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Results: 1-8 |
Results: 8
SERUM-PROTEIN BINDING OF HISTAMINE H-1-ANTAGONISTS - A COMPARATIVE-STUDY ON THE SERUM-PROTEIN BINDING OF A SEDATING ([H-3]MEPYRAMINE) AND ANONSEDATING H-1-ANTAGONIST ([H-3]LORATADINE)
Authors: TERLAAK AM BIJLOO GJ FISCHER MJE OPDENKELDER GMD WILTING J TIMMERMAN H
Citation: Am. Terlaak et al., SERUM-PROTEIN BINDING OF HISTAMINE H-1-ANTAGONISTS - A COMPARATIVE-STUDY ON THE SERUM-PROTEIN BINDING OF A SEDATING ([H-3]MEPYRAMINE) AND ANONSEDATING H-1-ANTAGONIST ([H-3]LORATADINE), European journal of pharmaceutical sciences, 4(5), 1996, pp. 307-319
MODELING AND MUTATION STUDIES ON THE HISTAMINE H-1-RECEPTOR AGONIST BINDING-SITE REVEAL DIFFERENT BINDING MODES FOR H-1-AGONISTS - ASP(116)(TM3) HAS A CONSTITUTIVE ROLE IN RECEPTOR STIMULATION
Authors: TERLAAK AM TIMMERMAN H LEURS R NEDERKOORN PHJ SMIT MJ DENKELDER GMDO
Citation: Am. Terlaak et al., MODELING AND MUTATION STUDIES ON THE HISTAMINE H-1-RECEPTOR AGONIST BINDING-SITE REVEAL DIFFERENT BINDING MODES FOR H-1-AGONISTS - ASP(116)(TM3) HAS A CONSTITUTIVE ROLE IN RECEPTOR STIMULATION, Journal of computer-aided molecular design, 9(4), 1995, pp. 319-330
COMPARATIVE-EVALUATION OF THE PREDICTIVE POWER OF CALCULATION PROCEDURES FOR MOLECULAR LIPOPHILICITY
Authors: MANNHOLD R REKKER RF SONNTAG C TERLAAK AM DROSS K POLYMEROPOULOS EE
Citation: R. Mannhold et al., COMPARATIVE-EVALUATION OF THE PREDICTIVE POWER OF CALCULATION PROCEDURES FOR MOLECULAR LIPOPHILICITY, Journal of pharmaceutical sciences, 84(12), 1995, pp. 1410-1419
THE HISTAMINE H-1-RECEPTOR ANTAGONIST BINDING-SITE - A STEREOSELECTIVE PHARMACOPHORIC MODEL-BASED UPON (SEMI-)RIGID H-1-ANTAGONISTS AND INCLUDING A KNOWN INTERACTION SITE ON THE RECEPTOR
Authors: TERLAAK AM VENHORST J DENKELDER GMDO TIMMERMAN H
Citation: Am. Terlaak et al., THE HISTAMINE H-1-RECEPTOR ANTAGONIST BINDING-SITE - A STEREOSELECTIVE PHARMACOPHORIC MODEL-BASED UPON (SEMI-)RIGID H-1-ANTAGONISTS AND INCLUDING A KNOWN INTERACTION SITE ON THE RECEPTOR, Journal of medicinal chemistry, 38(17), 1995, pp. 3351-3360
LYSINE(200) LOCATED IN THE 5TH TRANSMEMBRANE DOMAIN OF THE HISTAMINE H-1 RECEPTOR INTERACTS WITH HISTAMINE BUT NOT WITH ALL H-1 AGONISTS
Authors: LEURS R SMIT MJ MEEDER R TERLAAK AM TIMMERMAN H
Citation: R. Leurs et al., LYSINE(200) LOCATED IN THE 5TH TRANSMEMBRANE DOMAIN OF THE HISTAMINE H-1 RECEPTOR INTERACTS WITH HISTAMINE BUT NOT WITH ALL H-1 AGONISTS, Biochemical and biophysical research communications, 214(1), 1995, pp. 110-117
LIPOPHILICITY AND HYDROGEN-BONDING CAPACITY OF H-1-ANTIHISTAMINIC AGENTS IN RELATION TO THEIR CENTRAL SEDATIVE SIDE-EFFECTS
Authors: TERLAAK AM TSAI RS DENKELDER GMDO CARRUPT PA TESTA B TIMMERMAN H
Citation: Am. Terlaak et al., LIPOPHILICITY AND HYDROGEN-BONDING CAPACITY OF H-1-ANTIHISTAMINIC AGENTS IN RELATION TO THEIR CENTRAL SEDATIVE SIDE-EFFECTS, European journal of pharmaceutical sciences, 2(5-6), 1994, pp. 373-384
SITE-DIRECTED MUTAGENESIS OF THE HISTAMINE H-1-RECEPTOR REVEALS A SELECTIVE INTERACTION OF ASPARAGINE(207) WITH SUBCLASSES OF H-1-RECEPTOR AGONISTS
Authors: LEURS R SMIT MJ TENSEN CP TERLAAK AM TIMMERMAN H
Citation: R. Leurs et al., SITE-DIRECTED MUTAGENESIS OF THE HISTAMINE H-1-RECEPTOR REVEALS A SELECTIVE INTERACTION OF ASPARAGINE(207) WITH SUBCLASSES OF H-1-RECEPTOR AGONISTS, Biochemical and biophysical research communications, 201(1), 1994, pp. 295-301
STRUCTURE-ACTIVITY-RELATIONSHIPS WITHIN A SERIES OF ANALOGS OF THE HISTAMINE H-1-ANTAGONIST TERFENADINE
Authors: ZHANG MQ TERLAAK AM TIMMERMAN H
Citation: Mq. Zhang et al., STRUCTURE-ACTIVITY-RELATIONSHIPS WITHIN A SERIES OF ANALOGS OF THE HISTAMINE H-1-ANTAGONIST TERFENADINE, European journal of medicinal chemistry, 28(2), 1993, pp. 165-173
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