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Results: 1-25 | 26-50 | 51-55
Results: 1-25/55
Methods to determine the constitutive activity of histamine H-2 receptors
Authors: Leurs, R Hoffmann, M Alewijnse, AE Smit, MJ Timmerman, H
Citation: R. Leurs et al., Methods to determine the constitutive activity of histamine H-2 receptors, METH ENZYM, 343, 2002, pp. 405-416
Synthesis and use of FSCPX, an irreversible adenosine A(1) antagonist, as a 'receptor knock-down' tool
Authors: van Muijlwijk-Koezen, JE Timmerman, H van der Sluis, RP van de Stolpe, AC Menge, WMPB Beukers, MW van der Graaf, PH de Groote, M IJzerman, AP
Citation: Je. Van Muijlwijk-koezen et al., Synthesis and use of FSCPX, an irreversible adenosine A(1) antagonist, as a 'receptor knock-down' tool, BIOORG MED, 11(6), 2001, pp. 815-818
Pharmacological analysis of immepip and imetit homologues. Further evidence for histamine H-3 receptor heterogeneity?
Authors: Alves-Rodrigues, A Lemstra, S Vollinga, RC Menge, WMPB Timmerman, H Leurs, R
Citation: A. Alves-rodrigues et al., Pharmacological analysis of immepip and imetit homologues. Further evidence for histamine H-3 receptor heterogeneity?, BEH BRA RES, 124(2), 2001, pp. 121-127
Histamine H-1-receptor activation of nuclear factor-kappa B: Roles for G beta gamma- and G alpha(q/11)-subunits in constitutive and agonist-mediated signaling
Authors: Bakker, RA Schoonus, SBJ Smit, MJ Timmerman, H Leurs, R
Citation: Ra. Bakker et al., Histamine H-1-receptor activation of nuclear factor-kappa B: Roles for G beta gamma- and G alpha(q/11)-subunits in constitutive and agonist-mediated signaling, MOLEC PHARM, 60(5), 2001, pp. 1133-1142
Identification of rat H-3 receptor isoforms with different brain expression and signaling properties
Authors: Drutel, G Peitsaro, N Karlstedt, K Wieland, K Smit, MJ Timmerman, H Panula, P Leurs, R
Citation: G. Drutel et al., Identification of rat H-3 receptor isoforms with different brain expression and signaling properties, MOLEC PHARM, 59(1), 2001, pp. 1-8
Significance of GABAergic systems in the action of improgan, a non-opioid analgesic
Authors: Hough, LB Nalwalk, JW Leurs, R Menge, WMPB Timmerman, H
Citation: Lb. Hough et al., Significance of GABAergic systems in the action of improgan, a non-opioid analgesic, LIFE SCI, 68(24), 2001, pp. 2751-2757
Constitutive activity of histamine H-3 receptors stably expressed in SK-N-MC cells: Display of agonism and inverse agonism by H-3 antagonists
Authors: Wieland, K Bongers, G Yamamoto, Y Hashimoto, T Yamatodani, A Menge, WMBP Timmerman, H Lovenberg, TW Leurs, R
Citation: K. Wieland et al., Constitutive activity of histamine H-3 receptors stably expressed in SK-N-MC cells: Display of agonism and inverse agonism by H-3 antagonists, J PHARM EXP, 299(3), 2001, pp. 908-914
Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists
Authors: van Muijlwijk-Koezen, JE Timmerman, H Vollinga, RC Kunzel, JFV de Groote, M Visser, S Ijzerman, AP
Citation: Je. Van Muijlwijk-koezen et al., Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists, J MED CHEM, 44(5), 2001, pp. 749-762
Novel selective PDE4 inhibitors. 1. Synthesis, structure-activity relationships, and molecular modeling of 4-(3,4-dimethoxyphenyl)-2H-phthalazin-1-ones and analogues
Authors: Van der Mey, M Hatzelmann, A Van der Laan, IJ Sterk, GJ Thibaut, U Timmerman, H
Citation: M. Van Der Mey et al., Novel selective PDE4 inhibitors. 1. Synthesis, structure-activity relationships, and molecular modeling of 4-(3,4-dimethoxyphenyl)-2H-phthalazin-1-ones and analogues, J MED CHEM, 44(16), 2001, pp. 2511-2522
Novel selective PDE4 inhibitors. 2. Synthesis and structure-activity relationships of 4-aryl-substituted cis-tetra- and cis-hexahydrophthalazinones
Authors: Van der Mey, M Hatzelmann, A Van Klink, GPM Van der Laan, IJ Sterk, GJ Thibaut, U Ulrich, WR Timmerman, H
Citation: M. Van Der Mey et al., Novel selective PDE4 inhibitors. 2. Synthesis and structure-activity relationships of 4-aryl-substituted cis-tetra- and cis-hexahydrophthalazinones, J MED CHEM, 44(16), 2001, pp. 2523-2535
Development of a pharmacophore model for histamine H-3 receptor antagonists, using the newly developed molecular modeling program SLATE
Authors: De Esch, IJP Mills, JEJ Perkins, TDJ Romeo, G Hoffmann, M Wieland, K Leurs, R Menge, WMPB Nederkoorn, PHJ Dean, PM Timmerman, H
