CATALYTIC REDUCTIVE N-ALKYLATION OF ANILINES - APPLICATION TO THE SYNTHESIS OF N-ARYL AMINO-ACID PRECURSORS

Authors
FACHE F VALOT F MILENKOVIC A LEMAIRE M
Citation
F. Fache et al., CATALYTIC REDUCTIVE N-ALKYLATION OF ANILINES - APPLICATION TO THE SYNTHESIS OF N-ARYL AMINO-ACID PRECURSORS, Tetrahedron, 52(29), 1996, pp. 9777-9784
Citations number
26
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron → ACNP
ISSN journal
00404020
Volume
52
Issue
29
Year of publication
1996
Pages
9777 - 9784
Database
ISI
SICI code
0040-4020(1996)52:29<9777:CRNOA->2.0.ZU;2-G
Abstract
Different anilines have been monoalkylated by reductive alkylation usi ng ketones and alpha-ketoesters as alkylating agents with good isolate d yields. This provided access to aminoacid derivatives. Diastereosele ctive experiments were also performed. Copyright (C) 1996 Elsevier Sci ence Ltd.