A CONVENIENT SYNTHESIS OF 1,2-DIHYDRO-3H-INDOL-3-ONES AND 1,2-DIHYDRO-2H-INDOL-2-ONES BY BAEYER-VILLIGER OXIDATION

Authors
BOURLOT AS DESARBRE E MEROUR JY
Citation
As. Bourlot et al., A CONVENIENT SYNTHESIS OF 1,2-DIHYDRO-3H-INDOL-3-ONES AND 1,2-DIHYDRO-2H-INDOL-2-ONES BY BAEYER-VILLIGER OXIDATION, Synthesis, (4), 1994, pp. 411-416
Citations number
44
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synthesis → ACNP
ISSN journal
00397881
Issue
4
Year of publication
1994
Pages
411 - 416
Database
ISI
SICI code
0039-7881(1994):4<411:ACSO1A>2.0.ZU;2-2
Abstract
The Baeyer-Villiger rearrangement of substituted 1H-indole-3-carbaldeh ydes afforded the corresponding substituted 1,2-dihydro-3H-indol-3-one s. The influence of 3-carbony1 and 1-protecting groups has been examin ed. Reaction has been extended to 1H-indole-2-carbaldehydes and used f or synthesis of 1-(phenylsulfonyl)-1H-indol-2-yl trifluoromethanesulfo nate.