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Results: 1-20 |
Results: 20
DESIGN AND SYNTHESIS OF POTENT, SELECTIVE INHIBITORS OF ENDOTHELIN-CONVERTING ENZYME
Authors: JENG AY SAVAGE P CHOU M TRAPANI AJ MOLITERNI JA MOSKAL MA NEUBERT AD MARCOPULOS N STAMFORD LB WALLACE EM
Citation: Ay. Jeng et al., DESIGN AND SYNTHESIS OF POTENT, SELECTIVE INHIBITORS OF ENDOTHELIN-CONVERTING ENZYME, Naunyn-Schmiedeberg's archives of pharmacology, 358(1), 1998, pp. 3723-3723
ANTIHYPERTENSIVE AND NATRIURETIC EFFECTS OF CGS-30440, A DUAL INHIBITOR OF ANGIOTENSIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE-24.11
Authors: CHATELAIN RE GHAI RD TRAPANI AJ ODORICO LM DARDIK BN DELOMBAERT S LAPPE RW FINK CA
Citation: Re. Chatelain et al., ANTIHYPERTENSIVE AND NATRIURETIC EFFECTS OF CGS-30440, A DUAL INHIBITOR OF ANGIOTENSIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE-24.11, The Journal of pharmacology and experimental therapeutics, 284(3), 1998, pp. 974-982
DESIGN AND SYNTHESIS OF POTENT, SELECTIVE INHIBITORS OF ENDOTHELIN-CONVERTING ENZYME
Authors: WALLACE EM MOLITERNI JA MOSKAL MA NEUBERT AD MARCOPULOS N STAMFORD LB TRAPANI AJ SAVAGE P CHOU M JENG AY
Citation: Em. Wallace et al., DESIGN AND SYNTHESIS OF POTENT, SELECTIVE INHIBITORS OF ENDOTHELIN-CONVERTING ENZYME, Journal of medicinal chemistry, 41(9), 1998, pp. 1513-1523
DUAL INHIBITION OF ANGIOTENSIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE BY TRICYCLIC BENZAZEPINONE THIOLS
Authors: DELOMBAERT S BLANCHARD L STAMFORD LB SAKANE Y BERRY C GHAI RD TRAPANI AJ
Citation: S. Delombaert et al., DUAL INHIBITION OF ANGIOTENSIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE BY TRICYCLIC BENZAZEPINONE THIOLS, Bioorganic & medicinal chemistry letters, 6(23), 1996, pp. 2875-2880
ANTIHYPERTENSIVE AND NATRIURETIC EFFECTS OF CGS 30440, A DUAL INHIBITOR OF ANGIOTENSIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE-24.11
Authors: CHATELAIN RE ODORICO LM GHAI RD TRAPANI AJ FINK CA LAPPE RW
Citation: Re. Chatelain et al., ANTIHYPERTENSIVE AND NATRIURETIC EFFECTS OF CGS 30440, A DUAL INHIBITOR OF ANGIOTENSIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE-24.11, The FASEB journal, 10(3), 1996, pp. 4038-4038
MERCAPTOACYL DIPEPTIDES AS ORALLY-ACTIVE DUAL INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE
Authors: FINK CA CARLSON JE MCTAGGART PA QIAO Y WEBB R CHATELAIN R JENG AY TRAPANI AJ
Citation: Ca. Fink et al., MERCAPTOACYL DIPEPTIDES AS ORALLY-ACTIVE DUAL INHIBITORS OF ANGIOTENSIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE, Journal of medicinal chemistry, 39(16), 1996, pp. 3158-3168
A RAPID INDIRECT METHOD TO DETERMINE THE PLASMA-CONCENTRATIONS OF NEUTRAL ENDOPEPTIDASE INHIBITORS
Authors: GHAI RD DELOMBAERT S KSANDER GM BERRY C SAKANE Y TRAPANI AJ
