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Results: 1-11 |
Results: 11
Cystatins as calpain inhibitors: Engineered chicken cystatin- and stefin B-kininogen domain 2 hybrids support a cystatin-like mode of interaction with the catalytic subunit of mu-calpain
Authors: Diaz, BG Gross, S Assfalg-Machleidt, I Pfeiler, D Gollmitzer, N Gabrijelcic-Geiger, D Stubbs, MT Fritz, H Auerswald, EA Machledit, W
Citation: Bg. Diaz et al., Cystatins as calpain inhibitors: Engineered chicken cystatin- and stefin B-kininogen domain 2 hybrids support a cystatin-like mode of interaction with the catalytic subunit of mu-calpain, BIOL CHEM, 382(1), 2001, pp. 97-107
Synthesis and evaluation of diazine containing bioisosteres of (-)-ferruginine as ligands for nicotinic acetylcholine receptors
Authors: Gundisch, D Harms, K Schwarz, S Seitz, G Stubbs, MT Wegge, T
Citation: D. Gundisch et al., Synthesis and evaluation of diazine containing bioisosteres of (-)-ferruginine as ligands for nicotinic acetylcholine receptors, BIO MED CH, 9(10), 2001, pp. 2683-2691
Syntheses and evaluation of halogenated cytisine derivatives and of bioisosteric thiocytisine as potent and selective nAChR ligands
Authors: Imming, P Klaperski, P Stubbs, MT Seitz, G Gundisch, D
Citation: P. Imming et al., Syntheses and evaluation of halogenated cytisine derivatives and of bioisosteric thiocytisine as potent and selective nAChR ligands, EUR J MED C, 36(4), 2001, pp. 375-388
Factorising ligand affinity: A combined thermodynamic and crystallographicstudy of trypsin and thrombin inhibition
Authors: Dullweber, F Stubbs, MT Musil, D Sturzebecher, J Klebe, G
Citation: F. Dullweber et al., Factorising ligand affinity: A combined thermodynamic and crystallographicstudy of trypsin and thrombin inhibition, J MOL BIOL, 313(3), 2001, pp. 593-614
A new target for shigellosis: Rational design and crystallographic studiesof inhibitors of tRNA-guanine transglycosylase
Authors: Gradler, U Gerber, HD Goodenough-Lashua, DM Garcia, GA Ficner, R Reuter, K Stubbs, MT Klebe, G
Citation: U. Gradler et al., A new target for shigellosis: Rational design and crystallographic studiesof inhibitors of tRNA-guanine transglycosylase, J MOL BIOL, 306(3), 2001, pp. 455-467
exo-2-(pyridazin-4-yl)-7-azalbicyclo[2.2.1]heptanes: Syntheses and nicotinic acetylcholine receptor agonist activity of potent pyridazine analogues of (+/-)-epibatidine
Authors: Che, DQ Wegge, T Stubbs, MT Seitz, G Meier, H Methfessel, C
Citation: Dq. Che et al., exo-2-(pyridazin-4-yl)-7-azalbicyclo[2.2.1]heptanes: Syntheses and nicotinic acetylcholine receptor agonist activity of potent pyridazine analogues of (+/-)-epibatidine, J MED CHEM, 44(1), 2001, pp. 47-57
3-amidinophenylalanine-based inhibitors of urokinase
Authors: Sturzebecher, J Vieweg, H Steinmetzer, T Schweinitz, A Stubbs, MT Renatus, M Wikstrom, P
Citation: J. Sturzebecher et al., 3-amidinophenylalanine-based inhibitors of urokinase, BIOORG MED, 9(21), 1999, pp. 3147-3152
Crystal structures of the membrane-binding C2 domain of human coagulation factor V
Authors: Macedo-Ribeiro, S Bode, W Huber, R Quinn-Allen, MA Kim, SW Ortel, TL Bourenkov, GP Bartunik, HD Stubbs, MT Kane, WH Fuentes-Prior, P
Citation: S. Macedo-ribeiro et al., Crystal structures of the membrane-binding C2 domain of human coagulation factor V, NATURE, 402(6760), 1999, pp. 434-439
The structure of the human beta II-tryptase tetramer: Fo(u)r better or worse
Authors: Sommerhoff, CP Bode, W Pereira, PJB Stubbs, MT Sturzebecher, J Piechottka, GP Matschiner, G Bergner, A
Citation: Cp. Sommerhoff et al., The structure of the human beta II-tryptase tetramer: Fo(u)r better or worse, P NAS US, 96(20), 1999, pp. 10984-10991
Mutagenesis and crystallographic studies of Zymomonas mobilis tRNA-guaninetransglycosylase to elucidate the role of serine 103 for enzymatic activity
Authors: Gradler, U Ficner, R Garcia, GA Stubbs, MT Klebe, G Reuter, K
Citation: U. Gradler et al., Mutagenesis and crystallographic studies of Zymomonas mobilis tRNA-guaninetransglycosylase to elucidate the role of serine 103 for enzymatic activity, FEBS LETTER, 454(1-2), 1999, pp. 142-146
Structural and functional analyses of benzamidine-based inhibitors in complex with trypsin: Implications for the inhibition of factor Xa, tPA, and urokinase
Authors: Renatus, M Bode, W Huber, R Sturzebecher, J Stubbs, MT
Citation: M. Renatus et al., Structural and functional analyses of benzamidine-based inhibitors in complex with trypsin: Implications for the inhibition of factor Xa, tPA, and urokinase, J MED CHEM, 41(27), 1998, pp. 5445-5456
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