Authors:
MORTLOCK AA
BATH C
BUTLIN RJ
HEYS C
HUNT SJ
REID AC
SUMNER NF
TANG EK
WHITING E
WILSON C
WRIGHT ND
Citation: Aa. Mortlock et al., (3-METHOXY-5-METHYLPYRAZIN-2-YLSULFAMOYL)BENZAMIDE - ONE OF A CLASS OF NOVEL BENZENESULFONAMIDES WHICH ARE ORALLY-ACTIVE, ETA-SELECTIVE ENDOTHELIN ANTAGONISTS, Bioorganic & medicinal chemistry letters, 7(11), 1997, pp. 1399-1402
Authors:
BRADBURY RH
BATH C
BUTLIN RJ
DENNIS M
HEYS C
HUNT SJ
JAMES R
MORTLOCK AA
SUMNER NF
TANG EK
TELFORD B
WHITING E
WILSON C
Citation: Rh. Bradbury et al., NEW NONPEPTIDE ENDOTHELIN-A RECEPTOR ANTAGONISTS - SYNTHESIS, BIOLOGICAL PROPERTIES, AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF DIMETHYLAMINO)-N-PYRIDYL-1-NAPHTHALENESULFONAMIDE, THYLAMINO)-N-PYRIMIDINYL-1-NAPHTHALENESULFONAMIDE, THYLAMINO)-N-PYRIDAZINYL-1-NAPHTHALENESULFONAMIDE, AND IMETHYLAMINO)-N-PYRAZINYL-1-NAPHTHALENESULFONAMIDE, Journal of medicinal chemistry, 40(6), 1997, pp. 996-1004
Authors:
MCLEAN JS
KRUGER H
SWIFT D
TANG EK
BRENNAND JC
Citation: Js. Mclean et al., CELL-BASED ASSAY FOR FUNCTIONAL SCREENING OF COMPOUNDS ACTIVE AT THE HUMAN ENDOTHELIN A RECEPTOR, Journal of cardiovascular pharmacology, 26(6), 1995, pp. 978-982