Citation: Rd. Ghai et al., A RAPID INDIRECT METHOD TO DETERMINE THE PLASMA-CONCENTRATIONS OF NEUTRAL ENDOPEPTIDASE INHIBITORS, Research communications in molecular pathology and pharmacology, 87(2), 1995, pp. 211-220
NONPEPTIDIC INHIBITORS OP NEUTRAL ENDOPEPTIDASE-24.11 .2. DESIGN AND PHARMACOLOGY OF ORALLY-ACTIVE PHOSPHONATE PRODRUGS
Authors: DELOMBAERT S BLANCHARD L BERRY C GHAI RD TRAPANI AJ
Citation: S. Delombaert et al., NONPEPTIDIC INHIBITORS OP NEUTRAL ENDOPEPTIDASE-24.11 .2. DESIGN AND PHARMACOLOGY OF ORALLY-ACTIVE PHOSPHONATE PRODRUGS, Bioorganic & medicinal chemistry letters, 5(2), 1995, pp. 151-154
CGS-23425 - A SELECTIVE CHOLESTEROL-LOWERING, CARDIAC-SPARING THYROMIMETIC IN CYNOMOLGUS MONKEYS
Authors: BEIL ME HINTZE TH OCHOA M DOTSON RA YURACEK EC STEPHAN ZF TRAPANI AJ
Citation: Me. Beil et al., CGS-23425 - A SELECTIVE CHOLESTEROL-LOWERING, CARDIAC-SPARING THYROMIMETIC IN CYNOMOLGUS MONKEYS, The FASEB journal, 9(3), 1995, pp. 194-194
INHIBITION OF BIG ET-1-INDUCED PRESSOR-RESPONSE BY AN ORALLY-ACTIVE DUAL INHIBITOR OF ENDOTHELIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE-24.11
Authors: TRAPANI AJ DELOMBAERT S KUZMICH S JENG AY
Citation: Aj. Trapani et al., INHIBITION OF BIG ET-1-INDUCED PRESSOR-RESPONSE BY AN ORALLY-ACTIVE DUAL INHIBITOR OF ENDOTHELIN-CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE-24.11, Journal of cardiovascular pharmacology, 26, 1995, pp. 69-71
NEW ALPHA-THIOL DIPEPTIDE DUAL INHIBITORS OF ANGIOTENSIN-I CONVERTING-ENZYME AND NEUTRAL ENDOPEPTIDASE EC-3.4.24.11
Authors: FINK CA QIAO Y BERRY CJ SAKANE Y GHAI RD TRAPANI AJ
Citation: Ca. Fink et al., NEW ALPHA-THIOL DIPEPTIDE DUAL INHIBITORS OF ANGIOTENSIN-I CONVERTING-ENZYME AND NEUTRAL ENDOPEPTIDASE EC-3.4.24.11, Journal of medicinal chemistry, 38(26), 1995, pp. 5023-5030
A RAPID INDIRECT METHOD TO DETERMINE THE PHARMACOKINETICS OF NEUTRAL ENDOPEPTIDASE (NEP-3.4.24.11) INHIBITORS
Authors: GHAI RD DELOMBAERT S KSANDER GM BERRY C SAKANE Y TRAPANI AJ
Citation: Rd. Ghai et al., A RAPID INDIRECT METHOD TO DETERMINE THE PHARMACOKINETICS OF NEUTRAL ENDOPEPTIDASE (NEP-3.4.24.11) INHIBITORS, The FASEB journal, 8(4), 1994, pp. 10000099-10000099
INHIBITION OF NEUTRAL ENDOPEPTIDASE-24.11 (NEP) AND ENDOTHELIN-CONVERTING ENZYME (ECE) BY AMINOPHOSPHONATE ANALOGS IN-VITRO AND IN-VIVO
Authors: TRAPANI AJ BEIL ME BERRY C DELOMBAERT S GERLOCK TE GHAI RD GRAYBILL SC JENG AY SAKANE Y SAVAGE P
Citation: Aj. Trapani et al., INHIBITION OF NEUTRAL ENDOPEPTIDASE-24.11 (NEP) AND ENDOTHELIN-CONVERTING ENZYME (ECE) BY AMINOPHOSPHONATE ANALOGS IN-VITRO AND IN-VIVO, The FASEB journal, 8(4), 1994, pp. 10000104-10000104
PHARMACOLOGICAL PROFILE OF CGS-24128, A POTENT, LONG-ACTING INHIBITOROF NEUTRAL ENDOPEPTIDASE-24.11
