T. Pietzonka et al., PHOSPHONATE-CONTAINING ANALOGS OF CHOLESTERYL ESTER AS NOVEL INHIBITORS OF CHOLESTERYL ESTER TRANSFER PROTEIN, Bioorganic & medicinal chemistry letters, 6(16), 1996, pp. 1951-1954
A series of phosphorus-containing analogs of cholesteryl ester have be
en synthesized as potential inhibitors of cholesteryl ester transfer p
rotein (CETP). The most potent inhibitor, phosphonate 7, represents a
novel inhibitor of CETP. Copyright (C) 1996 Elsevier Science Ltd