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Results: 1-25 | 26-38
Results: 1-25/38
Effects of two-carbon bridge region methoxylation of benztropine: Discovery of novel chiral ligands for the dopamine transporter
Authors: Simoni, D Roberti, M Rondanin, R Baruchello, R Rossi, M Invidiata, FP Merighi, S Varani, K Gessi, S Borea, PA Marino, S Cavallini, S Bianchi, C Siniscalchi, A
Citation: D. Simoni et al., Effects of two-carbon bridge region methoxylation of benztropine: Discovery of novel chiral ligands for the dopamine transporter, BIOORG MED, 11(6), 2001, pp. 823-827
Aberrant amplification of A(2A) receptor signaling in striatal cells expressing mutant huntingtin
Authors: Varani, K Rigamonti, D Sipione, S Camurri, A Borea, PA Cattabeni, F Abbracchio, MP Cattaneo, E
Citation: K. Varani et al., Aberrant amplification of A(2A) receptor signaling in striatal cells expressing mutant huntingtin, FASEB J, 15(7), 2001, pp. 1245-1247
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor ligands: A starting point for searching A(2B) adenosine receptor antagonists
Authors: Baraldi, PG Cacciari, B Romagnoli, R Klotz, KN Spalluto, G Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor ligands: A starting point for searching A(2B) adenosine receptor antagonists, DRUG DEV R, 53(2-3), 2001, pp. 225-235
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new pharmacological tool for the characterization of the human A(3) adenosine receptor
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Varani, K Cessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives: A new pharmacological tool for the characterization of the human A(3) adenosine receptor, DRUG DEV R, 52(1-2), 2001, pp. 406-415
Comparison of Prazosin,Terazosin and tamsulosin: Functional and binding studies in isolated prostatic and vascular human tissues
Authors: Amadesi, S Varani, K Spisani, L Daniele, C Turini, A Agnello, G Zamboni, P Borea, PA Geppetti, P
Citation: S. Amadesi et al., Comparison of Prazosin,Terazosin and tamsulosin: Functional and binding studies in isolated prostatic and vascular human tissues, PROSTATE, 47(4), 2001, pp. 231-238
Structure-affinity relationships of a unique nicotinic ligand: N-1-dimethyl-N-4-phenylpiperazinium iodide (DMPP)
Authors: Romanelli, MN Manetti, D Scapecchi, S Borea, PA Dei, S Bartolini, A Ghelardini, C Gualtieri, F Guandalini, L Varani, K
Citation: Mn. Romanelli et al., Structure-affinity relationships of a unique nicotinic ligand: N-1-dimethyl-N-4-phenylpiperazinium iodide (DMPP), J MED CHEM, 44(23), 2001, pp. 3946-3955
Structure-activity studies of the Phe(4) residue of nociceptin(1-13)-NH2: Identification of highly potent agonists of the nociceptin/orphanin FQ receptor
Authors: Guerrini, R Calo, G Bigoni, R Rizzi, D Rizzi, A Zucchini, M Varani, K Hashiba, E Lambert, DG Toth, G Borea, PA Salvadori, S Regoli, D
Citation: R. Guerrini et al., Structure-activity studies of the Phe(4) residue of nociceptin(1-13)-NH2: Identification of highly potent agonists of the nociceptin/orphanin FQ receptor, J MED CHEM, 44(23), 2001, pp. 3956-3964
Met-Ile-Phe-Leu derivatives: full and partial agonists of human neutrophilformylpeptide receptors
Authors: Dalpiaz, A Scatturin, A Vertuani, G Pecoraro, R Borea, PA Varani, K Traniello, S Spisani, S
Citation: A. Dalpiaz et al., Met-Ile-Phe-Leu derivatives: full and partial agonists of human neutrophilformylpeptide receptors, EUR J PHARM, 411(3), 2001, pp. 327-333
Pharmacological and biochemical characterization of adenosine receptors inthe human malignant melanoma A375 cell line
Authors: Merighi, S Varani, K Gessi, S Cattabriga, E Iannotta, V Ulouglu, C Leung, E Borea, PA
Citation: S. Merighi et al., Pharmacological and biochemical characterization of adenosine receptors inthe human malignant melanoma A375 cell line, BR J PHARM, 134(6), 2001, pp. 1215-1226
Pharmacological and biochemical characterization of A(3) adenosine receptors in Jurkat T cells
Authors: Gessi, S Varani, K Merighi, S Morelli, A Ferrari, D Leung, E Baraldi, PG Spalluto, G Borea, PA
Citation: S. Gessi et al., Pharmacological and biochemical characterization of A(3) adenosine receptors in Jurkat T cells, BR J PHARM, 134(1), 2001, pp. 116-126
C-nucleoside analogues of furanfurin as ligands to A(1) adenosine receptors
Authors: Franchetti, P Cappellacci, L Marchetti, S Martini, C Costa, B Varani, K Borea, PA Grifantini, M
Citation: P. Franchetti et al., C-nucleoside analogues of furanfurin as ligands to A(1) adenosine receptors, BIO MED CH, 8(9), 2000, pp. 2367-2373
Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors
Authors: Baraldi, PG Cacciari, B Romagnoli, R Varani, K Merighi, S Gessi, S Borea, PA Leung, E Hickey, SL Spalluto, G
Citation: Pg. Baraldi et al., Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors, BIOORG MED, 10(3), 2000, pp. 209-211
Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors (vol 10, pg 209, 2000)
