Authors:
BRADY SF
STAUFFER KJ
LUMMA WC
SMITH GM
RAMJIT HG
LEWIS SD
LUCAS BJ
GARDELL SJ
LYLE EA
APPLEBY SD
COOK JJ
HOLAHAN MA
STRANIERI MT
LYNCH JJ
LIN JH
CHEN IW
VASTAG K
NAYLOROLSEN AM
VACCA JP
Citation: Sf. Brady et al., DISCOVERY AND DEVELOPMENT OF THE NOVEL POTENT ORALLY-ACTIVE THROMBIN INHIBITOR N-(9-HYDROXY-9-FLUORENECARBOXY)PROLYL TRANS-4-AMINOCYCLOHEXYLMETHYL AMIDE (L-372,460) - COAPPLICATION OF STRUCTURE-BASED DESIGN AND RAPID MULTIPLE ANALOG SYNTHESIS ON SOLID SUPPORT, Journal of medicinal chemistry, 41(3), 1998, pp. 401-406
Authors:
TUCKER TJ
BRADY SF
LUMMA WC
LEWIS SD
GARDELL SJ
NAYLOROLSEN AM
YAN YW
SISKO JT
STAUFFER KJ
LUCAS BJ
LYNCH JJ
COOK JJ
STRANIERI MT
HOLAHAN MA
LYLE EA
BASKIN EP
CHEN IW
DANCHECK KB
KRUEGER JA
COOPER CM
VACCA JP
Citation: Tj. Tucker et al., DESIGN AND SYNTHESIS OF A SERIES OF POTENT AND ORALLY BIOAVAILABLE NONCOVALENT THROMBIN INHIBITORS THAT UTILIZE NONBASIC GROUPS IN THE P1 POSITION, Journal of medicinal chemistry, 41(17), 1998, pp. 3210-3219
Authors:
LEWIS SD
NG AS
LYLE EA
MELLOTT MJ
APPLEBY SD
BRADY SF
STAUFFER KJ
SISKO JT
MAO SS
VEBER DF
NUTT RF
LYNCH JJ
COOK JJ
GARDELL SJ
SHAFER JA
Citation: Sd. Lewis et al., INHIBITION OF THROMBIN BY PEPTIDES CONTAINING LYSYL-ALPHA-KETO CARBONYL DERIVATIVES, Thrombosis and haemostasis, 74(4), 1995, pp. 1107-1112