SELENIUM-DIRECTED CONJUGATE ADDITION OF AMINES TO DIMETHYL 2-PHENYLSELENO FUMARATE - REGIO AND DIASTEREOSELECTIVE SYNTHESIS OF 2-PHENYLSELENO-3-AMINO SUCCINATES

Citation
M. Bella et al., SELENIUM-DIRECTED CONJUGATE ADDITION OF AMINES TO DIMETHYL 2-PHENYLSELENO FUMARATE - REGIO AND DIASTEREOSELECTIVE SYNTHESIS OF 2-PHENYLSELENO-3-AMINO SUCCINATES, Tetrahedron letters, 38(45), 1997, pp. 7917-7918
Citations number
17
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
ISSN journal
00404039
Volume
38
Issue
45
Year of publication
1997
Pages
7917 - 7918
Database
ISI
SICI code
0040-4039(1997)38:45<7917:SCAOAT>2.0.ZU;2-M
Abstract
Dimethyl 2-phenylseleno fumarate 1 acts as a strong Michael acceptor o f amines, providing the corresponding 2-phenylseleno-3-amino succinate s 2a and 2b in very high yields with complete regio-and good diastereo selectivity. (C) 1997 Elsevier Science Ltd.