THE AZIRIDINATION OF N-TOSYLIMINES WITH AMIDE-STABILIZED SULFONIUM YLIDES - A SIMPLE AND EFFICIENT PREPARATION OF AZIRIDINYL CARBOXAMIDES

Authors
ZHOU YG LI AH HOU XL DAI LX
Citation
Yg. Zhou et al., THE AZIRIDINATION OF N-TOSYLIMINES WITH AMIDE-STABILIZED SULFONIUM YLIDES - A SIMPLE AND EFFICIENT PREPARATION OF AZIRIDINYL CARBOXAMIDES, Tetrahedron letters, 38(41), 1997, pp. 7225-7228
Citations number
17
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
38
Issue
41
Year of publication
1997
Pages
7225 - 7228
Database
ISI
SICI code
0040-4039(1997)38:41<7225:TAONWA>2.0.ZU;2-W
Abstract
Reaction of N-sulfonylimines 2 with N,N-dialkylcarbamoylmethyl dimethy lsulfonium bromides 3 in the presence of solid KOH gives the aziridiny l carboxamides 4 in good to excellent yields. (C) 1997 Elsevier Scienc e Ltd.