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Results: 1-25 | 26-48 |
Results: 26-48/48
High constitutive activity of native H-3 receptors regulates histamine neurons in brain
Authors: Morisset, S Rouleau, A Ligneau, X Gbahou, F Tardivel-Lacombe, J Stark, H Schunack, W Ganellin, CR Schwartz, JC Arrang, JM
Citation: S. Morisset et al., High constitutive activity of native H-3 receptors regulates histamine neurons in brain, NATURE, 408(6814), 2000, pp. 860-864
Anti-inflammatory and antinociceptive properties of BP 2-94, a histamine H-3-receptor agonist prodrug
Authors: Rouleau, A Stark, H Schunack, W Schwartz, JC
Citation: A. Rouleau et al., Anti-inflammatory and antinociceptive properties of BP 2-94, a histamine H-3-receptor agonist prodrug, J PHARM EXP, 295(1), 2000, pp. 219-225
Histaprodifens: Synthesis, pharmacological in vitro evaluation, and molecular modeling of a new class of highly active and selective histamine H-1-receptor agonists
Authors: Elz, S Kramer, K Pertz, HH Detert, H ter Laak, AM Kuhne, R Schunack, W
Citation: S. Elz et al., Histaprodifens: Synthesis, pharmacological in vitro evaluation, and molecular modeling of a new class of highly active and selective histamine H-1-receptor agonists, J MED CHEM, 43(6), 2000, pp. 1071-1084
Novel histamine H-3-receptor antagonists with carbonyl-substituted 4-(3-(phenoxy)propyl)-1H-imidazole structures like ciproxifan and related compounds
Authors: Stark, H Sadek, B Krause, M Huls, A Ligneau, X Ganellin, CR Arrang, JM Schwartz, JC Schunack, W
Citation: H. Stark et al., Novel histamine H-3-receptor antagonists with carbonyl-substituted 4-(3-(phenoxy)propyl)-1H-imidazole structures like ciproxifan and related compounds, J MED CHEM, 43(21), 2000, pp. 3987-3994
New histamine H-3-receptor ligands of the proxifan series: Imoproxifan andother selective antagonists with high oral in vivo potency
Authors: Sasse, A Sadek, B Ligneau, X Elz, S Pertz, HH Luger, P Ganellin, CR Arrang, JM Schwartz, JC Schunack, W Stark, H
Citation: A. Sasse et al., New histamine H-3-receptor ligands of the proxifan series: Imoproxifan andother selective antagonists with high oral in vivo potency, J MED CHEM, 43(17), 2000, pp. 3335-3343
Distinct pharmacology of rat and human histamine H-3 receptors: role of two amino acids in the third transmembrane domain
Authors: Ligneau, X Morisset, S Tardivel-Lacombe, J Gbahou, F Ganellin, CR Stark, H Schunack, W Schwartz, JC Arrang, JM
Citation: X. Ligneau et al., Distinct pharmacology of rat and human histamine H-3 receptors: role of two amino acids in the third transmembrane domain, BR J PHARM, 131(7), 2000, pp. 1247-1250
Histamine H-3-receptor antagonists inhibit gastroprotection by (R)-alpha-methylhistamine in the rat
Authors: Morini, G Grandi, D Stark, HB Schunack, W
Citation: G. Morini et al., Histamine H-3-receptor antagonists inhibit gastroprotection by (R)-alpha-methylhistamine in the rat, BR J PHARM, 129(8), 2000, pp. 1597-1600
Utility of isotachophoresis-capillary zone electrophoresis, mass spectrometry and high-performance size-exclusion chromatography for monitoring of interleukin-6 dimer formation
Authors: Gysler, J Mazereeuw, M Helk, B Heitzmann, M Jaehde, U Schunack, W Tjaden, UR van der Greef, J
Citation: J. Gysler et al., Utility of isotachophoresis-capillary zone electrophoresis, mass spectrometry and high-performance size-exclusion chromatography for monitoring of interleukin-6 dimer formation, J CHROMAT A, 841(1), 1999, pp. 63-73
Monitoring of chemotherapy-induced proteinuria using capillary zone electrophoresis
Authors: Gysler, J Schunack, W Jaehde, U
Citation: J. Gysler et al., Monitoring of chemotherapy-induced proteinuria using capillary zone electrophoresis, J CHROMAT B, 721(2), 1999, pp. 207-216
Radiosynthesis and biodistribution of I-123-labeled antagonists of the histamine H-3 receptor as potential SPECT ligands
Authors: Windhorst, AD Timmerman, H Klok, RP Custers, FGJ Menge, WMPB Leurs, R Stark, H Schunack, W Gielen, EGJ van Kroonenburgh, MJPG Herscheid, JDM
Citation: Ad. Windhorst et al., Radiosynthesis and biodistribution of I-123-labeled antagonists of the histamine H-3 receptor as potential SPECT ligands, NUCL MED BI, 26(6), 1999, pp. 651-659
Electromigration peak dispersion of isotachophoretic protein zones during capillary zone electrophoresis
Authors: Gysler, J Jaehde, U Schunack, W
Citation: J. Gysler et al., Electromigration peak dispersion of isotachophoretic protein zones during capillary zone electrophoresis, FRESEN J AN, 365(5), 1999, pp. 398-403
