Authors:
MASUDA Y
SUGO T
KIKUCHI T
SATOH M
FUJISAWA Y
ITOH Y
WAKIMASU M
OHTAKI T
Citation: Y. Masuda et al., ANTAGONIST ACTIVITY OF [THR(18),GAMMA-METHYLLEUCINE(19)]ENDOTHELIN-1 IN HUMAN ENDOTHELIN RECEPTORS, European journal of pharmacology, 325(2-3), 1997, pp. 263-270
Authors:
MASUDA Y
SUGO T
KIKUCHI T
KAWATA A
SATOH M
FUJISAWA Y
ITOH Y
WAKIMASU M
OHTAKI T
Citation: Y. Masuda et al., RECEPTOR-BINDING AND ANTAGONIST PROPERTIES OF A NOVEL ENDOTHELIN RECEPTOR ANTAGONIST, TAK-044 2-(2-THIENYL)GLYCYL-L-LEUCYL-D-TRYPTOPHYL]DISODIUM SALT), IN HUMAN ENDOTHELIN(A) AND ENDOTHELIN(B) RECEPTORS, The Journal of pharmacology and experimental therapeutics, 279(2), 1996, pp. 675-685
Authors:
WATANABE T
AWANE Y
IKEDA S
FUJIWARA S
KUBO K
KIKUCHI T
KUSUMOTO K
WAKIMASU M
FUJINO M
Citation: T. Watanabe et al., PHARMACOLOGY OF A NONSELECTIVE ET(A) AND ET(B) RECEPTOR ANTAGONIST, TAK-044 AND THE INHIBITION OF MYOCARDIAL INFARCT SIZE IN RATS, British Journal of Pharmacology, 114(5), 1995, pp. 949-954
Authors:
KARAKI H
SUDJARWO SA
SHIMAMOTO N
WAKIMASU M
FUJINO M
Citation: H. Karaki et al., EFFECTS OF A POTENT, NONSELECTIVE ENDOTHELIN RECEPTOR ANTAGONIST, [THR(18), GAMMA-MELEU(19)]-ENDOTHELIN-1, ON THE ISOLATED BLOOD-VESSELS, Biochemical and biophysical research communications, 212(2), 1995, pp. 421-427
Authors:
KUSUMOTO K
KUBO K
KANDORI H
KITAYOSHI T
SATO S
WAKIMASU M
WATANABE T
FUJINO M
Citation: K. Kusumoto et al., EFFECTS OF A NEW ENDOTHELIN ANTAGONIST, TAK-044, ON POSTISCHEMIC ACUTE-RENAL-FAILURE IN RATS, Life sciences, 55(4), 1994, pp. 301-310
Authors:
IKEDA S
AWANE Y
KUSUMOTO K
WAKIMASU M
WATANABE T
FUJINO M
Citation: S. Ikeda et al., A NEW ENDOTHELIN RECEPTOR ANTAGONIST, TAK-044, SHOWS LONG-LASTING INHIBITION OF BOTH ET(A)-MEDIATED AND ET(B)-MEDIATED BLOOD-PRESSURE RESPONSES IN RATS, The Journal of pharmacology and experimental therapeutics, 270(2), 1994, pp. 728-733
Authors:
KIKUCHI T
OHTAKI T
KAWATA A
IMADA T
ASAMI T
MASUDA Y
SUGO T
KUSUMOTO K
KUBO K
WATANABE T
WAKIMASU M
FUJINO M
Citation: T. Kikuchi et al., CYCLIC HEXAPEPTIDE ENDOTHELIN RECEPTOR ANTAGONISTS HIGHLY POTENT FOR BOTH RECEPTOR SUBTYPES ET(A) AND ET(B), Biochemical and biophysical research communications, 200(3), 1994, pp. 1708-1712
Authors:
HATTORI N
WAKIMASU M
TAKAHASHI M
HIROSAWA M
SHIOTA K
OGAWA T
Citation: N. Hattori et al., CHARACTERIZATION OF RAT PLACENTAL LACTOGEN-ALPHA (PL-ALPHA) WITH AN ANTIPEPTIDE ANTIBODY-DIRECTED AGAINST RAT PLS, Endocrine journal, 40(6), 1993, pp. 727-735
Authors:
SHIMAMOTO N
KUBO K
WATANABE T
SUZUKI N
ABE M
KIKUCHI T
WAKIMASU M
FUJINO M
Citation: N. Shimamoto et al., PHARMACOLOGICAL PROFILE OF ENDOTHELIN-A B ANTAGONIST, [THR(18), GAMMA-METHYLLEU(19)]ENDOTHELIN-1/, Journal of cardiovascular pharmacology, 22, 1993, pp. 190000107-190000110
Authors:
KIKUCHI T
KUBO K
OHTAKI T
SUZUKI N
ASAMI T
SHIMAMOTO N
WAKIMASU M
FUJINO M
Citation: T. Kikuchi et al., ENDOTHELIN-1 ANALOGS SUBSTITUTED AT BOTH POSITION 18 AND 19 - HIGHLY POTENT ENDOTHELIN ANTAGONISTS WITH NO SELECTIVITY FOR EITHER RECEPTOR SUBTYPE ET(A) OR ET(B), Journal of medicinal chemistry, 36(25), 1993, pp. 4087-4093