE INHIBITOR OF THE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE, Antimicrobial agents and chemotherapy, 39(12), 1995, pp. 2602-2605
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SCHLEIF WA
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SARDANA VV
SCHNEIDER CL
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ROTH E
WOLFGANG JA
HOFFMAN JM
SMITH AM
GELOTTE KM
EMINI EA
Citation: Wa. Schleif et al., ATTEMPTED PROPHYLAXIS OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 INFECTION IN CHIMPANZEES WITH A NONNUCLEOSIDE REVERSE-TRANSCRIPTASE INHIBITOR, AIDS research and human retroviruses, 10(1), 1994, pp. 107-110
Authors:
CONDRA JH
BLAHY OM
BUSH BL
CULBERSON C
GOTLIB L
GRAHAM DJ
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HOLLOWAY MK
LAFEMINA RL
QUINTERO JC
RHODES A
ROTH E
SARDANA VV
SCHNEIDER CL
SCHLABACH AJ
SCHLEIF WA
TITUS DL
WOLANSKI BS
WOLFGANG JA
EMINI EA
Citation: Jh. Condra et al., MUTATIONS IN HIV-1 PROTEASE RESIDUES AFFECTING SUSCEPTIBILITY TO L-735,524, Journal of cellular biochemistry, 1994, pp. 166-166
Authors:
EMINI EA
BYRNES VW
CONDRA JH
SCHLEIF WA
SARDANA VV
Citation: Ea. Emini et al., THE GENETIC AND FUNCTIONAL BASIS OF HIV-1 RESISTANCE TO NONNUCLEOSIDEREVERSE-TRANSCRIPTASE INHIBITORS, Archives of virology, 1994, pp. 11-17
Authors:
BYRNES VW
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SCHLEIF WA
CONDRA JH
SCHNEIDER CL
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WOLFGANG JA
GRAHAM DJ
GOTLIB L
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BLAHY OM
QUINTERO JC
RHODES A
ROTH E
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SARDANA VV
Citation: Vw. Byrnes et al., SUSCEPTIBILITIES OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 ENZYME AND VIRAL VARIANTS EXPRESSING MULTIPLE RESISTANCE-ENGENDERING AMINO-ACID SUBSTITUTIONS TO REVERSE-TRANSCRIPTASE INHIBITORS, Antimicrobial agents and chemotherapy, 38(6), 1994, pp. 1404-1407
Authors:
VACCA JP
DORSEY BD
SCHLEIF WA
LEVIN RB
MCDANIEL SL
DARKE PL
ZUGAY J
QUINTERO JC
BLAHY OM
ROTH E
SARDANA VV
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GRAHAM PI
CONDRA JH
GOTLIB L
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LIN J
CHEN IW
VASTAG K
OSTOVIC D
ANDERSON PS
EMINI EA
HUFF JR
Citation: Jp. Vacca et al., L-735,524 - AN ORALLY BIOAVAILABLE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 PROTEASE INHIBITOR, Proceedings of the National Academy of Sciences of the United Statesof America, 91(9), 1994, pp. 4096-4100
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KARLSSON A
SARDANA VV
EMINI EA
CAMARASA MJ
DECLERCQ E
Citation: J. Balzarini et al., HUMAN-IMMUNODEFICIENCY-VIRUS-1 (HIV-1)-SPECIFIC REVERSE-TRANSCRIPTASE(RT) INHIBITORS MAY SUPPRESS THE REPLICATION OF SPECIFIC DRUG-RESISTANT (E138K)RT HIV-1 MUTANTS OR SELECT FOR HIGHLY RESISTANT (Y181C-]C181I)RT HIV-1 MUTANTS, Proceedings of the National Academy of Sciences of the United Statesof America, 91(14), 1994, pp. 6599-6603
Authors:
SARDANA VV
WOLFGANG JA
VELOSKI CA
LONG WJ
LEGROW K
WOLANSKI B
EMINI EA
LAFEMINA RL
Citation: Vv. Sardana et al., PEPTIDE SUBSTRATE CLEAVAGE SPECIFICITY OF THE HUMAN CYTOMEGALOVIRUS PROTEASE, The Journal of biological chemistry, 269(20), 1994, pp. 14337-14340
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SARDANA VV
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CULBERSON JC
GOTLIB L
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SCHNEIDER CL
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WOLFGANG JA
EMINI EA
Citation: Vv. Sardana et al., HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 PROTEASE INHIBITORS - EVALUATION OF RESISTANCE ENGENDERED BY AMINO-ACID SUBSTITUTIONS IN THE ENZYMES SUBSTRATE-BINDING SITE, Biochemistry, 33(8), 1994, pp. 2004-2010
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SCHLEIF WA
SARDANA VV
BYRNES VW
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EMINI EA
Citation: Wa. Schleif et al., PREVENTION OF HIV-1 INFECTION IN CHIMPANZEES BY A NONNUCLEOSIDE REVERSE-TRANSCRIPTASE INHIBITOR, Journal of cellular biochemistry, 1993, pp. 23-23
Authors:
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CONDRA JH
SCHLEIF WA
SCHNEIDER CL
WATERBURY JA
WOLFGANG JA
GRAHAM DJ
GOTLIB L
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LONG WJ
RHODES A
TITUS DL
ROTH E
BLAHY OM
EMINI EA
Citation: Vw. Byrnes et al., HIV-1 REVERSE-TRANSCRIPTASE RESIDUES THAT INFLUENCE SENSITIVITY TO NONNUCLEOSIDE INHIBITORS, Journal of cellular biochemistry, 1993, pp. 75-75
Authors:
BYRNES VW
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SCHLEIF WA
CONDRA JH
WATERBURY JA
WOLFGANG JA
LONG WJ
SCHNEIDER CL
SCHLABACH AJ
WOLANSKI BS
GRAHAM DJ
GOTLIB L
RHODES A
TITUS DL
ROTH E
BLAHY OM
QUINTERO JC
STASZEWSKI S
EMINI EA
Citation: Vw. Byrnes et al., COMPREHENSIVE MUTANT ENZYME AND VIRAL VARIANT ASSESSMENT OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE RESISTANCE TO NONNUCLEOSIDE INHIBITORS, Antimicrobial agents and chemotherapy, 37(8), 1993, pp. 1576-1579
Authors:
GOLDMAN ME
OBRIEN JA
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SCHLEIF WA
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EMINI EA
Citation: Me. Goldman et al., A NONNUCLEOSIDE REVERSE-TRANSCRIPTASE INHIBITOR ACTIVE ON HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 ISOLATES RESISTANT TO RELATED INHIBITORS, Antimicrobial agents and chemotherapy, 37(5), 1993, pp. 947-949
Authors:
WILLIAMS TM
CICCARONE TM
MACTOUGH SC
ROONEY CS
BALANI SK
CONDRA JH
EMINI EA
GOLDMAN ME
GREENLEE WJ
KAUFFMAN LR
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SARDANA VV
SCHLEIF WA
THEOHARIDES AD
ANDERSON PS
Citation: Tm. Williams et al., 5-CHLORO-3-(PHENYLSULFONYL)INDOLE-2-CARBOXAMIDE - A NOVEL, NONNUCLEOSIDE INHIBITOR OF HIV-1 REVERSE-TRANSCRIPTASE, Journal of medicinal chemistry, 36(9), 1993, pp. 1291-1294