SYNTHESIS OF CONFORMATIONALLY-CONSTRAINED ANALOGS OF GLUTAMIC-ACID ASSTRUCTURAL PROBES OF GLUTAMATERGIC RECEPTORS

Authors
TELLIER F ACHER F BRABET I PIN JP BOCKAERT J AZERAD R
Citation
F. Tellier et al., SYNTHESIS OF CONFORMATIONALLY-CONSTRAINED ANALOGS OF GLUTAMIC-ACID ASSTRUCTURAL PROBES OF GLUTAMATERGIC RECEPTORS, Comptes rendus de l'Academie des sciences. Serie II. Mecanique, physique, chimie, astronomie, 321(9), 1995, pp. 385-392
Citations number
26
Categorie Soggetti
Multidisciplinary Sciences
Journal title
Comptes rendus de l'Academie des sciences. Serie II. Mecanique, physique, chimie, astronomie → ACNP
ISSN journal
12518069
Volume
321
Issue
9
Year of publication
1995
Pages
385 - 392
Database
ISI
SICI code
1251-8069(1995)321:9<385:SOCAOG>2.0.ZU;2-T
Abstract
Norbornane-derived rigid analogs mimicking different potential conform ations of ACPD (1-amino-cyclopentane-1,3-dicarboxylic acid) and glutam ic acid have been synthesized, via the hydantoin route, to be used as conformational probes for bioactive conformations at the glutamatergic receptors of the central nervous system.