Citation: Ijp. De Esch et al., Development of a pharmacophore model for histamine H-3 receptor antagonists, using the newly developed molecular modeling program SLATE, J MED CHEM, 44(11), 2001, pp. 1666-1674
Constitutive signaling of the human cytomegalovirus-encoded chemokine receptor US28
Authors: Casarosa, P Bakker, RA Verzijl, D Navis, M Timmerman, H Leurs, R Smit, MJ
Citation: P. Casarosa et al., Constitutive signaling of the human cytomegalovirus-encoded chemokine receptor US28, J BIOL CHEM, 276(2), 2001, pp. 1133-1137
VUF-K-8788, a periphery-selective histamine H-1 antagonist with anti-pruritic activities
Authors: Takizawa, T Matsumoto, J Tohma, T Kanke, T Wada, Y Nagao, M Inagaki, N Nagai, H Zhang, MQ Timmerman, H
Citation: T. Takizawa et al., VUF-K-8788, a periphery-selective histamine H-1 antagonist with anti-pruritic activities, JPN J PHARM, 86(1), 2001, pp. 55-64
Recombinant Semliki Forest virus for over-expression and pharmacological characterisation of the histamine H-2 receptor in mammalian cells
Authors: Hoffmann, M Verzijl, D Lundstrom, K Simmen, U Alewijnse, AE Timmerman, H Leurs, R
Citation: M. Hoffmann et al., Recombinant Semliki Forest virus for over-expression and pharmacological characterisation of the histamine H-2 receptor in mammalian cells, EUR J PHARM, 427(2), 2001, pp. 105-114
New insights into the second generation antihistamines
Authors: Walsh, GM Annunziato, L Frossard, N Knol, K Levander, S Nicolas, JM Taglialatela, M Tharp, MD Tillement, JP Timmerman, H
Citation: Gm. Walsh et al., New insights into the second generation antihistamines, DRUGS, 61(2), 2001, pp. 207-236
Is histamine the final neurotransmitter in the entrainment of circadian rhythms in mammals?
Authors: Jacobs, EH Yamatodani, A Timmerman, H
Citation: Eh. Jacobs et al., Is histamine the final neurotransmitter in the entrainment of circadian rhythms in mammals?, TRENDS PHAR, 21(8), 2000, pp. 293-298
Cardiotoxic potential and CNS effects of first-generation antihistamines
Authors: Taglialatela, M Timmerman, H Annunziato, L
Citation: M. Taglialatela et al., Cardiotoxic potential and CNS effects of first-generation antihistamines, TRENDS PHAR, 21(2), 2000, pp. 52-56
H-3 receptor gene is cloned at last
Authors: Leurs, R Hoffmann, M Wieland, K Timmerman, H
Citation: R. Leurs et al., H-3 receptor gene is cloned at last, TRENDS PHAR, 21(1), 2000, pp. 11-12
Solid-phase synthesis of 4-substituted imidazoles using a scaffold approach
Authors: Gelens, E Koot, WJ Menge, WMPB Ottenheijm, HCJ Timmerman, H
Citation: E. Gelens et al., Solid-phase synthesis of 4-substituted imidazoles using a scaffold approach, BIOORG MED, 10(17), 2000, pp. 1935-1938
Special issue - Festschrift dedicated to Professor Dr. D. Breimer - Preface
Authors: Timmerman, H
Citation: H. Timmerman, Special issue - Festschrift dedicated to Professor Dr. D. Breimer - Preface, EUR J PH SC, 12(2), 2000, pp. 83-84
A qualitative model for the histamine H-3 receptor explaining agonistic and antagonistic activity simultaneously
Authors: de Esch, IJP Timmerman, H Menge, WMPB Nederkoorn, PHJ
Citation: Ijp. De Esch et al., A qualitative model for the histamine H-3 receptor explaining agonistic and antagonistic activity simultaneously, ARCH PHARM, 333(8), 2000, pp. 254-260
The Stichting Ambulante Preventie Projecten method: A comparative study ofrecidivism in first offenders in a Dutch outpatient setting
Authors: Ruddijs, F Timmerman, H
Citation: F. Ruddijs et H. Timmerman, The Stichting Ambulante Preventie Projecten method: A comparative study ofrecidivism in first offenders in a Dutch outpatient setting, INT J OFFEN, 44(6), 2000, pp. 725-739
Synthesis of benzylideneacetophenones and their inhibition of lipid peroxidation
Authors: Arty, IS Timmerman, H Samhoedi, M",Sastrohamidjojo,Sugiyanto,"van der Goot, H
Citation: Is. Arty et al., Synthesis of benzylideneacetophenones and their inhibition of lipid peroxidation, EUR J MED C, 35(4), 2000, pp. 449-457
Selective ligands as tools to study histamine receptors
Authors: van der Goot, H Timmerman, H
Citation: H. Van Der Goot et H. Timmerman, Selective ligands as tools to study histamine receptors, EUR J MED C, 35(1), 2000, pp. 5-20
Factors involved in the absence of sedative effects by the second-generation antihistamines
Authors: Timmerman, H
Citation: H. Timmerman, Factors involved in the absence of sedative effects by the second-generation antihistamines, ALLERGY, 55, 2000, pp. 5-10
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