SYNTHESIS OF ENANTIOPURE AZA-ANALOGS OF COCAINE

Authors
TEERHUIS NM HIEMSTRA H SPECKAMP WN
Citation
Nm. Teerhuis et al., SYNTHESIS OF ENANTIOPURE AZA-ANALOGS OF COCAINE, Tetrahedron letters, 38(1), 1997, pp. 159-162
Citations number
17
Categorie Soggetti
Chemistry Inorganic & Nuclear
Journal title
Tetrahedron letters → ACNP
ISSN journal
00404039
Volume
38
Issue
1
Year of publication
1997
Pages
159 - 162
Database
ISI
SICI code
0040-4039(1997)38:1<159:SOEAOC>2.0.ZU;2-M
Abstract
An enantiopure aza-analogue of pseudo-cocaine was synthesized starting from a 5-substituted 3-pyrazolidinone by using an N-acylhydrazonium i on cyclization with a dioxenone nucleophile as the key step. Copyright (C) 1996 Elsevier Science Ltd