Pharmacokinetic and pharmacodynamic comparison of two doses of calcium folinate combined with continuous fluorouracil infusion in patients with advanced colorectal cancer
Authors: Stremetzne, S Streit, M Kreuser, ED Schunack, W Jaehde, U
Citation: S. Stremetzne et al., Pharmacokinetic and pharmacodynamic comparison of two doses of calcium folinate combined with continuous fluorouracil infusion in patients with advanced colorectal cancer, PHARM WORLD, 21(4), 1999, pp. 184-189
Development and application of a simple assay to quantify cellular adductsof platinum complexes with DNA
Authors: Kloft, C Eickhoff, C Schulze-Forster, K Maurer, HR Schunack, W Jaehde, U
Citation: C. Kloft et al., Development and application of a simple assay to quantify cellular adductsof platinum complexes with DNA, PHARM RES, 16(3), 1999, pp. 470-473
Non-peptide G-protein activators as promising tools in cell biology and potential drug leads
Authors: Nurnberg, B Togel, W Krause, G Storm, R Breitweg-Lehmann, E Schunack, W
Citation: B. Nurnberg et al., Non-peptide G-protein activators as promising tools in cell biology and potential drug leads, EUR J MED C, 34(1), 1999, pp. 5-30
Determination of platinum complexes in clinical samples by a rapid flameless atomic absorption spectrometry assay
Authors: Kloft, C Appelius, H Siegert, W Schunack, W Jaehde, U
Citation: C. Kloft et al., Determination of platinum complexes in clinical samples by a rapid flameless atomic absorption spectrometry assay, THER DRUG M, 21(6), 1999, pp. 631-637
New synthesis of roxatidine acetate
Authors: Tarpanov, V Vlahov, R Penkov, M Krikorian, D Parushev, S Mechkarova, P Angelova, N Schunack, W
Citation: V. Tarpanov et al., New synthesis of roxatidine acetate, SYN COMMUN, 29(1), 1999, pp. 15-20
Stereoselective inhibition of ethanol-induced gastric lesions in the rat by the H-3-receptor agonist (R)-alpha-methylhistamine and its (S)-configuredisomer
Authors: Morini, G Grandi, D Bertaccini, G Leschke, C Schunack, W
Citation: G. Morini et al., Stereoselective inhibition of ethanol-induced gastric lesions in the rat by the H-3-receptor agonist (R)-alpha-methylhistamine and its (S)-configuredisomer, PHARMACOL, 59(4), 1999, pp. 192-200
Histaprodifen, methylhistaprodifen, and dimethylhistaprodifen are potent H-1-receptor agonists in the pithed and in the anaesthetized rat
Authors: Malinowska, B Piszcz, J Schlicker, E Kramer, K Elz, S Schunack, W
Citation: B. Malinowska et al., Histaprodifen, methylhistaprodifen, and dimethylhistaprodifen are potent H-1-receptor agonists in the pithed and in the anaesthetized rat, N-S ARCH PH, 359(1), 1999, pp. 11-16
Development of chiral N-alkylcarbamates as new leads for potent and selective H-3-receptor antagonists: Synthesis, capillary electrophoresis, and in vitro and oral in vivo activity
Authors: Sasse, A Kiec-Kononowicz, K Stark, H Motyl, M Reidemeister, S Ganellin, CR Ligneau, X Schwartz, JC Schunack, W
Citation: A. Sasse et al., Development of chiral N-alkylcarbamates as new leads for potent and selective H-3-receptor antagonists: Synthesis, capillary electrophoresis, and in vitro and oral in vivo activity, J MED CHEM, 42(4), 1999, pp. 593-600
Novel partial agonists for the histamine H-3 receptor with high in vitro and in vivo activity
Authors: Sasse, A Stark, H Reidemeister, S Huls, A Elz, S Ligneau, X Ganellin, CR Schwartz, JC Schunack, W
Citation: A. Sasse et al., Novel partial agonists for the histamine H-3 receptor with high in vitro and in vivo activity, J MED CHEM, 42(20), 1999, pp. 4269-4274
Synthesis of potent non-imidazole histamine H-3-receptor antagonists
Authors: Ganellin, CR Leurquin, F Piripitsi, A Arrang, JM Garbarg, M Ligneau, X Schunack, W Schwartz, JC
Citation: Cr. Ganellin et al., Synthesis of potent non-imidazole histamine H-3-receptor antagonists, ARCH PHARM, 331(12), 1998, pp. 395-404
Medicinal chemistry of histamine H-3 receptor agonists
Authors: Krause, M Stark, H Schunack, W
Citation: M. Krause et al., Medicinal chemistry of histamine H-3 receptor agonists, PHARMCHEM L, 30, 1998, pp. 175-196
Ciproxifan and chemically related compounds are highly potent and selective histamine H-3-receptor antagonists
Authors: Kathmann, M Schlicker, E Marr, L Werthwein, S Stark, H Schunack, W
Citation: M. Kathmann et al., Ciproxifan and chemically related compounds are highly potent and selective histamine H-3-receptor antagonists, N-S ARCH PH, 358(6), 1998, pp. 623-627
Risultati: 1-25 | 26-48 |