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Results: 1-7 |
Results: 7
ORALLY-ACTIVE TRIFLUOROMETHYL KETONE INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE
Authors: VEALE CA BERNSTEIN PR BOHNERT CM BROWN FJ BRYANT C DAMEWOOD JR EARLEY R FEENEY SW EDWARDS PD GOMES B HULSIZER JM KOSMIDER BJ KRELL RD MOORE G SALCEDO TW SHAW A SILBERSTEIN DS STEELMAN GB STEIN M STRIMPLER A THOMAS RM VACEK EP WILLIAMS JC WOLANIN DJ WOOLSON S
Citation: Ca. Veale et al., ORALLY-ACTIVE TRIFLUOROMETHYL KETONE INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE, Journal of medicinal chemistry, 40(20), 1997, pp. 3173-3181
NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .5. DESIGN, SYNTHESIS, AND X-RAY CRYSTALLOGRAPHY OF A SERIES OF ORALLY-ACTIVE 5-AMINOPYRIMIDIN-6-ONE-CONTAINING TRIFLUOROMETHYL KETONES
Authors: VEALE CA BERNSTEIN PR BRYANT C CECCARELLI C DAMEWOOD JR EARLEY R FEENEY SW GOMES B KOSMIDER BJ STEELMAN GB THOMAS RM VACEK EP WILLIAMS JC WOLANIN DJ WOOLSON S
Citation: Ca. Veale et al., NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .5. DESIGN, SYNTHESIS, AND X-RAY CRYSTALLOGRAPHY OF A SERIES OF ORALLY-ACTIVE 5-AMINOPYRIMIDIN-6-ONE-CONTAINING TRIFLUOROMETHYL KETONES, Journal of medicinal chemistry, 38(1), 1995, pp. 98-108
NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .6. DESIGN OF A POTENT, INTRATRACHEALLY ACTIVE, PYRIDONE-BASED TRIFLUOROMETHYL KETONE
Authors: BERNSTEIN PR GOMES BC KOSMIDER BJ VACEK EP WILLIAMS JC
Citation: Pr. Bernstein et al., NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .6. DESIGN OF A POTENT, INTRATRACHEALLY ACTIVE, PYRIDONE-BASED TRIFLUOROMETHYL KETONE, Journal of medicinal chemistry, 38(1), 1995, pp. 212-215
EXAMINATION OF PEPTIDIC ALPHA',BETA-DIAMINO-ALPHA,ALPHA-DIFLUOROKETONES AS INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE
Authors: BERNSTEIN PR KOSMIDER BJ VACEK EP VEALE CA GOMES BC
Citation: Pr. Bernstein et al., EXAMINATION OF PEPTIDIC ALPHA',BETA-DIAMINO-ALPHA,ALPHA-DIFLUOROKETONES AS INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE, Bioorganic & medicinal chemistry letters, 4(18), 1994, pp. 2175-2178
DESIGN OF ORALLY-ACTIVE, NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE
Authors: BROWN FJ ANDISIK DW BERNSTEIN PR BRYANT CB CECCARELLI C DAMEWOOD JR WOOLSON SA EDWARDS PD EARLEY RA FEENEY S GREEN RC GOMES B KOSMIDER BJ KRELL RD SHAW A STEELMAN GB THOMAS RN VACEK EP VEALE CA TUTHILL PA WARNER P WILLIAMS JC WOLANIN DJ
Citation: Fj. Brown et al., DESIGN OF ORALLY-ACTIVE, NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE, Journal of medicinal chemistry, 37(9), 1994, pp. 1259-1261
SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, AND PHARMACOLOGICAL EVALUATION OF A SERIES OF FLUORINATED 3-BENZYL-5-INDOLECARBOXAMIDES - IDENTIFICATION OF ]-3-METHOXY-N-[(2-METHYLPHENYL)SULFONYL]BENZAMIDE, A POTENT, ORALLY-ACTIVE ANTAGONIST OF LEUKOTRIENES D(4) AND E(4)
Authors: JACOBS RT BERNSTEIN PR CRONK LA VACEK EP NEWCOMB LF AHARONY D BUCKNER CK KUSNER EJ
Citation: Rt. Jacobs et al., SYNTHESIS, STRUCTURE-ACTIVITY-RELATIONSHIPS, AND PHARMACOLOGICAL EVALUATION OF A SERIES OF FLUORINATED 3-BENZYL-5-INDOLECARBOXAMIDES - IDENTIFICATION OF ]-3-METHOXY-N-[(2-METHYLPHENYL)SULFONYL]BENZAMIDE, A POTENT, ORALLY-ACTIVE ANTAGONIST OF LEUKOTRIENES D(4) AND E(4), Journal of medicinal chemistry, 37(9), 1994, pp. 1282-1297
NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .3. DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF ORALLY-ACTIVE 3-AMINO-6-PHENYLPYRIDIN-2-ONE TRIFLUOROMETHYL KETONES
Authors: BERNSTEIN PR ANDISIK D BRADLEY PK BRYANT CB CECCARELLI C DAMEWOOD JR EARLEY R EDWARDS PD FEENEY S GOMES BC KOSMIDER BJ STEELMAN GB THOMAS RM VACEK EP VEALE CA WILLIAMS JC WOLANIN DJ WOOLSON SA
Citation: Pr. Bernstein et al., NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .3. DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF ORALLY-ACTIVE 3-AMINO-6-PHENYLPYRIDIN-2-ONE TRIFLUOROMETHYL KETONES, Journal of medicinal chemistry, 37(20), 1994, pp. 3313-3326
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