Jj. Acton et Ab. Jones, SYNTHESIS AND DERIVATIZATION OF A VERSATILE ALPHA-SUBSTITUTED LACTAM DIPEPTIDE ISOSTERE, Tetrahedron letters, 37(25), 1996, pp. 4319-4322
The diastereoselective synthesis of a versatile lactam constrained dip
eptide isostere is described. The facile derivatization of this interm
ediate is demonstrated. Copyright (C) 1996 Elsevier Science Ltd.