PRACTICAL SYNTHESES OF FUNCTIONALIZED OXO-1,2,3,4-TETRAHYDRO-BETA-CARBOLINE-3-CARBOXYLIC ACID-ESTERS

Authors
JEANNIN L SAPI J VASSILEVA E RENARD P LARONZE JY
Citation
L. Jeannin et al., PRACTICAL SYNTHESES OF FUNCTIONALIZED OXO-1,2,3,4-TETRAHYDRO-BETA-CARBOLINE-3-CARBOXYLIC ACID-ESTERS, Synthetic communications, 26(9), 1996, pp. 1711-1719
Citations number
9
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synthetic communications → ACNP
ISSN journal
00397911
Volume
26
Issue
9
Year of publication
1996
Pages
1711 - 1719
Database
ISI
SICI code
0039-7911(1996)26:9<1711:PSOFO>2.0.ZU;2-5
Abstract
Three methods have been proposed for the preparation of functionalized o-1,2,3,4-tetrahydro-beta-carboline-3-carboxylates (3) from which the ''acylazide formation-Curtius rearrangement-acid catalyzed ring closu re'' sequence starting from hemi-ester hemi-acids (8) seemed to be qui te general.