Authors:
POPPE SM
SLADE DE
CHONG KT
HINSHAW RR
PAGANO PJ
MARKOWITZ M
HO DD
MO H
GORMAN RR
DUEWEKE TJ
THAISRIVONGS S
TARPLEY WG
Citation: Sm. Poppe et al., ANTIVIRAL ACTIVITY OF THE DIHYDROPYRONE PNU-140690, A NEW NONPEPTIDICHUMAN-IMMUNODEFICIENCY-VIRUS PROTEASE INHIBITOR, Antimicrobial agents and chemotherapy, 41(5), 1997, pp. 1058-1063
Authors:
OLMSTED RA
SLADE DE
KOPTA LA
POPPE SM
POEL TJ
NEWPORT SW
RANK KB
BILES C
MORGE RA
DUEWEKE TJ
YAGI Y
ROMERO DL
THOMAS RC
SHARMA SK
TARPLEY WG
Citation: Ra. Olmsted et al., (ALKYLAMINO)PIPERIDINE BIS(HETEROARYL)PIPERIZINE ANALOGS ARE POTENT, BROAD-SPECTRUM NONNUCLEOSIDE REVERSE-TRANSCRIPTASE INHIBITORS OF DRUG-RESISTANT ISOLATES OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 (HIV-1) AND SELECT FOR DRUG-RESISTANT VARIANTS OF HIV-1(IIIB) WITH REDUCED REPLICATION PHENOTYPES, Journal of virology, 70(6), 1996, pp. 3698-3705
Authors:
THAISRIVONGS S
SKULNICK HI
TURNER SR
STROHBACH JW
TOMMASI RA
JOHNSON PD
ARISTOFF PA
JUDGE TM
GAMMILL RB
MORRIS JK
ROMINES KR
CHRUSCIEL RA
HINSHAW RR
CHONG KT
TARPLEY WG
POPPE SM
SLADE DE
LYNN JC
HORNG MM
TOMICH PK
SEEST EP
DOLAK LA
HOWE WJ
HOWARD GM
SCHWENDE FJ
TOTH LN
PADBURY GE
WILSON GJ
SHIOU LH
ZIPP GL
WILKINSON KF
RUSH BD
RUWART MJ
KOEPLINGER KA
ZHAO ZY
COLE S
ZAYA RM
KAKUK TJ
JANAKIRAMAN MN
WATENPAUGH KD
Citation: S. Thaisrivongs et al., STRUCTURE-BASED DESIGN OF HIV PROTEASE INHIBITORS - SULFONAMIDE-CONTAINING 5,6-DIHYDRO-4-HYDROXY-2-PYRONES AS NONPEPTIDIC INHIBITORS, Journal of medicinal chemistry, 39(22), 1996, pp. 4349-4353
Authors:
FAN NS
RANK KB
SLADE DE
POPPE SM
EVANS DB
KOPTA LA
OLMSTED RA
THOMAS RC
TARPLEY WG
SHARMA SK
Citation: Ns. Fan et al., A DRUG-RESISTANCE MUTATION IN THE INHIBITOR BINDING POCKET OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVERSE-TRANSCRIPTASE IMPAIRS DNA-SYNTHESIS AND RNA DEGRADATION, Biochemistry, 35(30), 1996, pp. 9737-9745
Authors:
SHARMA SK
FAN N
RANK KB
KOPTA LA
OLMSTED RA
POPPE SM
SLADE DE
THOMAS RC
TARPLEY WG
Citation: Sk. Sharma et al., A DRUG-RESISTANCE MUTATION (G190E) IN THE INHIBITOR BINDING POCKET IMPAIRS BOTH RNA-DEPENDENT DNA-POLYMERASE AND RIBONUCLEASE-H ACTIVITIES OF HIV-1 REVERSE-TRANSCRIPTASE, Journal of acquired immune deficiency syndromes and human retrovirology, 10, 1995, pp. 2-2