Y. Hitotsuyanagi et al., A FACILE SYNTHESIS OF THE 4-AZA-ANALOGS OF 1-ARYLNAPHTHALENE LIGNANS - CHINENSIN, JUSTICIDIN-B, AND TAIWANIN-C, Tetrahedron letters, 38(48), 1997, pp. 8295-8296
Reaction of anilines 1a-d with tetronic acid (2) or 1,3-cyclopentanedi
one (3) produced anilinolactones 4a-d and anilinocyclopentenone 5a, re
spectively, which were then condensed with benzaldehydes to yield 4-az
a-1-arylnaphthalene lignan analogs 6-19. (C) 1997 Elsevier Science Ltd
.