REACTION OF N-ARYLCITRACONISOIMIDIUM PERCHLORATES WITH AROMATIC-HYDROCARBONS UNDER FRIEDEL-CRAFTS CONDITIONS, A NEW AND CONVENIENT ONE-STEPMETHOD FOR THE SYNTHESIS OF BETA-AROYL-ALPHA-ARYL-N-ARYLBUTYRAMIDES

Authors
ISMAIL MF SAYED FS DERBALA HAY MANSOUR MM
Citation
Mf. Ismail et al., REACTION OF N-ARYLCITRACONISOIMIDIUM PERCHLORATES WITH AROMATIC-HYDROCARBONS UNDER FRIEDEL-CRAFTS CONDITIONS, A NEW AND CONVENIENT ONE-STEPMETHOD FOR THE SYNTHESIS OF BETA-AROYL-ALPHA-ARYL-N-ARYLBUTYRAMIDES, Synthetic communications, 26(6), 1996, pp. 1223-1231
Citations number
8
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synthetic communications → ACNP
ISSN journal
00397911
Volume
26
Issue
6
Year of publication
1996
Pages
1223 - 1231
Database
ISI
SICI code
0039-7911(1996)26:6<1223:RONPWA>2.0.ZU;2-L
Abstract
A number of beta-Aroyl-alpha-aryl-N-arylbutyramides (<4(a)under bar>-( h) under bar) have been synthesized using a new methodology involving arylation at the alpha,beta-unsaturated ketonic systems of N-aryl-citr aconisoimidium perchlorates (<2(a)under bar>-(c) under bar), followed by a subsequent ring opening via addition on the carbonyl group to giv e the title compounds (<4(a)under bar>-(h) under bar).