Ac. Gillard et al., THIAZOLO[4,3-C][1,4]BENZODIAZEPINES .1. SYNTHESIS OF AMIDINE DERIVATIVES, Journal of heterocyclic chemistry, 32(6), 1995, pp. 1741-1745
Reactivity of thiazolo[4,3-c][1,4]benzodiazepin-5-one-11-thione, and H
-thiazolo[4,3-c][1,4]benzodiazepine-5,11-dithione was evaluated agains
t various amines. The synthetic pathways involved in these reactions w
hich led to new thiazolo[4,3-c][1,4]benzodiazepine amidines are descri
bed.