SYNTHESES OF (S)-BETA-PYRAZOLYLALANINE AND (S)-QUISQUALIC ACID FROM ASERINE-DERIVED AZIRIDINE

Authors
FARTHING CN BALDWIN JE RUSSELL AT SCHOFIELD CJ SPIVEY AC
Citation
Cn. Farthing et al., SYNTHESES OF (S)-BETA-PYRAZOLYLALANINE AND (S)-QUISQUALIC ACID FROM ASERINE-DERIVED AZIRIDINE, Tetrahedron letters, 37(29), 1996, pp. 5225-5226
Citations number
15
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
37
Issue
29
Year of publication
1996
Pages
5225 - 5226
Database
ISI
SICI code
0040-4039(1996)37:29<5225:SO(A(A>2.0.ZU;2-2
Abstract
The naturally occurring amino acids (S)-beta-pyrazolylalanine and (S)- quisqualic acid are synthesised via the nucleophilic ring-openings of an optically active aziridine by pyrazole and 1,2,4-oxadiazolidine-3,5 -dione, respectively. Copyright (C) 1996 Published by Elsevier Science Ltd