Authors:
MAGNIN DR
BILLER SA
CHEN Y
DICKSON JK
FRYSZMAN OM
LAWRENCE RM
LOGAN JVH
SIEBERMCMASTER ES
SULSKY RB
TRAEGER SC
HSIEH DC
LAN SJ
RINEHART JK
HARRITY TW
JOLIBOIS KG
KUNSELMAN LK
RICH LC
SLUSARCHYK DA
CIOSEK CP
Citation: Dr. Magnin et al., ALPHA-PHOSPHONOSULFONIC ACIDS - POTENT AND SELECTIVE INHIBITORS OF SQUALENE SYNTHASE, Journal of medicinal chemistry, 39(3), 1996, pp. 657-660
Authors:
LAWRENCE RM
BILLER SA
DICKSON JK
LOGAN JVH
MAGNIN DR
SULSKY RB
DIMARCO JD
GOUGOUTAS JZ
BEYER BD
TAYLOR SC
LAN SJ
CIOSEK CP
HARRITY TW
JOLIBOIS KG
KUNSELMAN LK
SLUSARCHYK DA
Citation: Rm. Lawrence et al., ENANTIOSELECTIVE SYNTHESIS OF ALPHA-PHOSPHONO SULFONATE SQUALENE SYNTHASE INHIBITORS - CHIRAL RECOGNITION IN THE INTERACTIONS OF AN ALPHA-PHOSPHONO SULFONATE INHIBITOR WITH SQUALENE SYNTHASE, Journal of the American Chemical Society, 118(46), 1996, pp. 11668-11669
Authors:
MAGNIN DR
BILLER SA
DICKSON JK
LOGAN JV
LAWRENCE RM
CHEN Y
SULSKY RB
CIOSEK CP
HARRITY TW
JOLIBOIS KG
KUNSELMAN LK
RICH LC
SLUSARCHYK DA
Citation: Dr. Magnin et al., 1,1-BISPHOSPHONATE SQUALENE SYNTHASE INHIBITORS - INTERPLAY BETWEEN THE ISOPRENOID SUBUNIT AND THE DIPHOSPHATE SURROGATE, Journal of medicinal chemistry, 38(14), 1995, pp. 2596-2605
Authors:
HARRITY TW
GEORGE RJ
CIOSEK CP
BILLER SA
CHEN Y
DICKSON JK
FRYSZMAN OM
JOLIBOIS KJ
KUNSELMAN LK
LAWRENCE RM
LOGAN JV
MAGNIN DR
RICH LC
SLUSARCHYK DA
SULSKY RB
GREGG RE
Citation: Tw. Harrity et al., BMS-188494, AN ORALLY-ACTIVE SQUALENE SYNTHASE INHIBITOR PRODRUG, POTENTLY LOWERS PLASMA-CHOLESTEROL AND TRIGLYCERIDES IN RATS, HAMSTERS AND PRIMATES, Circulation, 92(8), 1995, pp. 484-484
Authors:
CIOSEK CP
MAGNIN DR
HARRITY TW
LOGAN JVH
DICKSON JK
GORDON EM
HAMILTON KA
JOLIBOIS KG
KUNSELMAN LK
LAWRENCE RM
MOOKHTIAR KA
RICH LC
SLUSARCHYK DA
SULSKY RB
BILLER SA
Citation: Cp. Ciosek et al., LIPOPHILIC 1,1-BISPHOSPHONATES ARE POTENT SQUALENE SYNTHASE INHIBITORS AND ORALLY-ACTIVE CHOLESTEROL-LOWERING AGENTS IN-VIVO, The Journal of biological chemistry, 268(33), 1993, pp. 24832-24837