SYNTHESIS OF 7-INDOLYL-IMINES BY THE REACTION OF 4,6-DIMETHOXYINDOLESWITH SECONDARY AMIDES AND PHOSPHORYL CHLORIDE

Authors
BLACK DS BOWYER MC IVORY AJ JOLLIFFE KA KUMAR N
Citation
Ds. Black et al., SYNTHESIS OF 7-INDOLYL-IMINES BY THE REACTION OF 4,6-DIMETHOXYINDOLESWITH SECONDARY AMIDES AND PHOSPHORYL CHLORIDE, Tetrahedron, 52(13), 1996, pp. 4687-4696
Citations number
28
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron → ACNP
ISSN journal
00404020
Volume
52
Issue
13
Year of publication
1996
Pages
4687 - 4696
Database
ISI
SICI code
0040-4020(1996)52:13<4687:SO7BTR>2.0.ZU;2-U
Abstract
4,6-Dimethoxy-2,3-diphenylindole 1 undergoes reaction with formanilide , acetanilide, benzanilide and several dimethoxy analogs in the presen ce of phosphoryl chloride to give the corresponding 7-imino derivative s 2-6. This reaction has been extended to include the synthesis of 7-i ndolyl-pyrrolines and tetrahydropyridines 7-9, 11 and oxazolines 14,15 .