SYNTHESIS OF 3-ACETYL-2-AMINO-4-PYRIDONE

Citation
Va. Dorokhov et al., SYNTHESIS OF 3-ACETYL-2-AMINO-4-PYRIDONE, Russian chemical bulletin, 45(1), 1996, pp. 168-170
Citations number
10
Categorie Soggetti
Chemistry
Journal title
ISSN journal
10665285
Volume
45
Issue
1
Year of publication
1996
Pages
168 - 170
Database
ISI
SICI code
1066-5285(1996)45:1<168:SO3>2.0.ZU;2-5
Abstract
A method for synthesizing 3-acetyl-2-amino-4-pyridone has been suggest ed. The synthesis involves the condensation of dimethylformamide dimet hylacetal at the NH2 group of diphenylboron chelate diacetylketene ami nal followed by its intramolecular cyclization under the action of NaO Me in MeOH.