Ce. Neipp et al., DIENOPHILICITY OF IMIDAZOLE IN INVERSE ELECTRON DEMAND DIELS-ALDER REACTIONS - INTRAMOLECULAR REACTIONS WITH 1,2,4-TRIAZINES, Tetrahedron letters, 38(43), 1997, pp. 7499-7502
Imidazole and a-phenylimidazole undergo intramolecular cycloadditions
with 1,2,4-triazines tethered between an imidazole nitrogen and the tr
iazinyl C3 position with a trimethylene chain to produce tetrahydro-1,
5-naphthyridines following loss of N-2 and a nitrile. (C) 1997 Elsevie
r Science Ltd.