CONFORMATIONALLY CONSTRAINED DIPEPTIDES - SYNTHESIS OF BICYCLIC LACTAMS BY STEREOSELECTIVE RADICAL CYCLIZATIONS

Citation
L. Colombo et al., CONFORMATIONALLY CONSTRAINED DIPEPTIDES - SYNTHESIS OF BICYCLIC LACTAMS BY STEREOSELECTIVE RADICAL CYCLIZATIONS, Gazzetta chimica italiana, 126(8), 1996, pp. 543-554
Citations number
55
Categorie Soggetti
Chemistry
Journal title
ISSN journal
00165603
Volume
126
Issue
8
Year of publication
1996
Pages
543 - 554
Database
ISI
SICI code
0016-5603(1996)126:8<543:CCD-SO>2.0.ZU;2-4
Abstract
Regio- and stereoselective radical cyclizations of beta-substituted al pha-N-acetyl acrylamides have been performed. 6,5- and 7,5-fused bicyc lic lactams were obtained, which can be viewed as conformationally res tricted dipeptide mimetics.