Authors: TRAPANI AJ BELL ME COTE DT DELOMBAERT S ERION MD GERLOCK TE GHAI RD HOPKINS MF PEPPARD JV WEBB RL LAPPE RW WORCEL M
Citation: Aj. Trapani et al., PHARMACOLOGICAL PROFILE OF CGS-24128, A POTENT, LONG-ACTING INHIBITOROF NEUTRAL ENDOPEPTIDASE-24.11, Journal of cardiovascular pharmacology, 23(3), 1994, pp. 358-364
N-PHOSPHONOMETHYL DIPEPTIDES AND THEIR PHOSPHONATE PRODRUGS, A NEW-GENERATION OF NEUTRAL ENDOPEPTIDASE (NEP,EC-3.4.24.11) INHIBITORS
Authors: DELOMBAERT S ERION MD TAN J BLANCHARD L ELCHEHABI L GHAI RD SAKANE Y BERRY C TRAPANI AJ
Citation: S. Delombaert et al., N-PHOSPHONOMETHYL DIPEPTIDES AND THEIR PHOSPHONATE PRODRUGS, A NEW-GENERATION OF NEUTRAL ENDOPEPTIDASE (NEP,EC-3.4.24.11) INHIBITORS, Journal of medicinal chemistry, 37(4), 1994, pp. 498-511
PHARMACOLOGICAL PROFILE OF A NONPEPTIDIC DUAL INHIBITOR OF NEUTRAL ENDOPEPTIDASE-24.11 AND ENDOTHELIN-CONVERTING ENZYME
Authors: DELOMBAERT S GHAI RD JENG AY TRAPANI AJ WEBB RL
Citation: S. Delombaert et al., PHARMACOLOGICAL PROFILE OF A NONPEPTIDIC DUAL INHIBITOR OF NEUTRAL ENDOPEPTIDASE-24.11 AND ENDOTHELIN-CONVERTING ENZYME, Biochemical and biophysical research communications, 204(1), 1994, pp. 407-412
EFFECTS OF METALLOPROTEASE INHIBITORS ON THE CONVERSION OF PROENDOTHELIN-1 TO ENDOTHELIN-1
Authors: TRAPANI AJ BALWIERCZAK JL LAPPE RW STANTON JL GRAYBILL SC HOPKINS MF SAVAGE P SPERBECK DM JENG AY
Citation: Aj. Trapani et al., EFFECTS OF METALLOPROTEASE INHIBITORS ON THE CONVERSION OF PROENDOTHELIN-1 TO ENDOTHELIN-1, Biochemistry and molecular biology international, 31(5), 1993, pp. 861-867
THE PHARMACOLOGY OF CCS-25462 - A POTENT, ORALLY BIOAVAILABLE, LONG-ACTING INHIBITOR OF NEUTRAL ENDOPEPTIDASE 24.11
Authors: TRAPANI AJ DELOMBAERT S ERION MD GHAI RD PEPPARD JV LAPPE RW WORCEL M
Citation: Aj. Trapani et al., THE PHARMACOLOGY OF CCS-25462 - A POTENT, ORALLY BIOAVAILABLE, LONG-ACTING INHIBITOR OF NEUTRAL ENDOPEPTIDASE 24.11, Journal of hypertension, 11, 1993, pp. 190000220-190000221
DESIGN AND SYNTHESIS OF AN ORALLY-ACTIVE MACROCYCLIC NEUTRAL ENDOPEPTIDASE-24.11 INHIBITOR
Authors: MACPHERSON LJ BAYBURT EK CAPPARELLI MP BOHACEK RS CLARKE FH GHAI RD SAKANE Y BERRY CJ PEPPARD JV TRAPANI AJ
Citation: Lj. Macpherson et al., DESIGN AND SYNTHESIS OF AN ORALLY-ACTIVE MACROCYCLIC NEUTRAL ENDOPEPTIDASE-24.11 INHIBITOR, Journal of medicinal chemistry, 36(24), 1993, pp. 3821-3828
HETEROCYCLIC LACTAM DERIVATIVES AS DUAL ANGIOTENSIN-CONVERTING ENZYMEAND NEUTRAL ENDOPEPTIDASE-24.11 INHIBITORS
Authors: STANTON JL SPERBECK DM TRAPANI AJ COTE D SAKANE Y BERRY CJ GHAI RD
Citation: Jl. Stanton et al., HETEROCYCLIC LACTAM DERIVATIVES AS DUAL ANGIOTENSIN-CONVERTING ENZYMEAND NEUTRAL ENDOPEPTIDASE-24.11 INHIBITORS, Journal of medicinal chemistry, 36(24), 1993, pp. 3829-3833
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