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Citation: Wt. Ashton et al., Orally bioavailable, indole-based nonpeptide GnRH receptor antagonists with high potency and functional activity, BIOORG MED, 11(19), 2001, pp. 2597-2602

Authors: Ashton, WT Sisco, RM Yang, YT Lo, JL Yudkovitz, JB Cheng, K Goulet, MT

Citation: Wt. Ashton et al., Substituted indole-5-carboxamides and -acetamides as potent nonpeptide GnRH receptor antagonists, BIOORG MED, 11(13), 2001, pp. 1723-1726

Authors: Ashton, WT Sisco, RM Yang, YT Lo, JL Yudkovitz, JB Gibbons, PH Mount, GR Ren, RN Butler, BS Cheng, K Goulet, MT

Citation: Wt. Ashton et al., Potent nonpeptide GnRH receptor antagonists derived from substituted indole-5-carboxamides and -acetamides bearing a pyridine side-chain terminus, BIOORG MED, 11(13), 2001, pp. 1727-1731

Authors: DeVita, RJ Walsh, TF Young, JR Jiang, JL Ujjainwalla, F Toupence, RB Parikh, M Huang, SX Fair, JA Goulet, MT Wyvratt, MJ Lo, JL Ren, N Yudkovitz, JB Yang, YT Cheng, K Cui, JS Mount, G Rohrer, SP Schaeffer, JM Rhodes, L Drisko, JE McGowan, E MacIntyre, DE Vincent, S Carlin, JR Cameron, J Smith, RG

Citation: Rj. Devita et al., A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptor, J MED CHEM, 44(6), 2001, pp. 917-922

Authors: Walsh, TF Toupence, RB Young, JR Huang, SX Ujjainwalla, F DeVita, RJ Goulet, MT Wyvratt, MJ Fisher, MH Lo, JL Ren, N Yudkovitz, JB Yang, YT Cheng, K Smith, RG

Citation: Tf. Walsh et al., Potent antagonists of gonadotropin releasing hormone receptors derived from quinolone-6-carboxamides, BIOORG MED, 10(5), 2000, pp. 443-447

Authors: Young, JR Huang, SX Chen, I Walsh, TF DeVita, RJ Wyvratt, MJ Goulet, MT Ren, N Lo, J Yang, YT Yudkovitz, JB Cheng, K Smith, RG

Citation: Jr. Young et al., Quinolones as gonadotropin releasing hormone (GnRH) antagonists: Simultaneous optimization of the C(3)-aryl and C(6)-substituents, BIOORG MED, 10(15), 2000, pp. 1723-1727