THE PREPARATION OF FORSKOLIN ANALOGS VIA QUINONE DIELS-ALDER REACTIONS

Authors
LEVIN JI
Citation
Ji. Levin, THE PREPARATION OF FORSKOLIN ANALOGS VIA QUINONE DIELS-ALDER REACTIONS, Tetrahedron letters, 37(18), 1996, pp. 3079-3082
Citations number
25
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
37
Issue
18
Year of publication
1996
Pages
3079 - 3082
Database
ISI
SICI code
0040-4039(1996)37:18<3079:TPOFAV>2.0.ZU;2-P
Abstract
A practical synthetic route for the preparation of compound 2a, a carb ocyclic analog of the Delta(5)-derivative, 1, of forskolin has been co mpleted. A quinone Diels-Alder reaction is used for the rapid construc tion of the tricyclic framework of 2. Copyright (C) 1996 Elsevier Scie nce Ltd