Lds. Yadav et Ds. Yadav, CONVENIENT SYNTHESIS OF YRANOSYL)TETRAHYDRO-2-THIOXO-4H-1,3-THIAZIN-4-ONES OR YRANOSYL)TETRAHYDRO-2-THIOXO-4H-1,3-THIAZIN-4-ONES, Liebigs Annalen, (12), 1995, pp. 2231-2233
Michael addition of the sulfur nucleophiles N-(beta-D-galacto- or -bet
a-D-glucopyranosyl)dithiocarbamic acid (2a, b) to 4-arylidene-5-oxazol
ones (3a-d) followed by ring transformation of the resultant Michael a
dducts 4a-h and hydrolysis yielded new 5-amino-6-aryl-3-(beta-D-galact
o- or ranosyl)-tetrahydro-2-thioxo-4H-1,3-thiazin-4-ones 6a-h in a one
-pot procedure.