Authors: Baraldi, PG Cacciari, B Romagnoli, R Varani, K Merighi, S Gessi, S Borea, PA Leung, E Hickey, SL Spalluto, G
Citation: Pg. Baraldi et al., Synthesis and preliminary biological evaluation of [H-3]-MRE 3008-F20: thefirst high affinity radioligand antagonist for the human A(3) adenosine receptors (vol 10, pg 209, 2000), BIOORG MED, 10(12), 2000, pp. 1403-1403
Endocrine-disrupting agents on healthy human tissues
Authors: Paganetto, G Campi, F Varani, K Piffanelli, A Giovannini, G Borea, PA
Citation: G. Paganetto et al., Endocrine-disrupting agents on healthy human tissues, PHARM TOX, 86(1), 2000, pp. 24-29
Platelet alpha(2)-adrenoceptor alterations in patients with essential hypertension are normalized after treatment with doxazosin but not propranolol
Authors: Portaluppi, F Manfredini, R Varani, K Gessi, S Caiazza, A Borea, PA
Citation: F. Portaluppi et al., Platelet alpha(2)-adrenoceptor alterations in patients with essential hypertension are normalized after treatment with doxazosin but not propranolol, J HYPERTENS, 18(2), 2000, pp. 217-221
Ala scan analogues of HOE 140. Synthesis and biological activities
Authors: Quartara, L Ricci, R Meini, S Patacchini, R Giolitti, A Amadesi, S Rizzi, C Rizzi, A Varani, K Borea, PA Maggi, CA Regoli, D
Citation: L. Quartara et al., Ala scan analogues of HOE 140. Synthesis and biological activities, EUR J MED C, 35(11), 2000, pp. 1001-1010
A(3) adenosine receptor ligands: History and perspectives
Authors: Baraldi, PG Cacciari, B Romagnoli, R Merighi, S Varani, K Borea, PA Spalluto, G
Citation: Pg. Baraldi et al., A(3) adenosine receptor ligands: History and perspectives, MED RES REV, 20(2), 2000, pp. 103-128
[H-3]MRE 3008F20: A novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors
Authors: Varani, K Merighi, S Gessi, S Klotz, KN Leung, E Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Borea, PA
Citation: K. Varani et al., [H-3]MRE 3008F20: A novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors, MOLEC PHARM, 57(5), 2000, pp. 968-975
Binding thermodynamics and intrinsic activity of adenosine A(1) receptor ligands
Authors: Dalpiaz, A Scatturin, A Varani, K Pecoraro, R Pavan, B Borea, PA
Citation: A. Dalpiaz et al., Binding thermodynamics and intrinsic activity of adenosine A(1) receptor ligands, LIFE SCI, 67(12), 2000, pp. PL1517-PL1524
Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists: Influence of thechain at the N-8 pyrazole nitrogen
Authors: Baraldi, PG Cacciari, B Romagnoli, R Spalluto, G Moro, S Klotz, KN Leung, E Varani, K Gessi, S Merighi, S Borea, PA
Citation: Pg. Baraldi et al., Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as highly potent and selective human A(3) adenosine receptor antagonists: Influence of thechain at the N-8 pyrazole nitrogen, J MED CHEM, 43(25), 2000, pp. 4768-4780
Design, radiosynthesis, and biodistribution of a new potent and selective ligand for in vivo imaging of the adenosine A(2A) receptor system using positron emission tomography
Authors: Todde, S Moresco, RM Simonelli, F Baraldi, PG Cacciari, B Spalluto, G Varani, K Monopoli, A Matarrese, M Carpinelli, A Magni, F Kienle, MG Fazio, F
Citation: S. Todde et al., Design, radiosynthesis, and biodistribution of a new potent and selective ligand for in vivo imaging of the adenosine A(2A) receptor system using positron emission tomography, J MED CHEM, 43(23), 2000, pp. 4359-4362
Further studies on nociceptin-related peptides: Discovery of a new chemical template with antagonist activity on the nociceptin receptor
Authors: Guerrini, R Calo, G Bigoni, R Rizzi, A Varani, K Toth, G Gessi, S Hashiba, E Hashimoto, Y Lambert, DG Borea, PA Tomatis, R Salvadori, S Regoli, D
Citation: R. Guerrini et al., Further studies on nociceptin-related peptides: Discovery of a new chemical template with antagonist activity on the nociceptin receptor, J MED CHEM, 43(15), 2000, pp. 2805-2813
Dose and time effects of caffeine intake on human platelet adenosine A(2A)receptors - Functional and biochemical aspects
Authors: Varani, K Portaluppi, F Gessi, S Merighi, S Ongini, E Belardinelli, L Borea, PA
Citation: K. Varani et al., Dose and time effects of caffeine intake on human platelet adenosine A(2A)receptors - Functional and biochemical aspects, CIRCULATION, 102(3), 2000, pp. 285-289
A(2A) adenosine receptors in human peripheral blood cells
Authors: Gessi, S Varani, K Merighi, S Ongini, E Borea, PA
Citation: S. Gessi et al., A(2A) adenosine receptors in human peripheral blood cells, BR J PHARM, 129(1), 2000, pp. 2-11
Can thermodynamic measurements of receptor binding yield information on drug affinity and efficacy?
Authors: Borea, PA Dalpiaz, A Varani, K Gilli, P Gilli, G
Citation: Pa. Borea et al., Can thermodynamic measurements of receptor binding yield information on drug affinity and efficacy?, BIOCH PHARM, 60(11), 2000, pp. 1549-1556
Risultati: 1-25 | 26-38