MICROWAVE-PROMOTED TRANSFORMATIONS - FAST AND CHEMOSELECTIVE N-ACYLATION OF AMINO-ALCOHOLS USING CATALYTIC AMOUNTS OF DIBUTYLTIN OXIDE - INFLUENCE OF THE POWER OUTPUT AND THE NATURE OF THE ACYLATING AGENT ON THE SELECTIVITY
A. Morcuende et al., MICROWAVE-PROMOTED TRANSFORMATIONS - FAST AND CHEMOSELECTIVE N-ACYLATION OF AMINO-ALCOHOLS USING CATALYTIC AMOUNTS OF DIBUTYLTIN OXIDE - INFLUENCE OF THE POWER OUTPUT AND THE NATURE OF THE ACYLATING AGENT ON THE SELECTIVITY, Journal of organic chemistry, 61(16), 1996, pp. 5264-5270
The influence of the nature of the acylating agent and the power outpu
t on the chemoselectivity of the microwave-mediated acylation of 1,2-
and 1,3-amino alcohols catalyzed by dibutyltin oxide has been studied.
The method constitutes an efficient procedure for the selective N-acy
lation of amino alcohols.