Vv. Zhdankin et al., 1-AMIDO-3-(1H)-1,2-BENZIODOXOLES - STABLE AMIDOIODANES AND REAGENTS FOR DIRECT AMIDATION OF ORGANIC SUBSTRATES, Tetrahedron letters, 38(1), 1997, pp. 21-24
Amidobenziodoxoles 2 can be prepared from benziodoxole 1, trimethylsil
yltriflate and the appropriate amides in the form of stable, microcrys
talline compounds. Amidobenziodoxoles 2 react with adamantane 3 or N,N
-dimethylarylamines 5 to afford the corresponding products of amidatio
n, 4 and 6. Copyright (C) 1996 Elsevier Science Ltd