Dk. Mohapatra et A. Datta, EFFICIENT SYNTHESIS OF BIOLOGICALLY IMPORTANT CHIRAL 2-ALKYLAMINO BENZOXAZINONES, Bioorganic & medicinal chemistry letters, 7(19), 1997, pp. 2527-2530
A novel general method has been developed for the synthesis of various
amino acid derived chiral 2-substituted benzoxazinones, known inhibit
ors of standard serine proteases of the chymotrypsin superfamily. (C)
1997 Elsevier Science Ltd.