Citation: G. Marzoni et Md. Varney, AN IMPROVED LARGE-SCALE SYNTHESIS OF BENZ[CD]INDOL-2(1H)-ONE AND 5-METHYLBENZ[CD]INDOL-2(1H)-ONE, Organic process research & development, 1(1), 1997, pp. 81-84
Authors:
JONES TR
WEBBER SE
VARNEY MD
REDDY MR
LEWIS KK
KATHARDEKAR V
MAZDIYASNI H
DEAL J
NGUYEN D
WELSH KM
WEBBER S
JOHNSTON A
MATTHEWS DA
SMITH WW
JANSON CA
BACQUET RJ
HOWLAND EF
BOOTH CLJ
HERRMANN SM
WARD RW
WHITE J
BARTLETT CA
MORSE CA
Citation: Tr. Jones et al., STRUCTURE-BASED DESIGN OF SUBSTITUTED DIPHENYL SULFONES AND SULFOXIDES AS LIPOPHILIC INHIBITORS OF THYMIDYLATE SYNTHASE, Journal of medicinal chemistry, 40(5), 1997, pp. 677-683
Authors:
VARNEY MD
PALMER CL
ROMINES WH
BORITZKI T
MARGOSIAK SA
ALMASSY R
JANSON CA
BARTLETT C
HOWLAND EJ
FERRE R
Citation: Md. Varney et al., PROTEIN STRUCTURE-BASED DESIGN, SYNTHESIS, AND BIOLOGICAL EVALUATION OF 5-THIA-2,6-DIAMINO-4(3H)-OXOPYRIMIDINES - POTENT INHIBITORS OF GLYCINAMIDE RIBONUCLEOTIDE TRANSFORMYLASE WITH POTENT CELL-GROWTH INHIBITION, Journal of medicinal chemistry, 40(16), 1997, pp. 2502-2524
Authors:
JONES TR
VARNEY MD
WEBBER SE
LEWIS KK
MARZONI GP
PALMER CL
KATHARDEKAR V
WELSH KM
WEBBER S
MATTHEWS DA
APPELT K
SMITH WW
JANSON CA
VILLAFRANCA JE
BACQUET RJ
HOWLAND EF
BOOTH CLJ
HERRMANN SM
WARD RW
WHITE J
MOOMAW EW
BARTLETT CA
MORSE CA
Citation: Tr. Jones et al., STRUCTURE-BASED DESIGN OF LIPOPHILIC QUINAZOLINE INHIBITORS OF THYMIDYLATE SYNTHASE, Journal of medicinal chemistry, 39(4), 1996, pp. 904-917
Citation: Vn. Viswanadhan et al., AN APPROACH TO RAPID ESTIMATION OF RELATIVE BINDING AFFINITIES OF ENZYME-INHIBITORS - APPLICATION TO PEPTIDOMIMETIC INHIBITORS OF THE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 PROTEASE, Journal of medicinal chemistry, 39(3), 1996, pp. 705-712
Authors:
TAIT BD
DRUMMOND BP
VARNEY MD
HARRISON LC
Citation: Bd. Tait et al., HLA-DRB1-ASTERISK-0401 IS ASSOCIATED WITH SUSCEPTIBILITY TO INSULIN-DEPENDENT DIABETES-MELLITUS INDEPENDENTLY OF THE DQB1 LOCUS, European journal of immunogenetics, 22(4), 1995, pp. 289-297
Citation: Md. Varney et al., MOLECULAR TYPING AND HAPLOTYPIC ASSOCIATIONS OF HLA-B-ASTERISK-44 SUBTYPES, European journal of immunogenetics, 22(2), 1995, pp. 215-220
Authors:
VARNEY MD
PALMER CL
DEAL JG
WEBBER S
WELSH KM
BARTLETT CA
MORSE CA
SMITH WW
JANSON CA
Citation: Md. Varney et al., SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL 2,6-DIAMINOBENZ[CD]INDOLE INHIBITORS OF THYMIDYLATE SYNTHASE USING THE PROTEIN-STRUCTURE AS A GUIDE, Journal of medicinal chemistry, 38(11), 1995, pp. 1892-1903
Authors:
VARNEY MD
ROMINES WH
BORITZKI T
MARGOSIAK SA
BARTLETT C
HOWLAND EJ
Citation: Md. Varney et al., SYNTHESIS AND BIOLOGICAL EVALUATION OF IN-5-YL]METHYL)THIO]CYCLOBUTYL)BENZOYL]-L-GLUTAMIC ACID A NOVEL 5-THIAPYRIMIDINONE INHIBITOR OF DIHYDROFOLATE-REDUCTASE, Journal of heterocyclic chemistry, 32(5), 1995, pp. 1493-1498
Citation: J. Greer et al., APPLICATION OF THE 3-DIMENSIONAL STRUCTURES OF PROTEIN TARGET MOLECULES IN STRUCTURE-BASED DRUG DESIGN, Journal of medicinal chemistry, 37(8), 1994, pp. 1035-1054
Authors:
REDDY MR
VARNEY MD
KALISH V
VISWANADHAN VN
APPELT K
Citation: Mr. Reddy et al., CALCULATION OF RELATIVE DIFFERENCES IN THE BINDING FREE-ENERGIES OF HIV-1 PROTEASE INHIBITORS - A THERMODYNAMIC CYCLE PERTURBATION APPROACH, Journal of medicinal chemistry, 37(8), 1994, pp. 1145-1152
Authors:
VARNEY MD
APPELT K
KALISH V
REDDY MR
TATLOCK J
PALMER CL
ROMINES WH
WU BW
MUSICK L
Citation: Md. Varney et al., CRYSTAL-STRUCTURE-BASED DESIGN AND SYNTHESIS OF NOVEL C-TERMINAL INHIBITORS OF HIV PROTEASE, Journal of medicinal chemistry, 37(15), 1994, pp. 2274-2284