1-(PHENYLSULFONYL)INDOL-2-YL TRIFLATE - A VERSATILE REAGENT FOR THE SYNTHESIS OF 2-SUBSTITUTED INDOLES

Authors
JOSEPH B MALAPEL B MEROUR JY
Citation
B. Joseph et al., 1-(PHENYLSULFONYL)INDOL-2-YL TRIFLATE - A VERSATILE REAGENT FOR THE SYNTHESIS OF 2-SUBSTITUTED INDOLES, Synthetic communications, 26(17), 1996, pp. 3289-3295
Citations number
19
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Synthetic communications → ACNP
ISSN journal
00397911
Volume
26
Issue
17
Year of publication
1996
Pages
3289 - 3295
Database
ISI
SICI code
0039-7911(1996)26:17<3289:1T-AVR>2.0.ZU;2-7
Abstract
The palladium-catalysed reaction of 1-(phenyl sulfonyl)indol-2-yl trif late 1 with a variety of aryl and heteroaryl boronic acids 2 or vinyl tributylstannane 3 provides a general and an efficient method for the synthesis of 2-substituted indoles 4.