CONFORMATIONALLY RESTRICTED ANALOGS OF TRYPTOPHAN - SYNTHESIS OF CHIRAL 3-AMINO-4-INDOLYL-2-PIPERIDONES

Authors
RODRIGUEZ R VINETS I DIEZ A RUBIRALTA M GIRALT E
Citation
R. Rodriguez et al., CONFORMATIONALLY RESTRICTED ANALOGS OF TRYPTOPHAN - SYNTHESIS OF CHIRAL 3-AMINO-4-INDOLYL-2-PIPERIDONES, Synthetic communications, 26(16), 1996, pp. 3029-3059
Citations number
29
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synthetic communications → ACNP
ISSN journal
00397911
Volume
26
Issue
16
Year of publication
1996
Pages
3029 - 3059
Database
ISI
SICI code
0039-7911(1996)26:16<3029:CRAOT->2.0.ZU;2-L
Abstract
The {Trp-phenylglycinol} pseudodipeptide (alpha toxy-1-phenylethyl)-3- amino-4-indolyl-2-piperidone 33 has been synthezised by condensation o f the 3-amino-substituted anhydride 30 with (R)-(-)-phenylglycinol fol lowed by reduction of the resulting imide.