Bm. Swahn et al., NEW HETEROARYL-SPACED PHOSPHONO ALPHA-AMINO-ACIDS ARE COMPETITIVE NMDA ANTAGONISTS WITH ANALGESIC ACTIVITY, Bioorganic & medicinal chemistry letters, 6(14), 1996, pp. 1635-1640
The synthesis and the NMDA receptor binding affinities of -amino-3-(ph
osphonomethyl)-2-naphthalene-propanoic acid, ha-amino-3-(phosphonometh
yl)-2-benzofuranpropanoic acid, a series of substituted pha-amino-3-(p
hosphonomethyl)-2-quinolinepropanoic acids, -3-(phosphonomethyl)-1,8-n
aphthyridine-2-propanoic acid and -3-(phosphonomethyl)-1,6-naphthyridi
ne-2-propanoic acid are reported. Copyright (C) 1996 Elsevier Science
Ltd